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5-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-N-phenylpyrimidin-2-amine
3-[2-(2,4-difluorophenyl)ethyl]-1-[4-(propan-2-yl)-1,2,3-thiadiazole-5-carbonyl]piperidine
1-{[3-({1-[4-(4-fluorophenyl)benzoyl]piperidin-4-yl}oxy)phenyl]methyl}-4-(pyridin-2-yl)piperazine
1-(4-ethyl-5-methylpyrimidin-2-yl)-4-(morpholine-4-sulfonyl)-1,4-diazepane
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-(pyrrolidine-1-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
6-(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidin-3-yl)-2-methyl-3,4-dihydropyrimidin-4-one
10-methoxy-5-(oxolan-3-ylmethyl)-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
N-[2-(6-hydroxypyrimidin-4-yl)ethyl]-3-(5-methylfuran-2-yl)benzamide
4-({1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}methyl)-2-ethoxy-6-(prop-2-en-1-yl)phenol
N-ethyl-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
8-[(2S)-2-amino-3-(1H-imidazol-4-yl)propanoyl]-3-(2-ethylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N3-[(2-ethyl-4-methyl-1,3-thiazol-5-yl)methyl]-N1,N1-dimethylpiperidine-1,3-dicarboxamide
N-[(3,4-dimethoxyphenyl)methyl]-4-methyl-5-{1-[2-(thiophen-2-yl)ethyl]-1H-pyrazol-3-yl}-1,3-thiazol-2-amine
3-[(cyclohex-3-en-1-ylmethyl)amino]-5-(dimethylsulfamoyl)-N-methyl-N-[1-(pyridin-2-yl)ethyl]benzamide
(2R,3S,6R)-3-(3-methoxyphenyl)-5-(1-methyl-1H-pyrrole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-acetyl-N-{2-hydroxy-2-[4-(trifluoromethyl)phenyl]ethyl}-1H-pyrazole-5-carboxamide
3-[1-(1H-imidazol-1-ylmethyl)cyclopropanecarbonyl]-9-methyl-3,9-diazaspiro[5.6]dodecan-10-one
2-ethyl-8-[2-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)butanoyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
N-({3-methyl-7-[2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-2-carboxamide
(3aR,6aR)-2-(oxane-4-carbonyl)-5-(pyridin-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(4-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-1-(thiophen-2-ylmethyl)piperazin-2-yl)ethan-1-ol
(3S,5S)-1-(cyclopentylmethyl)-5-[(pyridin-2-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
6-(dimethylamino)-N-[(3-methylthiophen-2-yl)methyl]-N-(pyridin-2-ylmethyl)pyridine-3-carboxamide
(2S,4S)-4-amino-N,N-diethyl-1-(1-methyl-1H-indole-3-carbonyl)pyrrolidine-2-carboxamide
3,3,3-trifluoro-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]propanamide
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxy-N-(oxan-4-ylmethyl)benzamide
(2S,4R)-N,1-dimethyl-4-{3-[5-(thiophen-2-yl)furan-2-yl]propanamido}pyrrolidine-2-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-cyclopropyl-2-[(prop-2-en-1-yl)amino]benzamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-1-(pyrrolidin-1-yl)cyclopentane-1-carboxamide
2-[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidin-1-yl]pyridine-3-carboxylic acid
2-[2-oxo-2-(3-phenoxyazetidin-1-yl)ethyl]-1,2-dihydroisoquinolin-1-one
4-(1-butyl-1H-imidazol-2-yl)-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidine
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)-1-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
4-(3-methylphenoxy)-1-(6-methylpyridazin-3-yl)piperidine-4-carboxylic acid
N-[(4-fluorophenyl)methyl]-1-methyl-5-{[(3-methyloxetan-3-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-(quinolin-5-ylmethyl)piperidin-4-ol
methyl 4-[2-amino-3-cyano-6-(3,5-dimethyl-1H-pyrazol-4-yl)pyridin-4-yl]-1H-pyrazole-3-carboxylate
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methylacetamide
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-3-(1H-1,2,4-triazol-1-yl)propanamide
{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]amine
N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
(2S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-N-methyl-4-[(propan-2-yl)amino]pyrrolidine-2-carboxamide
4-(4-methoxy-2-methylphenyl)-3-(pyrrolidin-1-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(4-cyano-2-ethylphenyl)-4-[(2-methylpyrrolidin-1-yl)methyl]benzamide
2-amino-7-[4-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(oxan-2-ylmethoxy)ethan-1-one
6-hydroxy-N-(1H-indazol-7-yl)-1,4-oxazepane-4-carboxamide