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3-[(3S)-3-hydroxy-3-phenylpropyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-6-methoxypyrimidin-2-amine
2-(2-{[methyl(pyridin-4-ylmethyl)amino]methyl}phenyl)-3H,4H,5H,6H,7H,8H,9H-cyclohepta[d]pyrimidin-4-one
N-methyl-2-(phenylamino)-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}pyrimidine-5-carboxamide
1-ethyl-3-(oxan-4-yl)-5-[2-(trimethyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,4-triazole
N-cyclopentyl-N-[(2,5-dimethoxyphenyl)methyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
(2R,6R)-4-(4,4,4-trifluorobutanoyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
4-[3-(2-ethylphenoxy)azetidine-1-carbonyl]quinoline
6-(2-ethoxyphenyl)-2H-1,3-benzodioxole-5-carboxamide
1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidine
1-[(2,6-difluorophenyl)methyl]-3-[(dimethylamino)methyl]pyrrolidin-3-ol
5-[2-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)ethyl]-3-(2-methylphenyl)-1,2,4-oxadiazole
2-[3-(pyridin-2-yl)-1H-pyrazol-1-yl]-N-[1-(thiophen-2-ylmethyl)-1H-pyrazol-5-yl]acetamide
3-({5-[(2E)-but-2-en-2-yl]-4-phenyl-1H-imidazol-1-yl}methyl)pyridine
2-(5-ethyl-1-benzofuran-3-yl)-1-[4-(pyridin-3-ylmethyl)piperazin-1-yl]ethan-1-one
3-[2-(4-fluorophenyl)morpholin-4-yl]-1-(4-methylpiperidin-1-yl)propan-1-one
2-{4-[2-(dimethylamino)-2-(3-fluorophenyl)acetyl]piperazin-1-yl}benzonitrile
4-{1-[(7-methoxy-2-oxo-1,2-dihydroquinolin-3-yl)methyl]piperidin-3-yl}benzoic acid
4-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-3-(4-fluorophenyl)piperazin-2-one
(2R,6R)-11-methoxy-4-[2-oxo-2-(piperidin-1-yl)ethyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidine
2-{1-[2-(1H-imidazol-2-yl)benzoyl]pyrrolidin-2-yl}-6-methyl-1H-1,3-benzodiazole
4-[2-(2-methyl-1H-1,3-benzodiazol-1-yl)acetyl]-1-(4-methylphenyl)piperazin-2-one
4-{4-[(1,4-dioxan-2-ylmethyl)amino]piperidin-1-yl}-N,N,6-trimethylpyrimidin-2-amine
N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
5-cyclopropanecarbonyl-1'-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(2,5-dioxoimidazolidin-1-yl)-N-[(2-ethoxypyridin-3-yl)methyl]acetamide
5-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2-dihydropyridin-2-one
3-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]-2-ethyl-6-methyl-1-[(5-methylfuran-2-yl)methyl]-1,4-dihydropyridin-4-one
[4-({pyrazolo[1,5-a]pyridin-3-ylmethyl}sulfamoyl)phenyl]urea
(3R,5S)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(2-methylpropyl)-5-(morpholin-4-ylmethyl)piperidine-3-carboxamide
2-methyl-4-(4-{[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}phenyl)but-3-yn-2-ol
1-{3-[3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]propyl}piperidine
({3-[(4-ethylpiperazin-1-yl)methyl]-2,5-dimethylphenyl}methyl)(methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
1-ethyl-N-methyl-5-oxo-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)pyrrolidine-3-carboxamide
(oxolan-2-ylmethyl)(pyridin-2-ylmethyl){[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amine
N-{1-[1-(1H-indole-5-carbonyl)piperidin-4-yl]-2-phenylethyl}-N-methylthiophene-3-carboxamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(4-fluorophenoxy)acetamide
2-{cyclopropyl[4-(1-methyl-3-phenyl-1H-pyrazol-4-yl)-1H-1,2,3-triazol-1-yl]methyl}-4-methylpyridine
2-cyclohexyl-7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
3-(4-ethyl-1H-pyrazol-5-yl)-1-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]piperidine
5-(1-benzofuran-2-yl)-N-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1,2,4-triazin-3-amine
[(2S)-1-[(1-benzylpiperidin-2-yl)methyl]pyrrolidin-2-yl]methanol
3-[(4aR,7aS)-6,6-dioxo-4-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
1-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}-3-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
N3-benzyl-N5-(butan-2-yl)-1-cyclopentyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
9-[(4-methoxypyridin-2-yl)methyl]-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-ethyl-1'-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
8-[(2,3-dimethyl-1H-indol-7-yl)methyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
(1,4-dioxan-2-ylmethyl)({[7-(methylsulfanyl)-2-{[3-(trifluoromethyl)phenyl]methoxy}quinolin-3-yl]methyl})amine