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4-[5-(3-cyanophenyl)-3-cyclopropyl-1H-1,2,4-triazol-1-yl]benzene-1-sulfonamide
9-({2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
N-(1-cycloheptylpiperidin-3-yl)-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetamide
3-(4-{[4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)-2,3-dihydro-1H-inden-1-one
N-[4-(morpholin-4-yl)butan-2-yl]thieno[2,3-d]pyrimidin-4-amine
{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}[1-(4-methylpiperazin-1-yl)propan-2-yl]amine
1-(6-{methyl[(3-phenyl-1,2-oxazol-5-yl)methyl]amino}pyridin-2-yl)ethan-1-ol
3-[5-(2-phenylpropyl)-1,2,4-oxadiazol-3-yl]pyridazine
(1S,4S)-2-(3-chlorophenyl)-5-(2-propyl-1,3-thiazole-4-carbonyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
N-(3,5-dimethoxyphenyl)-3-[1-(2-phenoxyacetyl)piperidin-3-yl]propanamide
methyl 1-[(4-amino-6,7-dimethoxyquinazolin-2-yl)methyl]piperidine-2-carboxylate
5-(methoxymethyl)-N-[(5-methylpyrazin-2-yl)methyl]furan-2-carboxamide
5-acetyl-N-[(5-tert-butyl-1,3-benzoxazol-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-({4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-4-(1H-pyrazol-1-yl)benzamide
1-{2-[5-(1-methyl-1H-pyrrol-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}pyrrolidin-2-one
4-(hydroxymethyl)-N-[3-(pyridin-3-yl)propyl]pyridine-2-carboxamide
3-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-5,6,7,8-tetrahydroquinoline
N-[(2-ethoxyphenyl)methyl]-3-(morpholin-4-yl)-N-(prop-2-en-1-yl)butanamide
(1R,5R)-3-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-6-propyl-3,6-diazabicyclo[3.2.2]nonane
N4-[1-(4-cyclopentyl-4H-1,2,4-triazol-3-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
5-{1-[2-(1H-imidazol-1-yl)ethyl]-1H-imidazol-2-yl}quinoline
{6-[3-(2-fluorophenoxymethyl)piperidine-1-carbonyl]pyridin-2-yl}methanol
7-fluoro-1-[2-(piperidin-1-yl)ethyl]-3-({[(trimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-1,2-dihydroquinolin-2-one
(1R,5R)-N,N-dimethyl-6-[4-(methylsulfanyl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
3-ethyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}pentanamide
3-cyclopropyl-5-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1-(2-phenylethyl)-1H-1,2,4-triazole
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-6-(2-methoxyphenyl)-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}pyridine-3-carboxamide
1-[(2E)-3-phenylprop-2-en-1-yl]-4-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazine
3-{2-[(3S,4S)-4-(4-fluorophenyl)-3-hydroxypiperidin-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
5-(2,4-difluorophenoxymethyl)-N-[3-(propan-2-yloxy)propyl]-1,2-oxazole-3-carboxamide
4-(cyclobutylsulfamoyl)-N-[2-(pyrazin-2-yl)ethyl]benzamide
4-{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,3λ6,4-oxathiazinane-3,3-dione
5-({3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)isoquinoline
2-[ethyl(methyl)amino]-1-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
4-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}benzonitrile
N-({3-methyl-7-[2-(phenylsulfanyl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)furan-2-carboxamide
1-[4-(3-methyl-1,2,4-oxadiazol-5-yl)phenyl]-3-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]urea
methyl (2S,4R)-4-(dimethylamino)-1-{[4-hydroxy-3-(methoxycarbonyl)phenyl]methyl}pyrrolidine-2-carboxylate
5-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}quinoxaline
(3S,4S)-4-cyclopropyl-1-{[3-(hydroxymethyl)-4-(propan-2-yloxy)phenyl]methyl}pyrrolidine-3-carboxylic acid
1-(oxan-4-ylmethyl)-3-[4-(propylsulfamoyl)phenyl]urea
2-(2,3-dimethoxyphenyl)-6,7-dimethoxyquinazolin-4-amine
methyl[(3-methyl-1,2-oxazol-5-yl)methyl](quinoxalin-2-ylmethyl)amine
4-ethyl-3-{1-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl}-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{imidazo[1,2-a]pyridine-2-carbonyl}-4-methanesulfonyl-1,4-diazepane
3-butyl-4-[2-(3,4-dihydro-2H-1,4-benzoxazin-4-yl)-2-oxoethyl]-1-methylpiperazin-2-one
N-{[3-(2-phenylethyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}benzamide
7-chloro-4-[(1R,5S,6S)-3-(furan-3-ylmethyl)-3-azabicyclo[3.1.0]hexane-6-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[1'-(5-ethyl-1,3,4-thiadiazol-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
N-{[3-(methylsulfanyl)phenyl]methyl}-9H-purin-6-amine