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5-(2-methylpropyl)-1'-(1H-pyrrole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
6-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-2,3,4,5-tetrahydropyridazin-3-one
N-(1H-imidazol-2-ylmethyl)-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
N-(4-cyano-2-ethylphenyl)-2-(1H-imidazol-4-ylmethyl)-3-oxopiperazine-1-carboxamide
3-[2-oxo-2-(7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-2-yl)ethyl]-1,2,3-oxadiazol-3-ium-5-olate
3-{2-[4-(2,3-dichlorophenyl)-1H-1,2,3-triazol-1-yl]ethyl}-1,3-oxazolidin-2-one
(2S,4S)-1-[(2-chlorophenyl)methyl]-4-{[(9-ethyl-9H-carbazol-3-yl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
1-ethyl-3-methyl-N-[3-(1H-1,2,4-triazol-1-yl)propyl]piperidine-3-carboxamide
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-3,6-dimethyl-N-(propan-2-yl)-1-benzofuran-2-carboxamide
(2R,6S)-4-{2-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-methyl-1H-1,2,4-triazol-5-yl]ethyl}-2,6-dimethylmorpholine
(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-6-[3-(methylsulfanyl)propyl]-3,6-diazabicyclo[3.2.2]nonane
N-{[1-({6-oxo-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-7-yl}methyl)piperidin-3-yl]methyl}acetamide
1-[(5-chlorofuran-2-yl)methyl]-4-(pyridin-3-yl)piperidin-4-ol
3-(azetidine-1-carbonyl)-N-[2-(pyrazin-2-yl)ethyl]benzene-1-sulfonamide
(2R)-2-hydroxy-1-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propan-1-one
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N,N-bis(prop-2-en-1-yl)acetamide
(3S,5S)-1-[(2-methoxyphenyl)methyl]-5-[(pyridin-2-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
8-(3,4-difluorobenzoyl)-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
3-{5-[2-(naphthalen-2-yloxy)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
6-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}quinoline
7-fluoro-N,2-dimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]quinoline-4-carboxamide
3-({[(2,4-dimethoxyphenyl)methyl]amino}methyl)-7-fluoro-1-(2-methylpropyl)-1,2-dihydroquinolin-2-one
N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-2-(1H-pyrazol-1-yl)butanamide
1-(4-methyl-2-{[2-(pyridin-3-yl)ethyl]amino}pyrimidin-5-yl)ethan-1-one
2-ethyl-4-methyl-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)-1,3-oxazole-5-carboxamide
1-[4-(4-methoxybenzoyl)piperazin-1-yl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
6-(2-chlorophenyl)-2-(3-{[methyl(propyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
N-(2,4-dimethylphenyl)-3-[2-(2-methyl-1,3-thiazol-4-yl)acetamido]propanamide
N-cyclohexyl-3-[1-(3-fluorophenyl)-1H-1,2,4-triazol-5-yl]-N-methylpropanamide
1-[4-methyl-2-({[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}amino)pyrimidin-5-yl]ethan-1-one
4-[4-(3-chlorophenyl)-1H-imidazol-2-yl]-1-cyclopentylpyrrolidin-2-one
N-[2-(3-ethylphenoxy)ethyl]-1-(2-methoxyacetyl)-N-methylpiperidine-3-carboxamide
5-[(4-fluorophenyl)methyl]-5-(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-4-yl)imidazolidine-2,4-dione
3-[(3R,4S)-3-cyclopropanesulfonamido-4-phenylpyrrolidin-1-yl]-N-methylpropanamide
N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
1-(4-methyl-2-{[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]amino}pyrimidin-5-yl)ethan-1-one
1-{5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidine-4-carboxamide
3-(4-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperazin-1-yl)benzonitrile
N-(cyclopropylmethyl)-4-[(3-methoxypropyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
3-(4-fluorophenoxymethyl)-1-{imidazo[1,2-a]pyrimidine-2-carbonyl}piperidine
(1S,5R)-3-(3-phenylpropyl)-6-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(1S,5R)-3-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-{[(1-phenylcyclopropyl)amino]methyl}piperidin-2-one
N-{[4-(methylsulfanyl)phenyl]methyl}-N-propyl-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
5-acetamido-1-ethyl-2-(2-fluorophenyl)-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1H-1,3-benzodiazole-7-carboxamide
(3ar,6ar)-N-[1-(2-phenylethyl)piperidin-4-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
3-(4-methoxyphenyl)-N-[(5-methyl-1H-imidazol-4-yl)methyl]-3-phenylpropanamide
N-(1H-indol-2-ylmethyl)-1-methyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-[5-({[(2-ethoxyphenyl)methyl](ethyl)amino}methyl)thiophen-3-yl]prop-2-yn-1-ol
[(4aS,8aR)-6-{2-methylthieno[3,2-d]pyrimidin-4-yl}-decahydro-1,6-naphthyridin-4a-yl]methanol