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N-[1-(2,4-dimethylphenyl)propyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-(2-{[3-(2-oxopyrrolidin-1-yl)propyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
3-(2-methoxyphenoxymethyl)-5-methyl-1-propyl-1H-1,2,4-triazole
1-{1-[6-(4-hydroxy-3-methoxyphenyl)pyridine-3-carbonyl]piperidin-3-yl}-3-methylbutan-1-one
5-ethyl-N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
N-[2-(1-methylpiperidin-3-yl)ethyl]-3-(1H-1,2,4-triazol-3-yl)benzamide
5-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidine-1-carbonyl]-2-methoxyphenol
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-{[(1-carbamoylethyl)(methyl)amino]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
(2S,4S)-N-ethyl-1-({[(2-fluorophenyl)methyl]carbamoyl}methyl)-4-propanamidopyrrolidine-2-carboxamide
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
1-(2-{[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)piperidine-3-carboxamide
4-[1-(4-fluorophenyl)-1H-pyrazol-4-yl]-N-{1-oxaspiro[4.4]nonan-3-yl}pyrimidin-2-amine
(3R,4S)-4-{4-[(3-chloro-4-ethoxyphenyl)methyl]-1,4-diazepan-1-yl}oxolan-3-ol
1-ethyl-6-methyl-N-[(5-methylpyrazin-2-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
ethyl 4-[(3-fluorophenyl)methyl]-1-[(2-hydroxy-6-methoxyphenyl)methyl]piperidine-4-carboxylate
{4-methyl-5-[1-(pyrimidin-2-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methanol
N-[2-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)ethyl]pyridine-3-carboxamide
4-[(2-phenylphenyl)methyl]-N-(pyridin-2-ylmethyl)piperazine-2-carboxamide
methyl[1-(pyridin-2-yl)ethyl]{[6-(trifluoromethyl)pyridin-3-yl]methyl}amine
(7R,9aR)-7-benzyl-N-(3-fluorophenyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
3-{[(5-methylthiophen-2-yl)methyl]({[5-(oxolan-2-yl)thiophen-2-yl]methyl})amino}propan-1-ol
1-[4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-4-(oxan-4-yl)piperazine
2-(3-methoxypropyl)-1-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)piperidine
N-[3-(1,3,6-trimethyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)phenyl]acetamide
3-(4-methylpiperazine-1-carbonyl)-N-[2-(1H-pyrazol-4-yl)ethyl]benzene-1-sulfonamide
4-{5-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidine-1-carbonyl]furan-2-yl}-2-methylbut-3-yn-2-ol
3-methyl-2-({4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}amino)butan-1-ol
{9-[(2-aminopyrimidin-5-yl)methyl]-3-(1H-pyrrole-3-carbonyl)-3,9-diazaspiro[5.5]undecan-1-yl}methanol
2-{2-[4-(pyridin-4-yl)piperidin-1-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
5-butyl-1'-(dimethyl-1,2-oxazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-[(3R,4S)-4-(dimethylamino)-1-{[3-(methylsulfanyl)phenyl]carbamoyl}piperidin-3-yl]propanoic acid
4-[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]-1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidine
(2-ethoxy-5-{[4-(4-fluorophenyl)-1,4-diazepan-1-yl]methyl}phenyl)methanol
5-chloro-2-{[4-(5,6-dimethylpyrimidin-4-yl)piperazin-1-yl]methyl}-3-methyl-1H-indole
5-(4-methylpiperidine-1-carbonyl)-N-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
4-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}-9,10-dihydroacridin-9-one
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
5-(cyclopropylamino)-N-[(4-fluorophenyl)methyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-(3-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-3-oxopropyl)methanesulfonamide
N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
N-cyclopentyl-N'-[(4-methylphenyl)methyl]-N'-(prop-2-yn-1-yl)butanediamide
(5S,9aS,9bS)-5-(2,1,3-benzothiadiazol-5-yl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-[2-chloro-5-(trifluoromethyl)phenyl]-1-(1,4-oxazepan-6-ylmethyl)urea
5-[(2-methyl-1H-imidazol-1-yl)methyl]-3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazole
N-[2-(ethanesulfonyl)ethyl]-2-(4,6,7-trimethyl-1-benzofuran-3-yl)acetamide
4-(oxolane-2-carbonyl)-N-(1,2,3-thiadiazol-5-yl)-1,4-diazepane-1-carboxamide
2-[2-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]benzonitrile
2-{2-oxo-2-[2-(1,3-thiazol-2-yl)piperidin-1-yl]ethyl}-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
1-(3-methoxypropyl)-3-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3R,4S)-3,4-dimethyl-1-[(4-methylpiperazin-1-yl)sulfonyl]piperidin-4-ol