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[1-(2-methylpyrimidin-4-yl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-3-methoxypropan-1-one
2-[3-(3-fluorophenoxymethyl)-5-(4-propylpyrimidin-5-yl)-1H-1,2,4-triazol-1-yl]acetic acid
ethyl 3-benzyl-1-(thiophene-2-sulfonyl)piperidine-3-carboxylate
N-{[1-(1-butanoylpiperidin-4-yl)pyrrolidin-3-yl]methyl}methanesulfonamide
5-(1-cyclopentyl-1H-pyrazol-3-yl)-4-methyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1,3-thiazol-2-amine
N-{[7-fluoro-2-(4-methylphenyl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)-5-methylthiophene-2-carboxamide
N-butyl-N-(furan-2-ylmethyl)-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
2-[(adamantan-1-ylmethyl)({[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl})amino]ethan-1-ol
2-(4-methoxyphenyl)-7-methyl-3-(1,4-oxazepan-4-ylmethyl)quinoline
6-{7-methyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}pyridine-2-carbonitrile
N-(cyclopropylmethyl)-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
(1R,5S,6R)-3-[(2,3-dichloro-4-methylphenyl)methyl]-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
3-[(dimethylamino)methyl]-1-(quinolin-5-ylmethyl)piperidin-3-ol
2-[2-(1H-imidazol-4-yl)ethyl]-9-[3-(pyridin-3-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
[(1-tert-butyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](propyl)(pyridin-3-ylmethyl)amine
(2S,4R)-N-[4-(3-acetylphenyl)phenyl]-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidine-1-carboxamide
6-tert-butyl-1-methyl-N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}propane-1,2-dione
1-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-3-(3,5-dimethyl-1H-pyrazol-4-yl)propan-1-one
2-{2-[4-(1-hydroxyethyl)piperidin-1-yl]-4-(morpholin-4-yl)pyrimidin-5-yl}-2-methylpropanoic acid
1-[2-(1H-imidazol-2-yl)benzoyl]-4-methoxy-4-phenylpiperidine
4-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}piperazine-1-sulfonamide
(4aR,8aS)-1-butyl-6-(cyclohexylmethyl)-decahydro-1,6-naphthyridin-2-one
2-(2-oxo-1,2-dihydropyridin-1-yl)-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]acetamide
N-methyl-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]-N-(oxan-4-ylmethyl)acetamide
4-fluoro-N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}benzamide
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-5-(methoxymethyl)thiophene-2-carboxamide
8-(1-benzofuran-5-carbonyl)-2-methyl-2,8-diazaspiro[4.5]decan-3-one
N-methyl-3-(1H-pyrazol-1-yl)-N-[1-(1,3-thiazol-5-yl)ethyl]benzamide
3,3-dimethyl-1-[(3S,4R)-1-(2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetyl)-4-(propan-2-yl)pyrrolidin-3-yl]urea
2-{3-[3-(pyridin-3-yl)-1H-pyrazol-1-yl]phenoxy}propanamide
1-[5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]azetidin-3-ol
2-methyl-N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}propanamide
3-(4-fluorophenyl)-3-{[3-(4H-1,2,4-triazol-4-yl)phenyl]formamido}propanoic acid
2-methyl-4-[4-(piperidin-1-ylmethyl)piperidin-1-yl]pyridine
3-(1-methylpiperidin-2-yl)-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}propanamide
1-[(4-methoxyphenyl)methyl]-4-[2-(pyridin-3-yl)acetyl]piperazin-2-one
1-methyl-3-(propan-2-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-pyrazole-5-carboxamide
(3S)-2-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-3-carboxylic acid
2-methyl-7-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-(cyclohexylmethyl)-1-cyclopropyl-4-oxo-5-[4-(piperidin-1-yl)piperidine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
2-[(2-fluorophenyl)methyl]-4-{4-[(4-methoxy-2,5-dimethylphenyl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
4-[(4-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}furan-2-yl)methyl]morpholine
7-[(5,7-dimethyl-2,1,3-benzoxadiazol-4-yl)sulfonyl]-2-oxa-7-azaspiro[4.5]decane
3-[3-(4-ethylpiperazin-1-yl)propyl]-8-(pyridine-4-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[2-(3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl)-2-oxoethyl]-3-phenylcyclopent-2-en-1-one
N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-4-pentanamidobenzamide
N-{[2-fluoro-3-(trifluoromethyl)phenyl]methyl}-4-(2-oxopyrrolidin-1-yl)butanamide
2-(2-fluorophenyl)-N-[2-(pyrrolidine-3-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]acetamide