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2-(2-hydroxyethyl)-6-(4-methyl-3,4-dihydro-2H-1,4-benzoxazine-2-carbonyl)-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
(2S,4S,5R)-5-(4-chlorophenyl)-1,2-dimethyl-4-(4-methylpiperazine-1-carbonyl)pyrrolidine-2-carboxylic acid
4-(2,2-dimethylpropanoyl)-1-(4-methylphenyl)piperazin-2-one
N-[(3-chlorophenyl)methyl]-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-cyclopropyl-N-[(4-methylphenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-[(2R)-1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-1-oxobutan-2-yl]acetamide
3-[benzyl(2-phenylethyl)amino]-2-methylpropan-1-ol
1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(methylamino)ethan-1-one
1-(2-aminoethyl)-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
3-{1-[1-(2-cyclopentylacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methoxyphenyl)urea
(1-{[7-chloro-2-(2-methoxyphenyl)quinolin-3-yl]methyl}piperidin-4-yl)methanol
N-[(5-chloro-2-ethoxyphenyl)methyl]-N-methyl-3-(pyridin-4-yl)propanamide
3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-N-(1-ethyl-1H-1,2,3-triazol-4-yl)benzamide
8-[(2S,3R)-2-amino-3-hydroxybutanoyl]-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{2-methyl-2,8-diazaspiro[4.5]decan-8-yl}ethan-1-amine
N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
4-benzoyl-1-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidine
2-ethyl-N-(4-methoxy-3-pentanamidophenyl)-4-methyl-1,3-oxazole-5-carboxamide
2-(2-{1-oxa-8-azaspiro[4.6]undecan-8-yl}-2-oxoethyl)-2,3-dihydro-1,2-benzothiazol-3-one
2-(2-{1-ethyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1H-pyrrol-1-yl)-1,3-thiazole
3-(4-{spiro[azepane-4,2'-chromene]-1-ylmethyl}phenyl)prop-2-yn-1-ol
(4aR,8aS)-1-(3,3-diphenylpropyl)-6-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-decahydro-1,6-naphthyridin-2-one
4-(naphthalen-2-ylmethyl)-1-(3-phenoxypropanoyl)-1,4-diazepan-5-one
N-(2,2-dimethyloxan-4-yl)-6-{[4-(hydroxydiphenylmethyl)piperidin-1-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidin-3-yl}propanamide
2,4-dimethyl-N-[1-methyl-4-(2-oxo-1,3-oxazolidin-3-yl)-1H-indazol-3-yl]-1,3-thiazole-5-carboxamide
methyl 3-chloro-4-[(4,4-difluoropiperidine-1-carbonyl)amino]benzoate
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[3-(4-hydroxyphenyl)propyl]acetamide
diethyl({[3-(1,4-oxazepane-4-carbonyl)pyrazolo[1,5-a]pyrimidin-6-yl]methyl})amine
N-[3-(tert-butylcarbamoyl)-2-methylphenyl]-6-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
1-[1-(3-methoxybenzoyl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine
(1S,5R)-6-benzyl-3-[(3-phenyl-1,2-oxazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
6-(4-{2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carbonyl}piperazin-1-yl)pyridine-3-carbonitrile
4-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}thiomorpholine
5-[2-(4-fluorophenyl)piperidine-1-carbonyl]-N-phenylpyrimidin-2-amine
4-{[(4-methyl-5-{1-[(3-methylthiophen-2-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)sulfanyl]methyl}pyridine
2-(2-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}phenoxy)acetic acid
{1-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
(3S,4R)-1-[4-(2-methyl-1H-imidazol-1-yl)butanoyl]-4-phenylpyrrolidine-3-carboxylic acid
9-{[1-(4-methoxyphenyl)-1H-pyrrol-2-yl]methyl}-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]-N-[4-(pyridin-2-yl)butyl]piperidine-3-carboxamide
3-{2-[(8-fluoroquinolin-2-yl)formamido]acetamido}propanoic acid
5-methoxy-4-oxo-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1,4-dihydropyridine-2-carboxamide
1-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(phenylsulfanyl)ethan-1-one
1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-3-(3-methylphenoxymethyl)piperidine
2-(2-ethoxypyridin-3-yl)-2-[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]acetic acid
N,N-diethyl-2-[(5-methylpyrazin-2-yl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
2-[8-(pyrimidin-2-yl)-1,8-diazaspiro[4.5]decan-1-yl]acetic acid
5-{2-[1-(2-methylpyridin-4-yl)-3-phenyl-1H-1,2,4-triazol-5-yl]ethyl}imidazolidine-2,4-dione
3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1-methyl-1,2-dihydroquinoxalin-2-one