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2-(3,4-dimethoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(4aS,7aR)-1-[(4-methyl-1,3-thiazol-5-yl)methyl]-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-benzyl-4-(3-phenylbenzoyl)piperazin-2-one
8-(2,5-dimethylfuran-3-carbonyl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
2-ethyl-N-[(3R,5S)-5-(ethylcarbamoyl)-1-[2-(methylsulfanyl)acetyl]pyrrolidin-3-yl]pyridine-4-carboxamide
N-(1-{1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)oxolane-3-carboxamide
3-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}-4,5-dihydro-1,2-oxazole-5-carboxamide
(2R,4S)-1-[2-(2,5-dimethoxyphenyl)acetyl]-4-hydroxypiperidine-2-carboxylic acid
4-({1-[3-(4-fluorophenyl)propyl]piperidin-2-yl}methyl)morpholine
ethyl 5-(thiophene-2-carbonyl)-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
9-[3-(4-hydroxyphenyl)propanoyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-cyclopentyl-N-[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
2-{[(3S,4S)-3,4-bis(hydroxymethyl)pyrrolidin-1-yl]methyl}-5,8-dimethylquinolin-4-ol
7-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
methyl 4-[4-(oxolane-3-carbonyl)piperazin-1-yl]benzoate
3-{2-methyl-[1,2,4]triazolo[1,5-a]pyridin-8-yl}-1-(oxolan-2-ylmethyl)-1-(pyridin-2-ylmethyl)urea
{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}(4-phenylbutan-2-yl)amine
5-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-2-(propan-2-yl)-3,4-dihydropyrimidin-4-one
7-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
3-(1-benzofuran-2-yl)-1-benzyl-4-{[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}-1H-pyrazole
5-methyl-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1,3,4-oxadiazol-2-amine
N-ethyl-4-(6-oxo-1,6-dihydropyridin-3-yl)benzamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[3-(furan-2-yl)propyl]-1-methylpiperidine-2-carboxamide
4-[2-(aminomethyl)-1H,2H-naphtho[2,1-b]furan-7-yl]-2-methoxypyridine-3-carbonitrile
(2S,4S)-4-amino-1-[3-(cyclooctylcarbamoyl)propanoyl]-N-methylpyrrolidine-2-carboxamide
3-[3-(2-amino-1,3-thiazol-4-yl)propyl]-1-[3-(propan-2-yloxy)phenyl]urea
N-cyclopropyl-N-({4-[3-(1,3-dioxo-2,3-dihydro-1H-isoindol-2-yl)propoxy]phenyl}methyl)-2-(trifluoromethyl)benzamide
1-[(4-fluorophenyl)methyl]-4-(thiophen-3-ylmethyl)-1,4-diazepane
(3S,4R)-3-ethyl-4-methyl-1-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]piperidin-4-ol
4-(4-{[(5-methylpyrazin-2-yl)methyl]amino}piperidin-1-yl)-N-[2-(morpholin-4-yl)ethyl]benzamide
N-[1-(6-chloropyridazin-3-yl)piperidin-4-yl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
N2,N2,N4-trimethyl-N4-[(5-propyl-1H-pyrazol-3-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
3-(2-{1-[(3-fluoro-2-methoxyphenyl)methyl]piperidin-2-yl}ethyl)phenol
5-(2-chloro-4-fluorophenoxymethyl)-N-(furan-2-ylmethyl)-N-(prop-2-yn-1-yl)-1,2-oxazole-3-carboxamide
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(4-methyl-1H-imidazol-5-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
2-{2-[3-(1,2-oxazinan-2-yl)propanamido]ethyl}-1,3-thiazole-4-carboxylic acid
2-[4-(3-cyanophenyl)-3-oxopiperazin-1-yl]-N-(1,3-dimethyl-1H-pyrazol-4-yl)acetamide
[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl](oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
N-(2-cyclopentylethyl)-5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-amine
1-(2-{1-[(2S)-2-hydroxy-3-phenylpropanoyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
3-methyl-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)thiophene-2-carboxamide
(2S,4S)-4-({[3-(benzyloxy)phenyl]methyl}amino)-1-(2,3-dihydro-1H-inden-2-yl)-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
2-cyclopentyl-9-[3-(dimethylamino)benzoyl]-2,9-diazaspiro[5.5]undecan-3-one
1-{5-acetyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propan-1-one
2-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}(methyl)amino)acetamide
(3S,4R)-N,N-dimethyl-4-(4-methylphenyl)-1-(thiophene-2-sulfonyl)pyrrolidin-3-amine
(2S)-1-{[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}pyrrolidine-2-carboxamide
1-ethyl-N-methyl-3-(2-methylpropyl)-N-(quinolin-5-ylmethyl)-1H-pyrazole-5-carboxamide
[1-(2,6-diaminopyrimidin-4-yl)-3-(3-phenylpropyl)piperidin-3-yl]methanol