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4-[(2-methoxyphenyl)methyl]-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-{1-[3-(4-methyl-1H-pyrazol-1-yl)propyl]pyrrolidin-2-yl}pyridine
methyl 2-[1-(cyclopentylcarbamoyl)propyl]-1-oxo-1,2-dihydroisoquinoline-7-carboxylate
N-methyl-N-[2-(2-methyl-1H-indol-1-yl)ethyl]-2-(methylamino)pyridine-4-carboxamide
3-[3-(pyridin-2-yl)azetidine-1-carbonyl]-1λ6-thiolane-1,1-dione
(3S,5R)-1-[(3-fluorophenyl)methyl]-5-(4-methylpiperazine-1-carbonyl)piperidine-3-carboxylic acid
dimethyl[3-(2-{1-[4-(prop-2-en-1-yl)benzoyl]piperidin-3-yl}-1H-imidazol-1-yl)propyl]amine
(5-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}-1-ethyl-1H-1,2,4-triazol-3-yl)(phenyl)methanol
(3S,7S,8aS)-7-(benzylamino)-3-[(1R)-1-hydroxyethyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
6-methyl-2-(2-phenylethyl)-3-(piperidine-1-carbonyl)-1-(pyridin-4-ylmethyl)-1,4-dihydropyridin-4-one
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
1-benzyl-N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]-1H-pyrazole-4-carboxamide
1-[2-(methylamino)pyridine-3-carbonyl]-4-phenylpiperidine-4-carbonitrile
N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-2-(morpholin-2-yl)acetamide
3-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-1-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)urea
1-[2-(2-methyl-1H-1,3-benzodiazol-5-yl)acetyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-amino-4-(2,2-dimethyloxan-4-yl)-6-(3,4,5-trifluorophenyl)pyridine-3-carbonitrile
N-(2-hydroxyethyl)-5-{pyrazolo[1,5-a]pyridine-3-carbonyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-[4-({[2-(2,4-dimethylphenoxy)ethyl](methyl)amino}methyl)phenyl]ethan-1-one
(2S,4R)-4-[4-(4-fluoro-2-methylbenzenesulfonamidomethyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
4-(1H-imidazol-4-ylmethyl)-1-(2-phenylethyl)piperazin-2-one
(1S,5R)-3-(2,1,3-benzoxadiazol-4-ylmethyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[3-chloro-4-(propylcarbamoyl)phenyl]-3-cyanopiperidine-1-carboxamide
3-{[2-(1H-imidazol-1-yl)ethyl]sulfamoyl}-N-(pyridin-3-yl)benzamide
(1R,9aR)-1-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-octahydro-1H-quinolizin-1-ol
2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-(pyridin-4-ylmethyl)acetamide
3-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-1-(5-methyl-2,1,3-benzothiadiazol-4-yl)urea
N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-4,5,6,7-tetrahydro-1,2-benzoxazole-3-carboxamide
5-ethyl-4-[4-(oxolan-2-ylmethyl)piperazin-1-yl]pyrimidin-2-amine
N-({1-cyclohexyl-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl}methyl)acetamide
8-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1,3-dioxa-8-azaspiro[4.5]decan-2-one
8-[4-(3-hydroxypiperidin-1-yl)pyrimidin-2-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
5-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}-1-ethyl-1H-indole
4-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-1,4-oxazepan-6-ol
N-methyl-2-(morpholin-4-yl)-N-[2-(phenylsulfanyl)ethyl]-2-(pyridin-3-yl)acetamide
N2-benzyl-6-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-yl]-1,3,5-triazine-2,4-diamine
3-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-ol
N-[2-methyl-2-(morpholin-4-ylmethyl)propyl]-1-(pyridin-2-ylmethyl)piperidin-3-amine
(3R,4S)-4-cyclopropyl-1-[3-(pyrrolidin-1-yl)pyrazin-2-yl]pyrrolidin-3-amine
[(3-methyl-1H-indol-2-yl)methyl]({1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl})amine
(1S,5R)-6-(pyridin-2-ylmethyl)-3-[2-(thiophen-2-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
ethyl 4-[4-(1-propyl-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxylate
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-(1,2-oxazol-3-ylmethyl)piperidine-3-carboxamide
3-(5-carbamoylthiophen-3-yl)benzoic acid
N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
2-{1-[2-(ethylamino)pyrimidine-5-carbonyl]pyrrolidin-3-yl}benzoic acid
N-[(3,5-dimethoxyphenyl)methyl]-1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide