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2-(2-fluorophenoxymethyl)-N-methyl-N-[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1,3-oxazole-4-carboxamide
N-[3-(3-chlorophenyl)phenyl]-1-(5-methyl-1H-pyrazole-3-carbonyl)piperidine-4-carboxamide
({5-[1-butyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]furan-2-yl}methyl)dimethylamine
3-(1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-N-(oxolan-2-ylmethyl)propanamide
N-cyclopropyl-4-{[2-(quinolin-8-yloxy)ethyl]amino}pyridine-2-carboxamide
N-(2-{[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]methyl}propyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}pyridine-3-carboxamide
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-[(trifluoromethyl)sulfanyl]ethan-1-one
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methyl-6-(pyridin-4-yl)pyridine-3-carboxamide
N-[(3,4-difluorophenyl)methyl]-3-[1-(oxane-4-carbonyl)piperidin-3-yl]propanamide
{1-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(3-methylbut-2-en-1-yl)piperidin-3-yl}methanol
({4-cyclopropyl-5-[1-(pyrrolidine-1-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
6-oxo-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-N-(prop-2-en-1-yl)-1,4,5,6-tetrahydropyridazine-3-carboxamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-(1H-indol-4-ylmethyl)acetamide
3-(2-aminoethyl)-4-(2,5-dimethoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[4-({methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)thiophen-2-yl]ethan-1-one
4-{4-[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]-1H-1,2,3-triazol-1-yl}butan-1-ol
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methyl-3-(1H-pyrazol-1-ylmethyl)benzamide
(3R,4R)-1-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-4-cyclopropyl-3-methylpiperidin-4-ol
N-(furan-2-ylmethyl)-N-(2-hydroxyethyl)-3-methyl-5-propyl-1-benzofuran-2-carboxamide
5-ethyl-5-(piperidin-4-yl)imidazolidine-2,4-dione
N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}-2-methanesulfonylacetamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
4-[hydroxy(thiophen-2-yl)methyl]-N-(6-methylpyridin-3-yl)piperidine-1-carboxamide
(3S,4S)-4-propyl-1-(quinolin-4-ylmethyl)pyrrolidine-3-carboxylic acid
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1H-1,3-benzodiazole-5-carboxamide
5-[4-(1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-N-cyclohexyl-1-cyclopropyl-4-oxo-1,4-dihydropyridine-3-carboxamide
3-[(3R,4S)-1-{2-[methyl(phenyl)amino]acetyl}-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]-3,6-dimethyl-1-benzofuran-2-carboxamide
N,3-dimethyl-4-oxo-N-(quinolin-5-ylmethyl)-3,4-dihydroquinazoline-7-carboxamide
2-(pyridin-3-yl)-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]acetamide
4-[(1-cyclopentylpiperidin-4-yl)oxy]-3-methoxy-N-(oxolan-3-yl)benzamide
N-(6-methylpyridin-3-yl)-1-[3-(2-oxo-1,2-dihydropyridin-1-yl)propanoyl]piperazine-2-carboxamide
9-(3-propyl-1H-pyrazole-4-carbonyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(4aR,7aS)-1-(2-methoxyacetyl)-4-[(2E)-3-phenylprop-2-en-1-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-propyl-8-(1H-pyrazole-3-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-3-methylfuran-2-carboxamide
(1S,5R)-3-methyl-6-[4-(2-phenylethoxy)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-2-(dimethylamino)-N-methyl-2-(2-methylphenyl)acetamide
1-[(2,3-dimethylphenyl)methyl]-3-(3-methyl-1,2,4-thiadiazol-5-yl)urea
N-cyclohexyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]imidazo[1,2-a]pyridine-6-carboxamide
N-[2-(prop-2-en-1-yloxy)phenyl]-4-(thian-4-yl)piperazine-1-carboxamide
4-[2-(ethylamino)pyrimidine-5-carbonyl]-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
3-amino-1-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}pyrrolidine-3-carboxylic acid
2-(3-methylphenyl)-5-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]pyrimidin-4-ol
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(9H-purin-6-yl)piperidin-3-ol
(1-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methanol
1-(2,4-dimethoxybenzoyl)-4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
5-[4-(1H-pyrazol-1-yl)phenyl]pyrazin-2-amine