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3-[(3S,7S,8aS)-3-[(2S)-butan-2-yl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-fluorophenyl)urea
2-chloro-4-{[(cyclopropylmethyl)(2-methoxyethyl)carbamoyl]amino}benzamide
{1-[6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-yl]-3-(2-phenylethyl)piperidin-3-yl}methanol
3-[1-(cyclohex-1-en-1-yl)ethyl]-1-{4-[2-(morpholin-4-yl)-2-oxoethoxy]phenyl}urea
(1S,3R)-3-amino-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]cyclopentane-1-carboxamide
2-(2,3-difluorophenoxymethyl)-N-methyl-N-(2-phenylethyl)-1,3-oxazole-4-carboxamide
N-{[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}morpholine-2-carboxamide
1-(2-methoxyphenyl)-5-[1-(2-methyl-1H-imidazol-1-yl)ethyl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
dimethyl({[(3S,4R)-4-(propan-2-yl)-1-(1H-1,2,4-triazole-5-carbonyl)pyrrolidin-3-yl]sulfamoyl})amine
5-(3-chloro-4-methoxyphenyl)-3-methyl-2-(4H-1,2,4-triazol-4-yl)pyridine
N-(1-ethoxy-2-methylpropan-2-yl)-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
(3S,4S)-1-[(2-chloro-5-methoxy-4-propoxyphenyl)methyl]piperidine-3,4-diol
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
1-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
N-(4-{1-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-1H-1,2,3-triazol-4-yl}phenyl)acetamide
2-[(3-{[1-(3,4-dimethoxyphenyl)propyl]carbamoyl}phenyl)amino]acetic acid
4-cyclopentyl-N-[1-(pyridin-4-yl)propyl]pyrimidin-2-amine
ethyl[(2-fluoro-4-methoxyphenyl)methyl](oxan-4-ylmethyl)amine
7-(2-methoxyacetamido)-N,1-dimethyl-2-phenyl-N-(quinoxalin-6-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
4-(2,5-dimethylfuran-3-carbonyl)-1-methyl-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
1-(5-chloro-2-oxo-1,2-dihydropyridine-3-carbonyl)-4-methylpiperidine-4-carboxylic acid
(3aR,7aS)-2-[1-methyl-3-(thiophen-2-yl)-1H-pyrazole-5-carbonyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-5-methyl-1,2-oxazole-3-carboxamide
5-[3-(propan-2-yl)phenoxy]-1-azabicyclo[3.2.1]octane
3-cyclopropyl-5-(thiophene-2-carbonyl)-1H-1,2,4-triazole
methyl 4-{[(4aR,8aS)-2-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}-decahydro-1,6-naphthyridin-6-yl]methyl}benzoate
(2R)-2-cyclohexyl-2-hydroxy-1-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}ethan-1-one
5-(2-fluoro-6-methoxyphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
4-{5-[3-cyclopropyl-1-(4-fluorophenyl)-1H-1,2,4-triazol-5-yl]pyrimidin-2-yl}morpholine
methyl[2-(pyrazin-2-yloxy)hex-5-en-1-yl](pyridin-3-ylmethyl)amine
1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
3-fluoro-N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
(1S,5R)-3-(5-chloropyridin-2-yl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(3-{[(2,2-dimethyloxan-4-yl)(methyl)amino]methyl}phenoxy)acetamide
1-phenyl-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
5-methyl-N-{4-[3-(1,2-oxazolidin-2-yl)propanamido]phenyl}furan-2-carboxamide
(1S,5R)-3-benzyl-6-(5-methyl-1,3-oxazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-amino-5-methyl-4-(4-methyl-1H-imidazol-5-yl)-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
3-chloro-N-(2-hydroxyethyl)-N-(1,3-thiazol-2-ylmethyl)-1H-indole-2-carboxamide
N-[(1-cyclohexylpiperidin-3-yl)methyl]-2-(phenylsulfanyl)-N-(pyridin-3-ylmethyl)acetamide
9-(2-aminopyridine-4-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
3-{[4-(2-methoxyacetyl)-1,4-diazepan-1-yl]methyl}-8-methyl-1,2-dihydroquinolin-2-one
[(2E)-2-methylbut-2-en-1-yl][(1-methylpiperidin-3-yl)methyl](2-phenylethyl)amine
N-{[4-(oxolan-2-ylmethoxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)-2H-1,3-benzodioxole-5-carboxamide
3-{2-[(3,4-dimethoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[2-(1H-indol-3-yl)ethyl]propanamide
2-{2-[1-(adamantane-1-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]acetamide
(3aR,7aS)-2-{2-[(6-methylpyridazin-3-yl)oxy]hex-5-en-1-yl}-2,3,3a,4,7,7a-hexahydro-1H-isoindole
4-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}-1-(pyridin-3-ylmethyl)pyrrolidin-2-one