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2-(4-fluoro-3-{6-[(pyridin-4-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)acetic acid
(1R,5R)-3-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
3-({[1-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperidin-4-yl]oxy}methyl)pyridine
8-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-methyl-1-(quinolin-4-ylmethyl)-1,4-diazepan-5-one
2-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-1-(piperidin-1-yl)ethan-1-one
(1S,5R)-3-benzoyl-6-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(2S,4R)-1-(naphthalen-1-ylmethyl)-N-(propan-2-yl)-4-[(propan-2-yl)amino]pyrrolidine-2-carboxamide
2-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]pyrrolidin-3-yl}acetic acid
methyl 4-({3-[(2-methoxyethyl)carbamoyl]-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)benzoate
2-ethyl-9-(5-ethyl-1,2,4-oxadiazol-3-yl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
4-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2-dihydroquinolin-2-one
7-(1-benzothiophen-3-yl)-4-[(2-ethylpyrimidin-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[2-(2-ethyl-1,3-thiazol-4-yl)ethyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-N-methyl-N-(propan-2-yl)acetamide
(4aR,8aS)-N,N-dimethyl-1-(2,4,5-trifluorobenzoyl)-decahydro-1,6-naphthyridine-6-sulfonamide
2-{9-ethyl-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}acetic acid
methyl 8-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-1-ethoxy-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-3-propyl-1H-pyrazole-4-carboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-[(4-methoxyphenyl)amino]-2-methylpropanamide
1-(2,6-dimethylpyridine-4-carbonyl)-3-phenylpiperazine
8-(but-3-en-1-yl)-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
1-[2-(methylsulfanyl)pyridine-3-carbonyl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamide
methyl({[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl})(pyridin-3-ylmethyl)amine
2-amino-6-(2-amino-4-methyl-1,3-thiazol-5-yl)-4-(1-ethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
4-({1-[3-(1H-pyrrol-1-yl)propanoyl]pyrrolidin-3-yl}methyl)benzoic acid
N-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-3-(1,2-oxazinan-2-yl)propanamide
2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]morpholine
1-cycloheptyl-N-[3-(1H-indol-1-yl)propyl]-6-oxopiperidine-3-carboxamide
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[1-(1,3-thiazol-2-yl)ethyl]benzamide
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-6-methyl-2-propylpyrimidin-4-amine
3-(2-phenylethyl)-5-[1-(1H-1,2,4-triazol-1-yl)ethyl]-1H-1,2,4-triazole
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2-(pyrrolidin-1-yl)pyrimidine-5-carboxamide
3-butyl-4-[4-(3-hydroxy-3-methylbutyl)benzoyl]-1-methylpiperazin-2-one
1-[1-(2,1,3-benzothiadiazol-5-ylmethyl)-4-phenylpiperidin-4-yl]ethan-1-one
2-(5-chloropyridin-2-yl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-(1-cyclopentyl-1H-pyrazol-5-yl)-4-{imidazo[1,2-b]pyridazin-6-yl}piperazine-1-carboxamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
4-[2-(benzyloxy)ethyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-[(5-propylfuran-2-yl)methyl]pyrrolidin-3-yl]methanol
(1H-imidazol-4-ylmethyl)({[2-(2-methylphenoxy)pyridin-3-yl]methyl})amine
(3S,4R)-1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-phenylpyrrolidine-3-carboxylic acid
6-methoxy-3-{[2-(pyridin-2-yl)piperidin-1-yl]methyl}-1H-indazole
(3aR,6aR)-2-acetyl-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
5-cyano-N-[(3S,5S)-5-(ethylcarbamoyl)-1-(2-methylpropyl)pyrrolidin-3-yl]-2-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
3-{1-[(4-phenyl-1,3-thiazol-5-yl)methyl]-1H-1,2,3-triazol-4-yl}phenol
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-6-cyclopropyl-3-methyl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
(1R,3S)-7-(4-cyclopentylpyrimidin-2-yl)-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-1-ol