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3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]propanamide
5-cyclobutyl-1-[(3-methoxyphenyl)methyl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
3-[(2-methylprop-2-en-1-yl)oxy]-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]benzamide
6-(benzyloxy)-1-(oxan-4-ylmethyl)-4-propyl-1,4-diazepan-2-one
1-[1-(4-fluorophenyl)-2,2-dimethylcyclopropanecarbonyl]-4-(pyrrolidine-1-carbonyl)piperidine
1-[4-(2-phenoxyethyl)piperazin-1-yl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]({imidazo[1,2-a]pyrimidin-6-ylmethyl})(2-methoxyethyl)amine
3-chloro-6-methyl-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
4-(4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1H-imidazol-2-yl}-1H-1,2,3-triazol-1-yl)piperidine
(3R,4R)-4-amino-1-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)piperidin-3-ol
2-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidine-1-carbonyl]benzonitrile
N-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)ethyl]-3-(5-methylfuran-2-yl)benzamide
5-methyl-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}-1-propyl-1H-pyrazole-4-carboxamide
4-phenyl-1-[6-(pyrrolidin-1-yl)pyridine-3-carbonyl]azepane
1,3-dimethyl-N-[(3-methylpyridin-4-yl)methyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
5-({[2-(ethylamino)pyrimidin-5-yl]formamido}methyl)thiophene-2-carboxylic acid
1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-3-(naphthalene-1-carbonyl)piperidine
1-(1-methyl-1H-pyrrole-2-carbonyl)-3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
N3-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-N1,N1-dimethylpiperidine-1,3-dicarboxamide
9-(cyclopropylmethyl)-4-[(4-methoxyphenyl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-ethyl-3-[3-(propan-2-yloxy)benzoyl]piperidine-1-carboxamide
1-(2-{[(2,3-difluoro-6-methoxyphenyl)methyl](methyl)amino}ethyl)piperidin-2-one
2-[2-(1H-pyrazol-1-yl)ethyl]-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidine
4-{[3-(trifluoromethoxy)phenyl]methyl}-1,3λ6,4-oxathiazinane-3,3-dione
N-(2,3-dimethylphenyl)-3-oxo-3-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}propanamide
4-[5-({4-[(4-fluorophenyl)methyl]piperidin-1-yl}methyl)-1,3-thiazol-2-yl]morpholine
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](1H-imidazol-4-ylmethyl)(2-methoxyethyl)amine
2-(3-methoxypropyl)-8-(4-methylpyrimidin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
3-(2-methoxyphenyl)-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
N-(2,4-difluorophenyl)-3-({methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)benzamide
3-({[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]amino}methyl)-7-fluoro-1-(2-phenylethyl)-1,2-dihydroquinolin-2-one
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-[4-(1H-pyrazol-5-yl)phenyl]piperidine-3-carboxamide
ethyl 5-{[3-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylate
(1R,5R)-3-(5-methoxy-1H-indole-2-carbonyl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-3-(4-oxo-3,4-dihydroquinazolin-3-yl)propanamide
7-[2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)acetyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
1-methyl-4-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
(1R,2S)-2-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-N-methylcyclohexane-1-carboxamide
5-methyl-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-methyl-3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)-N-(oxan-2-ylmethyl)propanamide
ethyl 3-[(2-fluorophenyl)methyl]-1-[2-(methylsulfanyl)acetyl]piperidine-3-carboxylate
7-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-(2-ethylphenyl)-3-(2-methanesulfonylacetamido)benzamide
N-[2-(2,4-difluorophenyl)-1-[1-(1-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]ethyl]-N-methylpyridine-3-carboxamide
N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}-2-(1H-imidazol-4-yl)acetamide
2-methyl-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]oxane-2-carboxamide
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-2-(3-methyl-1H-pyrazol-1-yl)acetamide
3-{[(4-fluorophenyl)methyl]sulfanyl}-1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-[2-(2,4-dimethoxyphenyl)ethyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide