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1,3-dimethyl-5-{[2-(2-methyl-1,3-oxazol-4-yl)-1H-imidazol-1-yl]methyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
4-(3-hydroxy-3-methylbutyl)-N-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]benzamide
N-(1-{4-[2-(3-methoxyphenoxy)ethyl]phenyl}ethyl)acetamide
benzyl({[3-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-1,2-oxazol-5-yl]methyl})methylamine
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-4-methyl-1,3-oxazole-5-carboxamide
3-[ethyl({2-phenylimidazo[1,2-a]pyridin-3-yl}methyl)amino]-1λ6-thiolane-1,1-dione
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-N-(2,3-dihydro-1H-inden-2-yl)acetamide
3-(1H-indol-3-yl)-1-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]propan-1-one
6-{4-[(4-tert-butylphenyl)methyl]piperazin-1-yl}pyrimidine-2,4-diamine
1-(oxan-4-yl)-4-{2-[4-(trifluoromethyl)phenyl]-1H-imidazol-1-yl}piperidine
3-[(3S,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,4-dichlorophenyl)urea
{[4-ethoxy-3-(prop-2-en-1-yl)phenyl]methyl}(1H-imidazol-2-ylmethyl)amine
1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-3-(propoxymethyl)pyrrolidine
N-(2-methoxyethyl)-5-methyl-N-(1,3-thiazol-2-ylmethyl)-1,2-oxazole-4-carboxamide
3-{[(2-hydroxyethyl)(propan-2-yl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
1-ethyl-N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}-2-oxo-1,2-dihydropyridine-4-carboxamide
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N,N-bis(prop-2-en-1-yl)acetamide
1-[1-methyl-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidine-3-carboxamide
(2R,3S,6R)-3-(2-methoxyphenyl)-5-(5-methylpyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(1-tert-butyl-1H-pyrazol-4-yl)-7-fluoro-N,N-dimethylquinoline-4-carboxamide
N-(2-methoxyethyl)-1-methyl-5-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-1H-1,3-benzodiazol-2-amine
1'-(1,3-thiazol-2-ylmethyl)-1,2-dihydrospiro[indole-3,4'-piperidine]
2-methyl-4-{4-[(1s,5s)-7,10-dimethyl-3,7,10-triazatricyclo[3.3.3.01,5]undecane-3-carbonyl]phenyl}butan-2-ol
2-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]benzonitrile
(1S,5R)-6-[2-(benzenesulfonyl)ethyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[2-(propane-2-sulfonyl)ethyl]piperidin-2-one
6-amino-N-({1-[(3,4-dimethylphenyl)methyl]pyrrolidin-3-yl}methyl)pyridine-3-carboxamide
N-{2-[ethyl(3-methylphenyl)amino]ethyl}-7-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide
6-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
1-(5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-yl)azetidin-3-ol
2-[5-oxo-4-(2-phenylethyl)-3-(thiophen-3-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]acetamide
4-fluoro-N-{[4-(2-methylpropoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)benzamide
(3S,4S)-1-[2-(4-chloro-3-methyl-1H-pyrazol-1-yl)acetyl]-4-cyclopropylpyrrolidine-3-carboxylic acid
9-[2-(morpholin-2-yl)acetyl]-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
1'-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
3-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)-5,6,7,8-tetrahydronaphthalen-2-ol
3-({9-hydroxy-4-oxo-4H-pyrido[1,2-a]pyrimidin-3-yl}formamido)-N-phenylpropanamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[2-(2-fluorophenyl)acetyl]pyrrolidine-3-carboxylic acid
9-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-1-oxa-9-azaspiro[5.5]undecan-5-ol
3-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-1-methyl-4,5,6,7-tetrahydro-1H-indazole
4-[(2-amino-6-methylpyrimidin-4-yl)amino]-1-[(4-fluorophenyl)methyl]pyrrolidin-2-one
methyl 6-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]pyrimidine-4-carboxylate
1-(cyclopropylmethyl)-4-(pyridin-3-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-(furan-2-yl)-1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]pyrrolidine
1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-4-(4H-1,2,4-triazol-3-yl)piperidine
N-(4-chloro-2-methylphenyl)-2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-1-carboxamide
2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-N-[5-(oxolan-2-yl)-1,3,4-thiadiazol-2-yl]acetamide
6-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)pyridine-3-carboxylic acid
3-(3-{2-methyl-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}-3-oxopropyl)-3,4-dihydroquinazolin-4-one
1-amino-N-({1-[(4-methoxy-2-methylphenyl)methyl]piperidin-3-yl}methyl)cyclobutane-1-carboxamide