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6-(8-methylquinolin-5-yl)pyrazine-2-carboxylic acid
4-[2-(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}phenyl)-1,3-oxazol-5-yl]-N,N-dimethylaniline
N-cyclopropyl-2-{1-[(4-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}acetamide
(3R,4S)-1-[1-(4-methoxyphenyl)cyclopropanecarbonyl]-4-(propan-2-yl)pyrrolidin-3-amine
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-[(dimethylcarbamoyl)amino]acetamide
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-(1,4-dioxan-2-ylmethyl)-5-methyl-1H-pyrazole-4-carboxamide
2-{[4-(1-methyl-1H-1,2,3,4-tetrazol-5-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}ethan-1-ol
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(1H-pyrazol-1-yl)propan-1-one
N-[(3S,4R)-1-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
2-(dimethyl-1,2-oxazol-4-yl)-2-({[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)acetic acid
ethyl 2-{1-[(3-methylquinoxalin-2-yl)methyl]piperidin-2-yl}acetate
1-(2-{[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]amino}pyrimidin-4-yl)piperidin-4-ol
7-methyl-3-{[4-(thiophen-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-indole
N-{[7-fluoro-2-(2-methoxyphenyl)quinolin-3-yl]methyl}-1,3-dimethyl-N-(oxolan-2-ylmethyl)-1H-pyrazole-5-carboxamide
3-chloro-5-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
N3-cyclohexyl-N5-ethyl-N3-methyl-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
4-(pyridin-3-yl)-N-[2-(pyridin-3-yloxy)propyl]pyrimidin-2-amine
(2S,4S)-4-amino-1-[2-(3,4-dimethoxyphenyl)acetyl]-N,N-diethylpyrrolidine-2-carboxamide
5-[1-(2,3-dihydro-1-benzofuran-7-carbonyl)pyrrolidin-2-yl]-N,N-dimethylthiophene-2-carboxamide
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]benzamide
4-[7-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]morpholine
4-(3-{[1-(furan-3-carbonyl)piperidin-4-yl]oxy}benzoyl)morpholine
5-ethyl-1'-(2-fluoro-6-methoxybenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-[(3-fluoro-4-methoxyphenyl)methyl]-N-[3-(1H-imidazol-1-yl)propyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[2-(2-oxopiperidin-1-yl)ethyl]-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
1-(4-aminopyrimidin-2-yl)-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylic acid
2-(4-chloro-3-methyl-1H-pyrazol-1-yl)-N-methyl-N-[1-(pyridin-2-yl)propan-2-yl]acetamide
3,5-dimethyl-4-{[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methyl}-1,2-oxazole
1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
5-[2-(2-fluorophenyl)benzoyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-[6-oxo-4-(piperidin-1-yl)-1,6-dihydropyridazin-1-yl]-N-[2-(propylsulfanyl)phenyl]acetamide
N-(2-chlorophenyl)-3-{1-[(3-ethyl-1,2-oxazol-5-yl)methyl]piperidin-4-yl}propanamide
3-[4-(4-fluorophenyl)piperazine-1-carbonyl]-2,6-dimethylquinoline
(3aR,6aR)-2-(cyclobutylmethyl)-5-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-cyclopropyl-2-[3-oxo-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-9-yl]pyridine-4-carboxamide
N-(2-hydroxyethyl)-4-(1H-pyrazol-4-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]butanamide
6-[4-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]pyrazine-2-carboxamide
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
(2R)-2-({[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}amino)propanamide
(2S,4S)-N-ethyl-1-(furan-3-carbonyl)-4-hexanamidopyrrolidine-2-carboxamide
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-propyl-1,3-thiazole-4-carboxamide
1-(4-{[2-(ethylsulfanyl)ethyl]amino}-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
3-(2-ethylbutyl)-8-[2-(morpholin-4-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{[6-chloro-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}-2,5-dimethylthiophene-3-sulfonamide
N-[(2R,3R)-1'-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
3-chloro-N-cyclopentyl-4-{[1-(thiophene-2-carbonyl)piperidin-4-yl]oxy}benzamide
[(3R,4S)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-[(1-propyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl]methanol
2-amino-3-ethyl-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-(1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-3-yl)-N-methylacetamide