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N-methyl-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]acetamide
3-[(3R,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3,5-dimethylphenyl)urea
(4aS,7aR)-1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-4-methanesulfonyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N'-(2,5-dimethoxyphenyl)-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]propanediamide
2-{3-azaspiro[5.5]undecan-9-yl}-7-methyl-2,7-diazaspiro[4.5]decan-6-one
methyl 4-[2-(1-phenylethyl)-1H-imidazol-1-yl]butanoate
2-cyclobutanecarbonyl-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
2-[1-(3-methylbutyl)-4-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}piperazin-2-yl]ethan-1-ol
(1S,5R)-3-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-acetyl-N-(1,2-oxazol-3-ylmethyl)thiophene-3-carboxamide
6-methyl-N-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
2-(2-methoxy-4-methylphenoxymethyl)-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,3-oxazole-4-carboxamide
2-{3-[1-(pyridin-4-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyrazine
N-methyl-N-{4-[3-methyl-1-(2-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]phenyl}methanesulfonamide
N-[(1-{[1-(propan-2-yl)piperidin-4-yl]methyl}pyrrolidin-3-yl)methyl]methanesulfonamide
3-[4-(3-methylphenyl)piperazin-1-yl]-N-[3-(4H-1,2,4-triazol-4-yl)propyl]propanamide
2-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-6-methoxyphenol
N,N-dimethyl-2-(pyridin-2-yl)-7-[(2S)-pyrrolidine-2-carbonyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(3aR,6aR)-2-(3-methoxy-5-methylthiophene-2-carbonyl)-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-3-(piperidine-1-carbonyl)benzene-1-sulfonamide
5-(2-chlorophenyl)-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]furan-2-carboxamide
3-cyclopropyl-5-[(dimethyl-1,3-thiazol-4-yl)methyl]-1-(4-methanesulfonylphenyl)-1H-1,2,4-triazole
4-(1-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}azetidin-3-yl)morpholine
2-(dimethylamino)-2-(2-fluorophenyl)-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]acetamide
N-cyclopropyl-3-(1-{[4-(2-hydroxyethoxy)phenyl]methyl}piperidin-4-yl)propanamide
1-{4-[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-1,4-diazepan-1-yl}ethan-1-one
7-[2-(pyrrolidin-1-yl)benzoyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
1-(3-{[(2-phenoxyethyl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]({[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl})methylamine
2-(1H-imidazol-1-yl)-1-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]ethan-1-one
5-(3-methylthiophen-2-yl)-4-phenyl-1H-imidazole
N-({3-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]phenyl}methyl)propanamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-1-(2-methoxyethyl)piperidine-4-carboxamide
1-(4-{4-cyclopropyl-5-[(dimethylamino)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(pyrrolidin-1-yl)ethan-1-one
N-methyl-4-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}-4-oxobutanamide
2-[(2-fluorophenyl)methyl]-4-(4-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperazin-1-yl)-2,3-dihydro-1H-isoindole-1,3-dione
1-(3-methoxybenzoyl)-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
2-amino-N-[(3S,4R)-4-ethoxyoxolan-3-yl]-1,3-benzothiazole-5-carboxamide
N'-(3-ethylphenyl)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}butanediamide
7-(1-benzothiophen-3-yl)-9-[2-(pyridin-2-yl)ethoxy]-4-(1H-pyrrol-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-methyl-5-[2-(propan-2-yl)-1H-imidazol-1-yl]furan-2-carboxamide
ethyl 1-[(2,4-difluorophenyl)carbamoyl]-3-[(2,4-difluorophenyl)methyl]piperidine-3-carboxylate
2-[3-(propan-2-yl)-5-[5-(propan-2-yl)-1,3-oxazol-4-yl]-1H-1,2,4-triazol-1-yl]pyridine
1-({1-[(6-chloro-2-fluoro-3-methylphenyl)methyl]pyrrolidin-3-yl}methyl)-3-ethylurea
(2S)-2-amino-N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}propanamide
1-[1-(5,6-dimethylpyrimidin-4-yl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
1-methyl-3-(1,3,4-thiadiazol-2-yl)-1-{[3-(trifluoromethyl)phenyl]methyl}urea
7-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-2-oxa-7-azaspiro[4.5]decan-8-one
2-(1-{1-[(3-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}pyrrolidin-2-yl)pyridine
N'-(2-ethoxyphenyl)-N-[(4-methyl-1,3-benzoxazol-2-yl)methyl]propanediamide