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6-(2,5-dimethylphenyl)-N-[2-(1H-imidazol-2-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[2-(1H-imidazol-1-yl)ethyl]-5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-methylpyridin-2-amine
1-(3-methylpyridin-4-yl)-4-[1-(propan-2-yl)piperidine-4-carbonyl]piperazine
4-acetamido-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]butanamide
5-{2-[4-(4-methoxypyrimidin-2-yl)piperazin-1-yl]-2-oxoethyl}-2,6-dimethyl-3,4-dihydropyrimidin-4-one
N-({3-methyl-7-[3-(3-methylphenyl)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)oxolane-2-carboxamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
4-methoxy-N-{[1-(5-methylpyrazine-2-carbonyl)piperidin-3-yl]methyl}benzene-1-sulfonamide
1-cyclopentyl-4-(1H-imidazol-2-ylmethyl)-1,4-diazepane
(4aR,7aS)-N,N-dimethyl-4-[2-(methylamino)pyridine-4-carbonyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N-{5-[2-(3-methylphenoxy)ethyl]-1,3,4-thiadiazol-2-yl}-2-(1,2,3,6-tetrahydropyridin-4-yl)acetamide
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2-methyl-2-(methylamino)propanamide
2-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-ethyl-N-methylpropanamide
3-(diphenylmethyl)-N-(1,2-oxazol-3-ylmethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
5-(methoxymethyl)-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-N-(2-phenylethyl)-1H-pyrazole-4-carboxamide
4-[2-(5-amino-3-methyl-1H-pyrazol-1-yl)acetyl]-1-(2-methylphenyl)piperazin-2-one
3-(2H-1,3-benzodioxol-5-yl)-N-[2-(methylsulfanyl)ethyl]-3-phenylpropanamide
N-cyclopentyl-N-[(5-methylthiophen-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
2-(2-chlorophenyl)-1-[(3S,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]ethan-1-one
1-[4-(3-hydroxyphenyl)piperazin-1-yl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one
N-benzyl-1-(furan-2-ylmethyl)-N-(1,3-thiazol-2-ylmethyl)piperidine-4-carboxamide
6-[(3-methyl-3-phenylpiperidin-1-yl)sulfonyl]-3,4-dihydro-2H-1,4-benzoxazin-3-one
(4aS,8aR)-1-(2-aminoethyl)-6-[(1-phenyl-1H-pyrazol-5-yl)methyl]-decahydro-1,6-naphthyridin-2-one
N-{[4-methyl-2-(propan-2-yl)-1,3-thiazol-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
methyl({[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl})(quinolin-5-ylmethyl)amine
7-(1H-inden-2-yl)-4-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
7-(5-chloropyridin-2-yl)-4-(2-propoxyethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-[3-({methyl[(3-methylthiophen-2-yl)methyl]amino}methyl)piperidin-1-yl]ethan-1-ol
4-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N,N-dimethylbenzamide
7-(5-chloro-2-methoxyphenyl)-9-methoxy-4-(1H-pyrazole-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-benzyl-2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidine-1-sulfonamide
3-(2-methoxyethyl)-1-(pyrimidin-2-yl)piperidine-3-carboxylic acid
N-(4-carbamoyl-3-chlorophenyl)-4-(cyclopropylmethyl)-3-(2-hydroxyethyl)piperazine-1-carboxamide
2-methyl-5-{3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl}pyrazine
2-methyl-3-[(4-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}piperidin-4-yl)oxy]pyridine
2-[1-(3-methylbut-2-en-1-yl)-4-(4-methylquinolin-2-yl)piperazin-2-yl]ethan-1-ol
1-[(1-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperidin-4-yl)methyl]pyrrolidin-2-one
{2-[4-(4-chlorobenzoyl)morpholin-2-yl]ethyl}dimethylamine
2-methyl-4-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}-5-propylpyrimidine
N,3-dimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-methyl-N-(quinolin-4-ylmethyl)-1H-pyrazole-4-carboxamide
1-(3-chlorophenyl)-4-[2-(2-fluorophenyl)acetyl]piperazin-2-one
5-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2-methylphenol
1-(2-{3-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)-4-phenylpyrrolidin-2-one
2-(2-methoxyethyl)-8-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
3-[4-(3-cyanophenyl)piperidine-1-carbonyl]piperidine-1-carboxamide
(5S)-5-[({[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(pyridin-2-ylmethyl)amino)methyl]pyrrolidin-2-one
4-methoxy-N-{1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
{1-[({[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)methyl]cyclopropyl}methanol
4-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-1,4-diazepane