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8-chloro-2-{[({1-[ethyl(methyl)amino]cyclopentyl}methyl)amino]methyl}quinolin-4-ol
{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}[1-(furan-2-yl)ethyl]methylamine
N-propyl-5-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}pyrimidin-2-amine
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-[1-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-amine
7-fluoro-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]quinazolin-4-amine
3-[(ethylamino)methyl]-6,7-dimethoxy-1-[(4-methylphenyl)methyl]-1,2-dihydroquinolin-2-one
2-({methyl[1-(pyridin-2-yl)propyl]amino}methyl)benzonitrile
N,4-dimethyl-6-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyrimidin-2-amine
ethyl 1-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
N-({1-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]-4-hydroxyazepan-4-yl}methyl)methanesulfonamide
2-[5-methyl-4-(2-methylpiperidine-1-carbonyl)-1H-pyrazol-1-yl]-4-(thiophen-2-yl)pyrimidine
3-{1-[1-methyl-5-(thiophen-2-yl)-1H-pyrazole-3-carbonyl]piperidin-3-yl}benzoic acid
3-hydroxy-1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
4-(5-{4-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}-1H-pyrazol-3-yl)phenol
2-methoxy-6-[(2-methyl-4-phenylpiperazin-1-yl)methyl]phenol
1-methyl-4-(2-{[4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}ethyl)piperidin-4-ol
1-(furan-2-ylmethyl)-N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)piperidine-3-carboxamide
N-[(2R,3R)-1'-cyclopentanecarbonyl-2-(pyridin-2-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl](methyl)[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amine
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
[7-chloro-5-(5-fluoropyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
3-methyl-1-{1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carbonyl}piperazine
1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-4-(3-methylphenoxy)piperidine
N4-methyl-N4-[(3-phenyl-1H-pyrazol-5-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
3-(3-methoxyphenyl)-N-[(1-methylpiperidin-3-yl)methyl]propanamide
N-{4-[1-(2,2,2-trifluoroethyl)-1H-imidazol-2-yl]phenyl}acetamide
4-{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-{4-[1-(2-phenylethyl)pyrrolidin-3-yl]piperidin-1-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one
5-cyclopropyl-N-[2-(diethylamino)ethyl]-N-ethyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
4-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-2-(4-methylpentyl)morpholine
N-cyclopropyl-2-(3-methyl-2-oxo-1,2-dihydroquinoxalin-1-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
3-(2-oxo-2-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}ethyl)-3-phenyl-1-(thiophen-2-ylmethyl)pyrrolidine-2,5-dione
7-({[(3-ethyl-1,2-oxazol-5-yl)methyl](methyl)amino}methyl)-4-methyl-2H-chromen-2-one
N-ethyl-4-hydroxy-3-methoxy-N-(oxan-4-ylmethyl)benzamide
1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-3-(1H-imidazol-1-ylmethyl)piperidine
3-(4-chloro-1H-pyrazol-1-yl)-1-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}propan-1-one
2-amino-N-{2-[4-(trifluoromethoxy)phenyl]phenyl}acetamide
3-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-[1-(5-methylthiophene-2-carbonyl)piperidin-4-yl]-5-propylimidazolidine-2,4-dione
N-[(2-chloro-6-fluorophenyl)methyl]-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
3-[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]-N-(2-hydroxy-2-phenylethyl)-N-methylpropanamide
2-{1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]piperidin-2-yl}pyridine
(3aS,7aR)-5-methyl-2-[2-methyl-6-(2-methylpropyl)pyrimidine-4-carbonyl]-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
N-(4-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazine-7-carbonyl}phenyl)ethane-1-sulfonamide
3-(3-chlorophenyl)-3-(3-hydroxyphenyl)-1-[4-(methoxymethyl)piperidin-1-yl]propan-1-one
(3R,4S)-4-cyclopropyl-1-(2-methyl-1H-pyrrole-3-carbonyl)pyrrolidin-3-amine
6-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-3-carbonitrile
5-{3-[1-(2-propoxyethyl)-1H-pyrazol-3-yl]phenyl}pyrimidine
4-hydroxy-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-2-(phenoxymethyl)pyrimidine-5-carboxamide