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2-(5-chloro-3-methyl-1H-indole-2-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
1-cyclopropyl-4-[4-(2-methoxybenzoyl)piperazine-1-carbonyl]pyrrolidin-2-one
8-[2-(4-hydroxyphenyl)acetyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
{3-[2-(1-cycloheptanecarbonylpiperidin-4-yl)-1H-imidazol-1-yl]propyl}dimethylamine
methyl({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amine
2-(1-methyl-3-oxopiperazin-2-yl)-N-[3-(propan-2-yloxy)propyl]acetamide
4-[4-(1H-imidazol-1-yl)phenyl]phenol
2-(cyclopropylmethyl)-7-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2-[(prop-2-en-1-yl)amino]benzamide
5-fluoro-3-methyl-2-[2-(trifluoromethyl)morpholine-4-carbonyl]-1H-indole
2-(4-chlorophenyl)-4-[4-(4H-1,2,4-triazol-4-yl)benzoyl]morpholine
N-{[2-(2-methoxyphenyl)pyrimidin-5-yl]methyl}-N-methyloxan-4-amine
1-{5-[(3-hydroxyphenyl)methyl]-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-3-ol
4-(5-fluoro-2-methylphenyl)-3-[3-(morpholin-4-yl)propyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S)-1-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N-[4-(1,3-thiazol-4-yl)phenyl]pyrrolidine-2-carboxamide
(1R,3S,5S)-3-(4-methoxyphenyl)-8-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-8-azabicyclo[3.2.1]octane
(2S,4S)-1-cyclopropanecarbonyl-N-ethyl-4-[2-(2-methyl-1,3-thiazol-4-yl)acetamido]pyrrolidine-2-carboxamide
1-[(2-fluoro-4-methoxyphenyl)methyl]-2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidine
(3aS,7aR)-2-(5-cyclopropyl-1,2-oxazole-3-carbonyl)-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
N-{2-[1-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)piperidin-2-yl]ethyl}acetamide
2-[4-(furan-2-carbonyl)piperazine-1-carbonyl]morpholine
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-(methylamino)pyridine-4-carboxamide
4-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-1-[2-(piperidin-1-yl)ethyl]-1,2,3,6-tetrahydropyridine
1-[(5-propylfuran-2-yl)methyl]-4-(pyridin-3-ylmethyl)piperazine
(3aR,6aS)-N-(4-methyl-2-oxo-1,2-dihydroquinolin-7-yl)-octahydropyrrolo[3,4-c]pyrrole-2-carboxamide
N-[(3S,4R)-1-(3-chloro-4-hydroxybenzoyl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
2-{[1-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]oxy}pyrimidine
3-[4-(furan-2-carbonyl)-1,4-diazepane-1-carbonyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazole
1-cycloheptyl-4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
2-(3-methylbutyl)-8-(quinoxalin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
N4-[1-(4-methylphenoxy)propan-2-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-(2-{[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]methyl}phenoxy)-3-(thiomorpholin-4-yl)propan-2-ol
3-(1-butyl-1H-imidazol-2-yl)-1-[4-(pyrrolidin-1-yl)benzoyl]piperidine
8-(2,5-dimethoxyphenyl)-2-(pyrrolidin-1-yl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-3-(1H-1,2,4-triazol-1-yl)propanamide
5-[6-amino-5-cyano-4-(5-cyano-1-methyl-1H-pyrrol-3-yl)pyridin-2-yl]thiophene-3-carboxylic acid
1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
1-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
N'-cycloheptyl-N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-N-methylbutanediamide
2-(5-acetylthiophen-3-yl)-N-[1-methyl-4-(propan-2-yloxy)-1H-indazol-3-yl]acetamide
methyl 2-(5-methyl-2-{[(3-methyl-4-oxo-3,4-dihydrophthalazin-1-yl)formamido]methyl}-2,3-dihydro-1-benzofuran-7-yl)benzoate
1-(1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-4-carbonyl)piperidin-4-ol
ethyl 4-{1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperidin-3-yl}piperazine-1-carboxylate
4-[3-carboxy-6-(4-fluorophenyl)pyridin-2-yl]morpholine-2-carboxylic acid
2-(1-{[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-amine
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[4-(3-methoxybenzoyl)piperazin-1-yl]propan-1-one
N-(2,3-dihydroxypropyl)-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
2-cyclopropanecarbonyl-8-(3-phenoxypropyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-(6-ethyl-2-methylpyrimidin-4-yl)-N-[3-(pyridin-3-yl)propyl]piperidin-4-amine