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3-(1H-imidazol-2-yl)-1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]piperidine
3-[4-(3-methylphenyl)piperazin-1-yl]-N-[(3-propyl-1,2-oxazol-5-yl)methyl]propanamide
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-3-ol
(2S,4R)-4-amino-1-{1-[(4-methoxyphenyl)amino]cyclohexanecarbonyl}-N-methylpyrrolidine-2-carboxamide
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-ethylthiophene-2-carboxamide
N-(1-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]propanoyl}piperidin-4-yl)methanesulfonamide
2-methoxy-N,N-dimethyl-5-({[1-(pyrazin-2-yl)propan-2-yl]carbamoyl}amino)benzamide
1-(2-methoxyethyl)-8-[(3-methoxyphenyl)methyl]-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{5-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1-methyl-1H-pyrazole
1-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
methyl 5-{[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}-3-(oxolane-3-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-({3-[2-(dimethylamino)ethoxy]phenyl}methyl)piperazine-1-carboxamide
4-(3-acetylbenzoyl)-1-[(3-fluorophenyl)methyl]piperazin-2-one
4-benzyl-1-(4-methylquinolin-2-yl)piperidine-4-carboxylic acid
1-(3-hydroxyazetidin-1-yl)-3-(4-methoxyphenyl)-3-phenylpropan-1-one
2-amino-4-[3-(pyridin-2-ylmethoxy)phenyl]-6-(1H-pyrrol-3-yl)pyridine-3-carbonitrile
3-{2-oxo-2-[3-(4-phenoxybenzoyl)piperidin-1-yl]ethyl}-1,3-thiazolidine-2,4-dione
N-(2,1,3-benzothiadiazol-5-ylmethyl)-3-{2-[(3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methylpropanamide
2-({2-[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N,N-dimethyl-2-[(2-phenoxypropanamido)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
4-(3,6-dimethylpyrazin-2-yl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
methyl[(3-{[1-(3-phenyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]oxy}phenyl)methyl](thiophen-2-ylmethyl)amine
4-(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)-4-oxobutane-1-sulfonamide
2-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]acetic acid
1-{1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
1-(2-aminoethyl)-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-methyl-5-{1-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]pyrrolidin-2-yl}thiophene-2-carboxamide
N-cyclopentyl-N-({4-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)propanamide
1,3-dimethyl-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
4-{2-methoxy-5-[3-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]phenyl}morpholine
3-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-1-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]urea
2,6-dimethyl-4-[3-(2-methylphenoxy)azetidine-1-carbonyl]quinoline
N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}-4-(3,3,3-trifluoropropyl)pyrimidine
N-[(2-chlorophenyl)methyl]-N'-(2-fluoro-5-methylphenyl)-N-(2-hydroxyethyl)butanediamide
(2S,4S)-4-amino-N,N-diethyl-1-(pyridine-3-sulfonyl)pyrrolidine-2-carboxamide
2-{1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]pyrrolidin-2-yl}pyridine
N-[(1-ethylcyclobutyl)methyl]-5-[(4-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
4-{4-[({[1-(2-methoxyethyl)piperidin-4-yl]methyl}(oxolan-2-ylmethyl)amino)methyl]phenyl}-2-methylbut-3-yn-2-ol
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(dimethylamino)-2-(2-fluorophenyl)acetamide
2-{[2-(1H-indol-3-yl)ethyl]amino}-N-[4-(N-methylacetamido)phenyl]acetamide
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carboxamide
N-cyclopropyl-1-[1-(3-propyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
2-(but-3-enoyl)-7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decan-6-one
1-(2-oxo-1,2-dihydroquinoline-4-carbonyl)-4-phenylpiperidine-4-carbonitrile
1-methyl-4-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
N-ethyl-N-(2-methylprop-2-en-1-yl)-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-ethyl-4-[3-(3-methylphenoxy)azetidine-1-carbonyl]pyrrolidin-2-one
N-(2H-1,3-benzodioxol-5-yl)-3-(3-chlorobenzoyl)piperidine-1-carboxamide
1-[3-(2-phenylacetyl)piperidin-1-yl]-3-(thiophen-3-yl)propan-1-one