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ethyl 4-{6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}-3,5-dimethyl-1H-pyrrole-2-carboxylate
4-phenyl-3-(piperidin-3-yl)-1-(pyridin-2-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
9-[3-(dimethylamino)benzoyl]-4-methyl-1-oxa-4,9-diazaspiro[5.5]undecan-3-one
(3S,7S)-5-(dimethyl-1,2-oxazole-4-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
N-[2-(1H-imidazol-4-yl)ethyl]-8-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-methyl-4-(propan-2-yl)-6-{4-[4-(pyrazin-2-yl)piperazin-1-yl]piperidin-1-yl}pyrimidine
1-(carbamoylmethyl)-N-[2-(7-methyl-1H-indol-3-yl)ethyl]piperidine-3-carboxamide
methyl 4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
1-{1-[(methylcarbamoyl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
1-[6-(piperazin-1-yl)pyridine-3-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane
(2,1,3-benzothiadiazol-5-ylmethyl)(methyl){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
3-(2-amino-1,3-thiazol-4-yl)-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
6-oxo-N-[2-(1H-pyrazol-4-yl)ethyl]-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
1-(1-ethyl-1H-pyrazole-3-carbonyl)-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
2-[({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)amino]-4,6-dimethylpyridine-3-carbonitrile
4-chloro-N-{[1-(4-methylpiperazin-1-yl)cyclopentyl]methyl}-1H-indole-2-carboxamide
2-[1-(2-methylpropyl)-4-[6-(propan-2-yl)-2-(trifluoromethyl)pyrimidin-4-yl]piperazin-2-yl]ethan-1-ol
3-oxo-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]-3,4-dihydro-2H-1,4-benzoxazine-6-sulfonamide
4-{[(cyclopropylcarbamoyl)methyl]sulfamoyl}-N-(2-methoxyethyl)benzamide
N-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
2-[(dimethylamino)methyl]-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]-1,3-thiazole-4-carboxamide
3-[1-(2-ethylpyrimidine-5-carbonyl)piperidin-4-yl]-1,3-oxazolidin-2-one
N-[(3S,4R)-1-(2-ethoxyacetyl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
4-[7-(1-carbamoylcyclopropanecarbonyl)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl]benzamide
1-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-3-(dimethyl-1H-1,2,4-triazol-3-yl)urea
N-{[4-(dimethylamino)oxan-4-yl]methyl}-5-ethylpyrimidin-2-amine
2-cyclopropyl-8-[(2-fluoro-4-methylphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
7-[(4-fluorophenyl)methyl]-2-(3-methylfuran-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-(2-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-5-methylphenyl)-1H-pyrazole
N-cyclopropyl-1-[4-(pyrrolidin-1-ylmethyl)benzoyl]piperazine-2-carboxamide
5-ethyl-5-{1-[(8-hydroxyquinolin-2-yl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-(1H-imidazol-4-ylmethyl)piperidine
2-{2-[2-(4-methoxy-2,3-dimethylphenyl)-1H-imidazol-1-yl]ethyl}-3-methylpyridine
N-[(1S,2R)-1-hydroxy-1-(4-hydroxyphenyl)propan-2-yl]-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-{[(pyridin-2-ylmethyl)amino]methyl}piperidin-2-one
2-[2-(1H-imidazol-4-yl)ethyl]-8-(2-methylfuran-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(1,3-benzoxazol-2-yl)-4-(4-chlorophenoxy)piperidine-4-carboxylic acid
3-(azepane-1-carbonyl)-1-(2-methylpropyl)-5-(3-phenylpiperidine-1-carbonyl)-1,4-dihydropyridin-4-one
6-fluoro-N-{2-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}-1H-1,3-benzodiazole-2-carboxamide
(1S,5R)-6-(cyclopropylmethyl)-3-{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
1-(dimethylamino)-3-(4-{[4-(2-methylpyrimidin-4-yl)piperidin-1-yl]methyl}phenoxy)propan-2-ol
N-[(1-cyclopropanecarbonylpiperidin-3-yl)methyl]-4-hydroxy-2-(4-methylphenyl)pyrimidine-5-carboxamide
1-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]-3-[4-(3-methylphenyl)piperazin-1-yl]propan-1-one
1-(3-{[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]methyl}phenyl)ethan-1-one
6-ethyl-N-[2-hydroxy-2-(pyridin-3-yl)ethyl]-2-methylquinoline-4-carboxamide
2-(3-methoxyphenyl)-N-(2,2,2-trifluoroethyl)-1,3-benzoxazole-6-carboxamide
N,N-dimethyl-2-[(1S,5R)-3-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
(4aR,7aS)-1-(cyclopropylmethyl)-4-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-ethyl-N-(2-methylprop-2-en-1-yl)acetamide