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1-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
5-tert-butyl-3-{[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1,2,4-oxadiazole
3-amino-N-(2-phenylethyl)-N-(propan-2-yl)-1H-1,2,4-triazole-5-carboxamide
3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]-1-[2-(2-oxopyrrolidin-1-yl)ethyl]urea
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl][2-(2-fluorophenyl)-1-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}ethyl]methylamine
4-[(dimethylamino)methyl]-1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}azepan-4-ol
{2-[4-(1-tert-butyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]ethyl}urea
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-2-(1H-1,2,3-triazol-1-yl)ethan-1-one
4-({2-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
(2S,4R)-N,N-diethyl-1-methyl-4-[4-(pyrrolidin-1-yl)benzamido]pyrrolidine-2-carboxamide
5-[4-(2-methylpropyl)phenyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-(azocan-1-yl)-3-(5-{[(cyclopropylmethyl)amino]methyl}-2-methoxyphenoxy)propan-2-ol
N-butyl-N-ethyl-3,6-dimethyl-2-(pyrimidin-5-yl)quinoline-4-carboxamide
4-{2-[3-(1H-pyrazol-3-yl)phenyl]pyridine-4-carbonyl}morpholine
N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
2-cyclopropyl-5-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine-1-carbonyl)pyrimidin-4-ol
6-methyl-2-(3-methyl-3-phenylpiperidin-1-yl)pyridine-3-carboxylic acid
1-[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-ethyl-N-[2-(2-fluorophenoxy)ethyl]-2-methylpyridine-3-carboxamide
3-methoxy-2-[3-(1H-pyrazol-3-yl)phenyl]pyridine
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
3-(2-amino-1,3-thiazol-4-yl)-1-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]propan-1-one
(1S,5R)-6-benzyl-3-[(2,6-difluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
dimethyl(2-{[(3-methylthiophen-2-yl)methyl]({[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl})amino}ethyl)amine
8-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-2,3,4,9-tetrahydro-1H-carbazole
5-(ethylsulfanyl)-N-(2-oxo-2,3-dihydro-1H-indol-5-yl)thiophene-2-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(3-fluorophenyl)-1,3-benzoxazole-5-carboxamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(1H-imidazol-4-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-(hydroxymethyl)-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)benzamide
5-{[2-(3-fluorophenyl)ethyl]amino}-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-[4-(quinazolin-4-yl)piperazine-1-carbonyl]-3,4-dihydroquinazolin-4-one
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-1,2-oxazole-3-carboxamide
4-(2-ethoxypyridine-3-carbonyl)-2-(4-methylpentyl)morpholine
2-[1-(2-phenylethyl)-4-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperazin-2-yl]ethan-1-ol
2-methyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1,3-thiazole-4-carboxamide
2-[3-(2-methylpropoxy)phenyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(1H-imidazol-4-yl)propan-1-one
3-(4-methoxyphenyl)-1-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]propan-1-one
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-[(4-methyl-1H-imidazol-5-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
3-methoxy-1-(7-{[2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
6-amino-N-({1-[(3-ethyl-1,2-oxazol-5-yl)methyl]pyrrolidin-3-yl}methyl)pyridine-3-carboxamide
N2-cyclopropyl-N4-[(1-methyl-1H-pyrazol-4-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
4-(cyclopropylmethyl)-N-(4-methylphenyl)-5-oxo-3-(propan-2-yl)-1,4-diazepane-1-carboxamide
1-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-4-(4-methyl-1,2,5-oxadiazol-3-yl)piperazine
N,N-dimethyl-2-{[(2-methyl-6-propylpyrimidin-4-yl)amino]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
[3-(prop-2-en-1-yl)-1-[4-(pyrrolidin-1-yl)benzoyl]piperidin-3-yl]methanol
N-[(3,4-dimethylphenyl)methyl]-8-methyl-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
7-(5-chloropyridin-2-yl)-4-(oxane-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol