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6-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]pyrimidin-4-amine
methyl 6-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)-3-(2-phenylacetamido)thieno[2,3-b]pyridine-2-carboxylate
2-(2-ethyl-1H-imidazol-1-yl)-N-[1-(pyridine-3-carbonyl)azepan-3-yl]acetamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}propanamide
(4aS,7aR)-1-(3-phenylpropyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1S,5R)-6-(1-methyl-1H-indole-3-carbonyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}-2-[(3-methylpiperidin-3-yl)methoxy]pyridine
N-[1-(4-fluorophenyl)ethyl]-2-{[4-(furan-2-carbonyl)piperazin-1-yl]methyl}quinazolin-4-amine
N-cyclopropyl-6-methyl-2-(4-methylphenoxymethyl)-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
(4aR,7aS)-1-benzyl-4-[2-(propan-2-ylsulfanyl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(3R,4S)-1-(carbamoylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]-1-(2-fluorophenyl)cyclopropane-1-carboxamide
2-methyl-1-(4-{[(1-phenoxypropan-2-yl)amino]methyl}piperidin-1-yl)propan-1-one
4-[(2S)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole
(2S,4R)-4-{[(3-chlorophenyl)methyl]amino}-N-ethyl-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
3-[1-(cyclopropylmethyl)-1H-pyrazol-5-yl]-1-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]urea
(3S)-1-{[5,8-dimethoxy-2-(2-methoxyphenyl)quinolin-3-yl]methyl}pyrrolidin-3-ol
3-{2-[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]-2-oxoethyl}-5-fluoro-2,3-dihydro-1H-indol-2-one
N-[(2,6-difluoro-3-methoxyphenyl)methyl]-3-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]propanamide
(2S,4R)-N-methyl-4-[(pyrimidin-2-yl)amino]-1-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]pyrrolidine-2-carboxamide
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-4-(1H-pyrazol-1-yl)benzamide
(2S)-4-methyl-2-phenyl-1-{[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}piperazine
1-(2-methoxy-2-methylpropyl)-5-methyl-5-phenylpiperidin-2-one
N-{2-[4-phenyl-5-(2-phenylethyl)-1H-imidazol-1-yl]ethyl}methanesulfonamide
{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}({[5-(3-methoxyphenyl)-1,2-oxazol-3-yl]methyl})amine
1-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-4-phenoxybutan-1-one
(2S,4S)-4-amino-1-{[4-(3,4-dimethylphenoxy)phenyl]methyl}-N-methylpyrrolidine-2-carboxamide
5-methyl-N-({1-[(2-methyl-1H-imidazol-4-yl)methyl]pyrrolidin-3-yl}methyl)pyrazine-2-carboxamide
1-{1-[(2E)-2-methylbut-2-enoyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
2-[2-(1H-imidazol-4-yl)ethyl]-8-(4-methylpiperidine-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
(2R,6R)-11-methoxy-4-[(2-methoxyphenyl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-(1-{[1-(benzenesulfonyl)-1H-pyrrol-2-yl]methyl}pyrrolidin-2-yl)pyridine
3-hydroxy-3-({[2-(methylamino)ethyl]amino}methyl)-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
3-{[(2-chloro-5-fluorophenyl)methyl](ethyl)amino}-1λ6-thiolane-1,1-dione
2-{4-[(3,4-dimethylpiperazin-1-yl)methyl]phenoxy}-1-(pyrrolidin-1-yl)ethan-1-one
(5-{1-[1-(oxolan-2-ylmethyl)piperidin-4-yl]-1H-imidazol-2-yl}furan-2-yl)methanol
(2S,4S)-4-{[(4-methoxy-2,3-dimethylphenyl)methyl]amino}-N-(propan-2-yl)-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
2-(2-aminoethyl)-N-[(2,4-dimethoxyphenyl)methyl]quinazolin-4-amine
(4aS,8aR)-6-(2-amino-4-methylpyrimidine-5-carbonyl)-1-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
5-chloro-N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]thiophene-2-sulfonamide
5-(morpholin-4-yl)-1-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(2-methoxyphenyl)piperazine
1-{3-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]phenyl}ethan-1-one
3-(2H-1,3-benzodioxol-5-yl)-1-[3-(5-methyl-2-{[2-(morpholin-4-yl)ethyl]sulfanyl}pyrimidin-4-yl)piperidin-1-yl]propan-1-one
2-cyclopentyl-9-[3-(pyridin-3-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
(4aS,8aR)-6-[1-(difluoromethyl)-1H-pyrazole-5-carbonyl]-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
3-hexyl-8-(6-methyl-4-oxo-1,4-dihydropyridine-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(3-methylbut-2-en-1-yl)-1-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-3-carboxylic acid
N-(3-carbamoyl-2-methylphenyl)-6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-[2-methoxy-5-(methylcarbamoyl)phenyl]-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carboxamide
1-[7-(1-benzothiophen-3-yl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(3,5-dimethyl-1H-pyrazol-1-yl)propan-1-one