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2-(2H-1,2,3-benzotriazol-2-yl)-N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]acetamide
1-{5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(methylsulfanyl)propan-1-one
2-(1-cyclohexyl-4-{5-ethyl-6-methylthieno[2,3-d]pyrimidin-4-yl}piperazin-2-yl)ethan-1-ol
N-[2-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)ethyl]-5-ethyl-1,3,4-oxadiazol-2-amine
1-{3-fluoro-7-methylimidazo[1,2-a]pyridine-2-carbonyl}-3-(3-methoxyphenoxy)azetidine
2-{1-[1-(2-fluorophenyl)-2,2-dimethylcyclopropanecarbonyl]azetidin-3-yl}pyridine
2-(2-hydroxyethyl)-9-[5-(methoxymethyl)thiophene-2-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[(3-fluorophenyl)methyl]-4-{4-[(3-methylthiophen-2-yl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
1,4,6-trimethyl-3-[4-(2-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]-1,2-dihydropyridin-2-one
7-(3-chlorophenyl)-4-(6-ethylpyrimidin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
7-(5-chloropyridin-2-yl)-4-[(5-methylfuran-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-methyl-4-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}benzene-1-sulfonamide
3-(3-methanesulfonamidopropanamido)-4-(2-methylpiperidin-1-yl)benzamide
1-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-3-propylurea
4-(1,4-dioxan-2-ylmethyl)-6-fluoro-3,4-dihydro-2H-1,4-benzoxazin-3-one
N-[(2-phenoxypyridin-3-yl)methyl]-2H-1,3-benzodioxole-5-carboxamide
3-(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-4-yl)-N-(oxolan-2-ylmethyl)propanamide
3-(3-chloro-1H-1,2,4-triazol-5-yl)-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
N-[(2-fluorophenyl)methyl]-5-methyl-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
4-({3-[(4-methylpiperazin-1-yl)methyl]piperidin-1-yl}methyl)benzoic acid
2-(3-chlorophenyl)-1-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-(6-methoxynaphthalen-2-yl)-4-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]morpholine
ethyl 1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-4-[(3-fluorophenyl)methyl]piperidine-4-carboxylate
2-(4-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}piperazin-1-yl)-1,3-benzoxazole
N-[(3R,4S)-4-cyclopropyl-1-(2-hydroxyethyl)pyrrolidin-3-yl]-1-propyl-1H-pyrazole-4-sulfonamide
{[5,8-dimethoxy-2-(3-methoxyphenyl)quinolin-3-yl]methyl}(thiophen-2-ylmethyl)amine
2-[(3S,4S)-3-carboxy-4-propylpyrrolidin-1-yl]-6-methylpyridine-3-carboxylic acid
N-(2,4-difluorophenyl)-2-[2-(morpholin-4-yl)ethyl]piperidine-1-carboxamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-3,5-dimethyl-1,2-oxazole-4-sulfonamide
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2-(2,4-dioxoimidazolidin-1-yl)acetamide
2-methoxy-2-methyl-N-[(3R,4S)-4-propyl-1-[2-(pyridin-2-yl)ethyl]pyrrolidin-3-yl]propanamide
2-ethoxy-N-(2-methoxyethyl)-N-(thiophen-2-ylmethyl)pyridine-3-carboxamide
4-[(4-methyl-5-{1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]piperidin-3-yl}-4H-1,2,4-triazol-3-yl)methyl]morpholine
1-ethyl-3-(naphthalen-1-ylmethyl)-8-(thian-4-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S,4R)-1-benzyl-N,N-diethyl-4-{[(3-hydroxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
6-(3-fluorophenyl)-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}pyridine-3-carboxamide
N-[1-benzyl-4-(propan-2-yloxy)-1H-indazol-3-yl]pyridazine-3-carboxamide
5-(methoxymethyl)-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-N-[(6-methylpyridin-2-yl)methyl]-1H-pyrazole-4-carboxamide
2-{1-[3-(4-methyl-1,4-diazepan-1-yl)propanoyl]pyrrolidin-3-yl}benzoic acid
(2S,4R)-4-amino-N-ethyl-1-[3-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)propanoyl]pyrrolidine-2-carboxamide
3-[(4-methoxyphenyl)methyl]-1-methyl-8-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(3R,4S)-1-(5-cyanopyridin-2-yl)-4-cyclopropylpyrrolidin-3-yl]oxane-4-carboxamide
6-(morpholin-4-yl)-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-3-propyl-1H-pyrazole-5-carboxamide
2-oxo-N-(2-phenylethyl)-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
(2S)-2-acetamido-N-(2-methoxyethyl)-4-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]pentanamide
({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]amine
(2S,3R)-2-amino-3-hydroxy-1-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}butan-1-one
N,1-dimethyl-N-(1,2-oxazol-5-ylmethyl)-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[3-(1,3-benzothiazol-2-yl)propyl]-4-(pyridin-2-yl)pyrimidin-2-amine