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3-benzoyl-1-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]piperidine
4-(azepane-1-carbonyl)-N-(1H-imidazol-2-ylmethyl)benzene-1-sulfonamide
2-[(4-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}phenyl)sulfanyl]ethan-1-ol
N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-3-(pyridin-3-yl)propanamide
2-[(5-chlorothiophen-2-yl)methyl]-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
3-[3-cyclopropyl-5-(2-ethyl-4-methyl-1,3-oxazol-5-yl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
1-(6-hydroxy-4-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-1,4-diazepan-1-yl)ethan-1-one
3-methyl-8-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-{3-[3-(4-fluorophenyl)pyrrolidin-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(3,4-dimethoxyphenyl)methyl]-2-ethyl-N-(pyridin-3-ylmethyl)butanamide
(1S,5R)-6-(cyclobutylmethyl)-3-[1-(pyridine-3-carbonyl)piperidin-4-yl]-3,6-diazabicyclo[3.2.2]nonan-7-one
benzyl N-{1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl}carbamate
N3-methyl-4-oxo-1-(2-phenylethyl)-N5-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-5-ylmethyl}-1,4-dihydropyridine-3,5-dicarboxamide
4-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-5,6-dimethylpyrimidine
(1S,5R)-6-[(4-methanesulfonylphenyl)methyl]-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
4-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]-2-methoxypyridine
5-[4-(3,4,5-trimethoxyphenyl)phenyl]-1,3-oxazole
ethyl 4-benzyl-1-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]piperidine-4-carboxylate
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-2-(3-oxo-3,4-dihydro-2H-1,4-benzothiazin-4-yl)acetamide
3-(2-fluoro-5-methoxyphenyl)-5-(pyrrolidine-1-sulfonyl)benzoic acid
1-(furan-3-carbonyl)-4-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-1,4-diazepane
N-[2-(1H-indol-3-yl)ethyl]-N'-[2-(propan-2-yl)phenyl]butanediamide
2-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-4-{4-[(2-fluorophenyl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
3-(2H-1,3-benzodioxol-5-yl)-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
1-(1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
methyl 5-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-5-oxopentanoate
3-ethyl-1-(3-fluoropyridin-4-yl)piperidine-3-carboxylic acid
N-[2-(1H-imidazol-4-yl)ethyl]-2-methyl-5-propylpyrimidin-4-amine
2-(2-ethyl-4-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]acetamide
1-(2,3-dihydro-1H-inden-2-yl)-4-[(3-fluorophenyl)methyl]-1,4-diazepan-5-one
1-(1-methylpiperidin-4-yl)-3-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}piperidine
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(6-methylpyrimidin-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
{2-[2-(methylsulfanyl)pyrimidin-4-yl]phenyl}methanol
N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-5-propyl-1,2-oxazole-3-carboxamide
1-methyl-5-[4-(2-phenylethyl)piperazine-1-carbonyl]-1H-1,3-benzodiazole
1-methyl-5-[2-(2-methylphenyl)benzoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-{3-[3-(4-fluorophenyl)oxolan-3-yl]-1,2,4-oxadiazol-5-yl}benzonitrile
4-{3-[3-(methoxymethyl)pyrrolidine-1-carbonyl]benzenesulfonyl}thiomorpholine
1-tert-butyl-5-oxo-N-[2-(pyridin-3-yl)ethyl]pyrrolidine-3-carboxamide
ethyl 1-(1-acetylpiperidin-4-yl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
2-{1-[(3,4-difluorophenyl)methyl]-4-(6-methylpyridazin-3-yl)piperazin-2-yl}ethan-1-ol
[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl](methyl){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
9-(cyclopropylmethyl)-1-methyl-4-[(2-methyl-1,3-oxazol-4-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-[(2-methoxyphenyl)methyl]-1-[(3-methylphenyl)methyl]pyrrolidine-2-carboxamide
N-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]cyclopentanecarboxamide
N-(1,3-benzoxazol-2-ylmethyl)-N-methyl-5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
1-[(4-chlorophenyl)methyl]-N-[(2S)-1-hydroxy-4-(methylsulfanyl)butan-2-yl]-1H-1,2,3-triazole-4-carboxamide
3-[(3,4-dimethylphenyl)amino]-N-(prop-2-en-1-yl)piperidine-1-carboxamide
2-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-5,6,7,8-tetrahydroquinoline
2-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1H-indole