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N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]-1-(propan-2-yl)piperidine-3-carboxamide
4-[3-(3-methoxyphenoxy)azetidine-1-carbonyl]-2,6-dimethylquinoline
3-[2-(3-methoxyphenyl)ethyl]-1-(2-methylfuran-3-carbonyl)piperidine
N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
5-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane-11-carbonyl}-4-ethyl-1,3-thiazol-2-amine
3-{[3-(dimethylamino)propyl](methyl)amino}-N,N-dimethylpiperidine-1-sulfonamide
3-[2-oxo-2-(thiomorpholin-4-yl)ethyl]-2,3-dihydro-1H-isoindol-1-one
2-{[6-(1-benzofuran-2-yl)pyridazin-3-yl]amino}ethan-1-ol
({4-ethyl-5-[1-(1-methyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
N-methyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-[(3-chloro-4-fluorophenyl)methyl]-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
ethyl 5-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carbonyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2,5-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
(3S,7S,8aS)-7-{[(3-fluorophenyl)methyl]amino}-3-(1H-indol-3-ylmethyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
6-{2,7-diazaspiro[4.5]decane-2-sulfonyl}-2,3-dihydro-1,3-benzoxazol-2-one
1-{2-[3-(4-methylphenoxymethyl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
N-[(3S,4R)-4-propyl-1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)pyrrolidin-3-yl]methanesulfonamide
N-(2-hydroxyethyl)-5-(morpholin-4-ylmethyl)-N-(propan-2-yl)-1,2-oxazole-3-carboxamide
1-[3-ethyl-3-(hydroxymethyl)piperidin-1-yl]-3-(pyrazin-2-yl)propan-1-one
1-[4-(1,3-benzoxazol-2-yl)piperazin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
6-(benzyloxy)-4-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
1-{3-[3-(3-ethylphenoxy)azetidine-1-carbonyl]piperidin-1-yl}propan-1-one
2-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
N-{[2-(3-hydroxypiperidin-1-yl)-7-methylquinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]-4-(trifluoromethyl)benzamide
5-{[4-(1-benzofuran-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1-ethyl-1H-1,2,4-triazole
N-[3-(dimethylamino)propyl]-N-methyl-1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-3-amine
(2H-1,3-benzodioxol-4-ylmethyl)[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl](prop-2-en-1-yl)amine
3-(piperidin-1-ylmethyl)-1-(quinoxalin-2-yl)pyrrolidin-3-ol
1-{6-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pyridin-3-yl}ethan-1-one
3-(1-ethyl-1H-1,2,3-triazol-4-yl)-1-{3-[(5-methylpyridin-2-yl)amino]propyl}urea
N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
1-[(4aS,8aS)-7-benzyl-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-3-(methylsulfanyl)propan-1-one
1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-2-(2-methyl-1H-indol-3-yl)ethan-1-one
N-(butan-2-yl)-N-[(2-fluorophenyl)methyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
(2-{2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}-2-oxoethyl)urea
(2S)-4-methanesulfonyl-2-[(6-methoxy-3-methyl-1-benzofuran-2-yl)formamido]butanoic acid
4-{[(4-fluoro-3-methoxyphenyl)methyl]amino}-1-[(4-fluorophenyl)methyl]pyrrolidin-2-one
5-methoxy-3-methyl-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}-1H-indole-2-carboxamide
7-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
2-({[5-(hydroxymethyl)furan-2-yl]methyl}(thiophen-3-ylmethyl)amino)butan-1-ol
8-fluoro-2-{[4-(pyridin-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}quinolin-4-ol
(3aS,6aS)-2-benzyl-5-[(3-fluoro-2-hydroxyphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
9-(4-chloro-3-fluorobenzoyl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(benzylsulfanyl)ethyl]-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]-3-phenylpropanoic acid
(1R,3S)-3-methoxy-7-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]-7-azaspiro[3.5]nonan-1-ol
(1S,5R)-6-(cyclobutylmethyl)-3-[(1-methyl-1H-imidazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(5-ethyl-2-methylpyrimidin-4-yl)-4-(pyrimidin-2-yl)-1,4-diazepane
2-(2-aminoethyl)-N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-5,6-dimethylthieno[2,3-d]pyrimidin-4-amine
(3R,4S)-4-cyclopropyl-1-(1H-pyrazole-4-sulfonyl)pyrrolidin-3-amine