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4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]-1-[(5-ethylfuran-2-yl)methyl]piperidine
1-[2-(furan-2-yl)ethyl]-2-(3-methylthiophen-2-yl)-1H-imidazole
N-[(2S)-1-hydroxy-3-phenylpropan-2-yl]-3,6-dimethyl-1-benzofuran-2-carboxamide
1-[4-(4-fluorophenoxy)piperidin-1-yl]-2-(morpholin-3-yl)ethan-1-one
methyl({[7-methyl-2-(morpholin-4-yl)quinolin-3-yl]methyl})[(5-methylfuran-2-yl)methyl]amine
N-[2-(dimethylamino)-2-(2-methylphenyl)ethyl]-5-phenyl-1,2-oxazole-4-carboxamide
1-{[(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)carbamoyl]methyl}piperidine-4-carboxamide
2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}piperidine
2-(1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)-1,2,3,4-tetrahydroisoquinoline
3-ethyl-3-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-1-[2-(2-oxo-1,3-oxazolidin-3-yl)phenyl]urea
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(methylamino)acetamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-(2-phenoxyethyl)-4-(pyridin-4-yl)piperazine
4-methoxy-2-{4-[(1-propyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}pyrimidine
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
methyl 4-methyl-1-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidine-4-carboxylate
2-[4-(morpholin-4-ylmethyl)phenyl]-6-(2-phenylethyl)-3,4-dihydropyrimidin-4-one
8-fluoro-2-{[3-(3-methoxybenzoyl)piperidin-1-yl]methyl}quinoline
N,N,5-trimethyl-2-[4-(prop-2-en-1-yl)piperazin-1-yl]pyrimidin-4-amine
N-benzyl-2-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]acetamide
3-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]-1-[2-(methylsulfamoyl)phenyl]urea
1-(cyclopropylmethyl)-N-[2-(4-methoxyphenyl)phenyl]pyrrolidine-2-carboxamide
8-[(2-ethoxyphenyl)methyl]-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
3-(2H-1,3-benzodioxol-5-ylmethyl)-N-(2,3-dihydro-1H-inden-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
2-[1-(3-ethyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]-6-methyl-1H-1,3-benzodiazole
5-benzyl-5-{3-[4-(2-fluorophenoxy)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-3-(1H-pyrazol-1-yl)benzamide
1-[2-(5-chloro-2-methoxypyridin-4-yl)pyridine-4-carbonyl]-4-methylpiperazine
2-(1-cyclohexylpiperidin-4-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
({5-methanesulfonyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)(methyl)[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]amine
methyl 2-[methyl({[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl})carbamoyl]piperidine-1-carboxylate
3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
1,3,7-trimethyl-2-[4-(thian-4-yl)piperazine-1-carbonyl]-1H-indole
N-(3-hydroxypropyl)-1-{1-[(4-phenylphenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
5-[1-(1H-imidazol-2-ylmethyl)pyrrolidin-2-yl]-3-(propan-2-yl)-1,2,4-oxadiazole
7-(2-methylphenyl)-4-(oxane-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-hydroxy-N-[3-(1,3-thiazol-4-yl)phenyl]-1-oxa-8-azaspiro[4.5]decane-8-carboxamide
1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-phenylpiperidine
3-{[7-(3-cyclopropyl-1,2-oxazole-5-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}pyridine
(3aS,6aR)-5-(3-methoxypyrazin-2-yl)-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]-1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperidine
N-{4-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-4-oxobutyl}acetamide
(3S,4R)-N,N-dimethyl-1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-4-(4-methylphenyl)pyrrolidin-3-amine
N-[(4-chlorophenyl)methyl]-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-cyclopropyl-1-(1-{[4-(propan-2-yl)phenyl]methyl}piperidin-4-yl)piperidine-3-carboxamide
2-({[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)amino}methyl)benzoic acid
methyl({[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl})(thiophen-3-ylmethyl)amine
3-[(2R,3R,6R)-5-[(5-fluoro-2-methoxyphenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
1-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}but-2-yn-1-one
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-3-(1,2-oxazinan-2-yl)propanamide