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(2S,4R)-4-amino-1-[3-(benzyloxy)propyl]-N-methylpyrrolidine-2-carboxamide
(3-phenylprop-2-yn-1-yl)(prop-2-en-1-yl)(pyridin-3-ylmethyl)amine
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-3-phenyl-1H-pyrazole-4-carboxamide
(1S,6R)-9-{[4-(benzyloxy)phenyl]methyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
[4-(3,5-dichloro-4-methylbenzoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methanol
[3-(2-methoxyethyl)-1-[4-methyl-6-(methylamino)pyrimidin-2-yl]piperidin-3-yl]methanol
N-methyl-2-({5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-yl}amino)acetamide
N-benzyl-1,1-dioxo-N-(1,3-thiazol-2-ylmethyl)-1λ6-thiolane-3-carboxamide
N-butyl-4-{[(2,3-dimethoxyphenyl)methyl]amino}-N,5-dimethylthieno[2,3-d]pyrimidine-6-carboxamide
2-ethyl-4-methyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-1,3-oxazole-5-carboxamide
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]piperidine
N-ethyl-2,3-difluoro-N-[(3R,4R)-3-hydroxy-1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]benzamide
4-(1-{[(3,4-dimethylphenyl)methyl]amino}ethyl)hepta-1,6-dien-4-ol
4-amino-1-[3-(2,6-dimethylphenoxy)azetidin-1-yl]-3-hydroxybutan-1-one
(2E)-N-{2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}-2-methylbut-2-enamide
6-cyano-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)pyridine-3-carboxamide
2-{1-[3-(methylsulfanyl)propyl]piperidin-2-yl}pyridine
4-(hydroxymethyl)-1-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-ol
2-(1-benzofuran-2-yl)-5-chloropyrazine
1-[4-(5-methylfuran-2-yl)phenyl]-2-(morpholin-4-yl)ethan-1-ol
N-[(4-methoxyphenyl)methyl]-3-(1-methylpiperidin-4-yl)-N-propylpropanamide
3-(1H-1,3-benzodiazol-1-yl)-1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
5-cyclopentyl-3-[2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)ethyl]-1,2,4-oxadiazole
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}[(1-ethyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl)amine
N-methyl-2-phenyl-N-(pyrazin-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-{6-[(piperidin-4-yl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-3-carboxamide
3-{4-[(3-ethyl-4-methylpiperazin-1-yl)methyl]-1H-pyrazol-1-yl}propanoic acid
N,5-diethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]thiophene-3-carboxamide
[5-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]methanol
(2S)-1-(pyridazine-4-carbonyl)-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
3-(1-methyl-1H-pyrazol-5-yl)-1-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]urea
2-methyl-6-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-1,3-benzothiazole
ethyl 4-(cyclopropylmethyl)-1-(2-methyl-1H-1,3-benzodiazole-6-carbonyl)piperidine-4-carboxylate
methyl (2S,4R)-4-(dimethylamino)-1-[2-(2-methyl-1H-1,3-benzodiazol-5-yl)acetyl]pyrrolidine-2-carboxylate
2-{2-oxo-2-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]ethyl}-1,2-dihydrophthalazin-1-one
4-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}morpholine
5-benzyl-4-methanesulfonyl-1-(4-methylphenyl)piperazin-2-one
1-(2-methoxyethyl)-3-{[(3-methylphenyl)carbamoyl]methyl}-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
(1S,3R)-3-{4-[(2-fluorophenyl)methyl]piperidine-1-carbonyl}cyclohexan-1-amine
{3-methyl-1-[3-(3-methylbutyl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]-1-oxobutan-2-yl}urea
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-cyclopropyl-1-{1-[(2-ethylphenyl)methyl]piperidin-4-yl}piperidine-3-carboxamide
N-(2-{2-methyl-7-oxo-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-6-yl}ethyl)pyridine-4-carboxamide
4'-[2-(2-hydroxyethoxy)ethyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-(2-ethyl-1H-imidazol-1-yl)-1-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[3-(methylsulfanyl)propyl]amine
5-{1-[1-(pyridin-3-yl)propan-2-yl]-1H-imidazol-2-yl}-2-(thiophen-2-yl)pyrimidine
4-[4-(2,5-dimethylthiophen-3-yl)-1H-imidazol-2-yl]-1-(2-methylpropyl)pyrrolidin-2-one
2-(5-fluoro-2-methoxyphenyl)-2-(4-methanesulfonylpiperazin-1-yl)acetic acid
2-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]pyridine-3-carboxamide