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8-(furan-3-carbonyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
2-[1-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-1H-1,2,3-triazol-4-yl]benzoic acid
2-(2-hydroxyethyl)-9-{[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(hexahydro-1H-pyrrolizin-7a-yl)ethyl]-4-(piperidin-3-ylmethyl)benzamide
N-(1H-1,2,3,4-tetrazol-5-ylmethyl)-5-{3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}pyridin-2-amine
2-ethyl-4-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]-1-(propan-2-yl)piperazine
3-(piperidin-1-ylmethyl)-1-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperidine
2-[2-(7-fluoro-2-methyl-1H-indol-3-yl)acetyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
(2R,3R)-3-[ethyl(methyl)amino]-1'-(3-methylpyridine-2-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
(2-ethoxy-5-{[(propan-2-yl)[(trimethyl-1H-pyrazol-4-yl)methyl]amino]methyl}phenyl)methanol
methyl 4-{[(2-benzyl-1,3-benzoxazol-5-yl)formamido]methyl}benzoate
3-chloro-6-methyl-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}pyrazolo[1,5-a]pyrimidine-2-carboxamide
(1S,5R)-3-(isoquinolin-1-yl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-[(4-methylphenyl)methyl]piperidine
N-[2-(1H-imidazol-4-yl)ethyl]-2-(trimethyl-1H-pyrazol-1-yl)acetamide
N,1-dimethyl-N-[2-(methylsulfanyl)ethyl]-5-phenyl-1H-pyrrole-2-carboxamide
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}acetamide
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
(3R,4S)-4-cyclopropyl-1-(5,6,7,8-tetrahydroquinolin-2-yl)pyrrolidin-3-amine
3-(1-methyl-1H-imidazole-2-carbonyl)-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperidine
1-(2-ethoxyethyl)-N-ethyl-N-[(2-methylphenyl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
3-{4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}phenol
(1S,5R)-6-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-(4-{[(3R,4S)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]methyl}phenoxy)ethan-1-ol
(1R,3R,5S)-3-(4-methoxyphenyl)-8-(1H-pyrrole-2-carbonyl)-8-azabicyclo[3.2.1]octane
1-(1-{1-[(4-chlorophenyl)methyl]piperidin-4-yl}ethyl)-4-methylpiperazine
1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-[(3-methylpyridin-2-yl)methyl]piperazine
N-[(4,6-dimethylpyridin-3-yl)methyl]-3-[(2-fluoroethyl)sulfamoyl]benzamide
N-{4-[2-(2-methoxyethyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carbonyl]phenyl}acetamide
(3R,4R)-1-[4-(2-methoxyphenyl)benzoyl]-3,4-dimethylpyrrolidin-3-ol
N-(3-chloro-4-propanamidophenyl)-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carboxamide
2-[3-({[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)-1H-indol-1-yl]acetamide
2-(3-acetyl-1H-pyrazol-1-yl)-N-[1-(cyclopropylmethyl)-1H-indazol-3-yl]acetamide
2-(1-{pyrazolo[1,5-a]pyridine-7-carbonyl}pyrrolidin-2-yl)-1,3-thiazole
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-(3-methoxyphenoxymethyl)-1,3-oxazole-4-carboxamide
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)thiophene-3-carboxamide
N-{[(2S,4S)-4-fluoro-1-(1-methyl-1H-pyrrole-2-carbonyl)pyrrolidin-2-yl]methyl}-1-phenylmethanesulfonamide
1-ethyl-N-(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)-6-oxopiperidine-3-carboxamide
1-[(3-fluorophenyl)methyl]-4-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}piperazin-2-one
3-{[(4-fluorophenyl)methyl]amino}-N-[1-(1H-1,2,4-triazol-5-yl)ethyl]benzamide
N-[1-(2,5-dimethoxyphenyl)ethyl]-4-hydroxy-2-(pyridin-2-yl)pyrimidine-5-carboxamide
1-[2-(2-cyclopentylacetamido)ethyl]-N-[1-(thiophen-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-[2-(dimethylamino)ethyl]-8-methoxy-3,4-dihydroquinazolin-4-one
4-[5-(2-methyloxolan-2-yl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-3-yl]benzamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2-(piperidin-1-yl)acetamide
1'-[4-(1H-pyrazol-3-yl)benzoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
ethyl 3-({1-[2-(3-fluorophenyl)ethyl]-6-oxopiperidin-3-yl}formamido)propanoate
1-[2-(1H-imidazol-5-yl)ethyl]-3-(oxan-4-yl)-5-(1H-pyrazol-1-ylmethyl)-1H-1,2,4-triazole
(4aS,7aR)-1-[(3,5-dimethylphenyl)methyl]-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-methyl-4-phenyl-3-(2-phenylpyrrolidine-1-carbonyl)pyridine