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[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl](methyl)[2-(2-methyl-1H-imidazol-1-yl)ethyl]amine
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-cyclopropyl-N-(pyridin-2-ylmethyl)-1H-pyrazole-3-carboxamide
4-{4-[1-(4-fluorophenyl)cyclopropanecarbonyl]-5-methyl-2-oxopiperazin-1-yl}benzonitrile
N-[(1-ethyl-1H-indazol-3-yl)methyl]-2,3-dimethylquinoxaline-6-carboxamide
6,8-dimethyl-3-({methyl[1-(4-methylpyridin-2-yl)propan-2-yl]amino}methyl)-1,2-dihydroquinolin-2-one
3-tert-butyl-1-[4-(5-sulfamoylthiophen-2-yl)phenyl]urea
(4aR,8aR)-2-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-7-methanesulfonyl-decahydro-2,7-naphthyridin-4a-ol
ethyl 5-({[1-(4-{[2-(morpholin-4-yl)ethyl]carbamoyl}phenyl)piperidin-4-yl]amino}methyl)furan-2-carboxylate
{[(3S,4R)-1-[(2-chlorophenyl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2,3-dihydro-1H-indene-1-carboxamide
4-{[4-(2-phenoxyethyl)piperazin-1-yl]methyl}-2,1,3-benzoxadiazole
2-propyl-8-[4-(1H-1,2,3,4-tetrazol-1-yl)butanoyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
[(3R,4S)-1-[(2,3-difluoro-4-methylphenyl)methyl]-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
6-{3-[(4-tert-butyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}quinoxaline
4-[(5-acetylthiophen-3-yl)methyl]-3-(3-fluorophenyl)piperazin-2-one
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-[1-(3-ethyl-1,2-oxazol-5-yl)ethyl]acetamide
2-[(1S,5R)-6-(2H-1,3-benzodioxol-5-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
7-[(1-phenylethyl)sulfamoyl]-N-propyl-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
1-ethyl-N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}piperidin-4-amine
1-[(3-fluorophenyl)methyl]-4-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}-1,4-diazepane
1-({1-[(2-aminopyrimidin-5-yl)methyl]pyrrolidin-3-yl}methyl)-3-(propan-2-yl)urea
5-({4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)pyrimidin-2-amine
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-1-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
(1R,5R)-6-{[4-(difluoromethoxy)phenyl]methyl}-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
2-(methoxymethyl)-1-{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}piperidine
N-(4H-1,2,4-triazol-4-yl)-2-(4,6,7-trimethyl-1-benzofuran-3-yl)acetamide
14-(2-phenylethyl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
5-[(3-benzoylpiperidin-1-yl)methyl]-2-(furan-2-yl)pyrimidine
3-{1-[2-oxo-2-(pyrrolidin-1-yl)acetyl]piperidin-3-yl}benzoic acid
(4aR,7aS)-1-ethyl-4-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-chloro-N-(2-ethoxypropyl)-N-methyl-3-phenyl-1H-indole-2-carboxamide
(2S,4R)-N-methyl-1-[2-(methylsulfanyl)acetyl]-4-(3-phenoxypropanamido)pyrrolidine-2-carboxamide
4-{2-[(dimethylamino)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-4-oxobutane-1-sulfonamide
dimethyl({2-[2-(1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}piperidin-4-yl)-1H-imidazol-1-yl]ethyl})amine
2-({[(1-cyclopentylpiperidin-4-yl)methyl](oxolan-2-ylmethyl)amino}methyl)quinolin-4-ol
5-methyl-1-propyl-N-[1-(pyridin-3-yl)propan-2-yl]-1H-pyrazole-4-carboxamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(6-oxo-1,6-dihydropyrimidin-5-yl)acetamide
(2S)-2-{[2-(2-methoxy-4-methylphenoxymethyl)-1,3-oxazol-4-yl]formamido}propanamide
2-{[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]oxy}-N-cyclopropyl-4-methoxybenzamide
1-[3-(2-methoxyphenyl)phenyl]-3-{2-[(2R)-pyrrolidin-2-yl]ethyl}urea
N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
7-fluoro-3-methyl-2-{3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl}-1H-indole
3-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-fluorophenyl)urea
(3aS,6aS)-2-ethyl-5-{[3-hydroxy-5-(hydroxymethyl)-2-methylpyridin-4-yl]methyl}-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4,6-dimethyl-N-[(5-methylpyrazin-2-yl)methyl]pyrimidin-2-amine
6-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyrimidin-4-amine
1-cyclopentyl-N3-(3-methylbutyl)-4-oxo-N5-(pyridin-3-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
N-[(3S,4S)-4-methoxy-1,1-dioxo-1λ6-thiolan-3-yl]-4-(piperidin-1-yl)benzamide
2-(1-benzyl-3-oxopiperazin-2-yl)-N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]acetamide
4,6-dimethyl-N-[2-(2-methylpropanesulfonyl)ethyl]-2-oxo-1,2-dihydropyridine-3-carboxamide