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N-[4-chloro-3-({[3-(1-methyl-1H-pyrazol-4-yl)propyl]carbamoyl}amino)phenyl]-2-methoxyacetamide
1-(1-cyclopropylethyl)-N-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-methyl-1H-pyrazol-5-amine
9-(6-methoxypyrimidin-4-yl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
methyl 2-[4-benzyl-5-oxo-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]butanoate
4-ethyl-1-[(2E)-3-phenylprop-2-en-1-yl]-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-3-(pyrrolidine-1-carbonyl)piperidine
3-[(5-cyclopentyl-4-phenyl-1H-imidazol-1-yl)methyl]-N-methylbenzamide
{[3,5-dichloro-4-(prop-2-en-1-yloxy)phenyl]methyl}({[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl})amine
N-methyl-3-(1-phenylethyl)-N-(thiophen-3-ylmethyl)-1,2-oxazole-5-carboxamide
2-[8-(3-methylbutyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]-1,3-thiazole-4-carboxamide
5-(propan-2-yl)-N-[1-(pyridin-3-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-[4-(4-{[2-(ethylamino)pyrimidin-5-yl]methyl}piperazin-1-yl)phenyl]ethan-1-one
4-(4-{[(5-chlorothiophen-2-yl)methyl]amino}piperidin-1-yl)-N-cyclopentylbenzamide
2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]-1-[4-(4H-1,2,4-triazol-4-yl)piperidin-1-yl]ethan-1-one
{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}[1-(furan-2-yl)ethyl]methylamine
N-[(3-methoxyphenyl)methyl]-2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]-N-(prop-2-en-1-yl)acetamide
5-(2,5-difluorophenyl)-1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-phenyl-1H-imidazole
ethyl 4-{5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}piperazine-1-carboxylate
8-chloro-2-[1-(methoxymethyl)cyclobutanecarbonyl]-1H,2H,3H,4H,5H-pyrido[4,3-b]indole
3-cyano-5-fluoro-N-(isoquinolin-5-ylmethyl)-N-methylbenzamide
(3R)-1-[(5-cyclohexylthiophen-2-yl)methyl]pyrrolidin-3-ol
4,4,4-trifluoro-1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]butan-1-one
3-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}(pyridin-3-ylmethyl)amino)propan-1-ol
3-{[3-(4-chlorophenyl)-1-(2-hydroxyethyl)-1H-1,2,4-triazol-5-yl]methyl}-4-ethylpiperazin-2-one
3-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-methylpyridine
2-fluoro-6-{6-[(2-methoxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
3-({[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}(prop-2-en-1-yl)amino)-1λ6-thiolane-1,1-dione
(4aR,6R,8aS)-8a-(methoxymethyl)-2-[(5-methylfuran-2-yl)methyl]-6-(morpholin-4-yl)-decahydroisoquinoline
2-(4-{2-methylimidazo[1,2-a]pyridine-6-carbonyl}piperazin-1-yl)pyrimidine
2-methyl-7-[(2-methyl-1,3-oxazol-4-yl)methyl]-N-(1H-1,2,4-triazol-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-{1-benzyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}-2-(4H-1,2,4-triazol-4-yl)pyridine
11-[1,3-dimethyl-5-(morpholin-4-yl)-1H-pyrazol-4-yl]-4,6,10,12-tetraazatricyclo[7.3.0.03,7]dodeca-1,3(7),8,10-tetraen-5-one
N-(2-phenylethyl)-3-{[1-(thiophen-2-ylmethyl)piperidin-4-yl]oxy}benzamide
N-{[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}thiophene-2-carboxamide
5-ethyl-N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-1,2-oxazole-4-carboxamide
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-N'-cyclopentylbutanediamide
N-(3-methoxyphenyl)-3-{1-[(4-methylthiophen-2-yl)sulfonyl]piperidin-4-yl}propanamide
N-{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyloxan-4-amine
2-(ethanesulfonyl)-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
4-[4-(pyrimidin-2-yloxy)piperidine-1-carbonyl]-1-oxaspiro[4.4]nonan-2-one
3-{2-[4-(1H-imidazol-4-ylmethyl)morpholin-2-yl]ethyl}-1-phenylurea
N-(3-methoxypropyl)-6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
4-phenyl-3-[1-(pyridin-2-ylmethyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[1-(4-cyclohexylpiperazine-1-carbonyl)-6-azaspiro[2.5]octan-6-yl]-2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]ethan-1-one
N-(1H-imidazol-2-ylmethyl)-1-[4-(3-methoxyphenyl)phenyl]piperidin-4-amine
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[(1-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)methyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
5-ethyl-N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}pyrimidin-2-amine
2-[3-(pyridin-3-yl)propyl]-1,2-dihydrophthalazin-1-one
(2S,4R)-4-amino-1-{[2-(2-hydroxyethoxy)phenyl]methyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide