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2-({[(1R,9aR)-1-hydroxy-octahydro-1H-quinolizin-1-yl]methyl}amino)-N-(2-methoxy-5-methylphenyl)acetamide
(1R,7S)-6-(4-fluoropiperidine-1-carbonyl)-3-(2-phenoxyethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
5-[3-(3-methoxyphenyl)-1H-pyrazole-5-carbonyl]-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
5-[6-(3-fluorophenyl)pyridine-3-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
2-methyl-6-[1-(2-phenylpropyl)piperidin-4-yl]pyrimidin-4-ol
6-(3-chlorophenyl)-7-(cyclopropylmethyl)-2-(2-methylpyrrolidine-1-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
(4aS,8aR)-6-[1-(methoxymethyl)cyclobutanecarbonyl]-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
1-{5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-4-methyl-1,4-diazepane
methyl N-{2-oxo-2-[9-oxo-8-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-2-yl]ethyl}carbamate
7-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-N,N-dimethyl-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{pyrazolo[1,5-a]pyridine-2-carbonyl}piperidin-3-ol
(1S,5R)-6-(3-fluoro-4-methylbenzoyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-(diphenylmethyl)-N-methyl-N-(1,2-oxazol-5-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
3-fluoro-N-methyl-N-(oxan-2-ylmethyl)pyridine-4-carboxamide
4-{1-[1-(1-phenylethyl)-1H-1,2,3,4-tetrazol-5-yl]azetidin-3-yl}pyridine
diethyl({2-ethyl-5-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]furan-3-yl}methyl)amine
N-[(5-methoxy-1H-indol-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
2-{[(2-ethoxypyridin-3-yl)methyl]amino}-N-(pyrazin-2-yl)acetamide
7-amino-4-[1-(propan-2-yl)piperidin-4-yl]-1,2,3,4-tetrahydro-1,8-naphthyridin-2-one
(3aS,7aR)-2-(1-benzothiophene-5-carbonyl)-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
6-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidine-1-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
6-{4-[2-(2-methoxyethyl)-1,3-benzoxazole-6-carbonyl]piperazin-1-yl}pyridine-3-carbonitrile
1-[(4R)-3-methyl-1,3-thiazolidine-4-carbonyl]-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
1-(1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperidin-4-yl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-6-oxo-1,6-dihydropyrimidine-5-carboxamide
2-{4-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]piperidin-1-yl}acetamide
1-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(2H-1,2,3-triazol-2-yl)ethan-1-one
2-{1-[3-(1H-pyrazol-1-yl)benzoyl]pyrrolidin-2-yl}-1,3-thiazole
5-(azocane-1-carbonyl)-N-[(4-methylphenyl)methyl]-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
6-{[(2S,5R)-5-[(4-ethylpiperazin-1-yl)methyl]oxolan-2-yl]methyl}-2-methylquinoline
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-5-methylpiperidin-2-one
2-{4-[(1S,3S,3aR,6aS)-3-(hydroxymethyl)-5-methyl-3-phenyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]-3,5-dimethyl-1H-pyrazol-1-yl}ethan-1-ol
2-(2-amino-6-methylpyrimidin-4-yl)-7-cyclohexyl-2,7-diazaspiro[4.5]decan-6-one
2-{3,9-diazaspiro[5.5]undecan-3-yl}-N-(2-ethylphenyl)-2-oxoacetamide
1-[4-(2,3-dimethylphenyl)piperazin-1-yl]-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}ethan-1-one
1-(3-propyl-1H-pyrazole-5-carbonyl)-4-(1H-pyrrole-2-carbonyl)piperazine
1-phenyl-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-2-(pyridin-3-yl)morpholine
{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}[(3-methylphenyl)methyl]amine
5-chloro-N,3-dimethyl-N-[1-(pyridin-2-yl)propyl]-1H-indole-2-carboxamide
2-{4-[(2-propylpyrimidin-5-yl)methyl]piperazin-1-yl}pyridine-4-carboxamide
1-[3-(2-methyl-1,3-thiazol-4-yl)phenyl]-N-[(3R)-oxolan-3-yl]piperidin-4-amine
1-cyclohexyl-4-{1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazin-2-one
N-(2-methoxyethyl)-N-(1-methylpiperidin-4-yl)-2-(pyridin-4-yl)pyrimidine-5-carboxamide
8-chloro-2-(1H-imidazol-2-yl)quinoline
(1S,5R)-6-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
[(3R,4S)-4-[(4-methylpiperazin-1-yl)methyl]-1-(3-phenylpropyl)pyrrolidin-3-yl]methanol
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[3-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]ethan-1-one
4-{1-[4-(2,4-dimethoxypyrimidin-5-yl)phenyl]ethyl}morpholine
3-(2-methoxyphenyl)-1-[2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]propan-1-one