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N3-cyclooctyl-1-(2-methylpropyl)-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-(pyrazin-2-yl)pyrrolidin-3-amine
1-(diethylamino)-3-(2-methoxy-4-{[(2-phenylethyl)amino]methyl}phenoxy)propan-2-ol
N-{[1-(4-fluorophenyl)pyrrolidin-3-yl]methyl}-4-methylpyrimidin-2-amine
N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-methyl-N-[(5-methylfuran-2-yl)methyl]-1H-pyrazole-3-carboxamide
3-chloro-N-[2-(dimethylamino)ethyl]-4-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}oxy)benzamide
2,2-dimethylpropyl 3-oxo-2,8-diazaspiro[4.5]decane-8-carboxylate
N-[(3R,4S)-4-cyclopropyl-1-[methyl(phenyl)carbamoyl]pyrrolidin-3-yl]-5-hydroxypyrazine-2-carboxamide
4-(2-oxo-2-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}ethyl)-1,2,3,6-tetrahydropyridazine-3,6-dione
methyl (2S)-2-cyclopropyl-2-{[2-(dimethylamino)-6-methylpyrimidin-4-yl]amino}acetate
N-ethyl-6-(3-fluorophenyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
7-butoxy-4-(2-methoxypyrimidin-5-yl)-1,2,3,4-tetrahydroquinolin-2-one
4-[1-(5-chloro-2,3-dimethoxyphenyl)-3-(pyrimidin-5-yl)prop-2-yn-1-yl]morpholine
4-{[2-(3,4-dimethoxyphenyl)ethyl]amino}-N-(1-hydroxy-2-methylpropan-2-yl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
1,6-dimethyl-N-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[2-(4-methoxyphenyl)ethyl]-6-oxo-N-[2-(pyrazin-2-yl)ethyl]piperidine-3-carboxamide
3-[1-(2,3,4-trifluorobenzoyl)piperidin-3-yl]benzoic acid
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-5-[(methylsulfanyl)methyl]furan-2-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-2-(dimethylamino)-1-[4-hydroxy-4-(hydroxymethyl)piperidin-1-yl]ethan-1-one
5-methyl-N-(2-{4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)-3-phenyl-1,2-oxazole-4-carboxamide
2-(cyclopropylmethyl)-7-[(6-hydroxy-1,4-oxazepan-6-yl)methyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
5-chloro-2-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyridine
(furan-2-ylmethyl)[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl](thiophen-3-ylmethyl)amine
9-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[4-(2,4-diethoxy-3-methylphenyl)-3-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-1-yl]acetic acid
N-methyl-N-[(5-phenyl-1H-pyrazol-3-yl)methyl]-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
3-hydroxy-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)propanamide
N-(4-{[4-(3-methoxybenzoyl)piperazin-1-yl]methyl}phenyl)acetamide
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
4-[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]pyridine
2-[(2-amino-6-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-yl)amino]ethan-1-ol
(2S,4R)-4-(2-methoxybenzamido)-N-(pyridin-2-ylmethyl)pyrrolidine-2-carboxamide
2-(4-fluorophenyl)-1-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
N-{[1-({5-[(N-methylmethanesulfonamido)methyl]furan-2-yl}methyl)piperidin-4-yl]methyl}acetamide
(3S,5R,9R)-5-hydroxy-11-[(4-methoxyphenyl)methyl]-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
ethyl 2-[({[2-(2,3-difluoro-4-methylphenoxy)pyridin-3-yl]methyl}carbamoyl)amino]acetate
N-[4-(2,2-dimethylpropanamido)-3-methoxyphenyl]-2-hydroxy-3-(2-methylphenoxy)propanamide
(1s,4s)-4-hydroxy-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]cyclohexane-1-carboxamide
2-ethyl-1-[4-(3-{[4-(furan-2-carbonyl)piperazin-1-yl]methyl}phenoxy)piperidin-1-yl]butan-1-one
7-(cyclobutylmethyl)-2-[2-(methylsulfanyl)pyrimidin-4-yl]-2,7-diazaspiro[4.5]decan-6-one
1-[3-(6-hydroxypyrimidin-4-yl)piperidin-1-yl]-2-[1-(propan-2-yl)piperidin-4-yl]ethan-1-one
2-[2-({2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}amino)pyrimidin-4-yl]pyridine-4-carboxylic acid
[5-(2-amino-5-ethylpyrimidin-4-yl)-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]methanol
4-{1-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]piperidin-4-yl}thiomorpholine
[1-(4-tert-butylbenzoyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
N-{4-[(4aR,8aS)-6-benzoyl-decahydro-1,6-naphthyridine-1-carbonyl]phenyl}acetamide
1-acetyl-N-[2-(pyridin-3-yloxy)propyl]piperidine-4-carboxamide
2-(ethylsulfanyl)-1-[4-(4-methoxyphenoxy)piperidin-1-yl]propan-1-one
1-[(2-butoxy-3-methoxyphenyl)methyl]piperidine-4-carboxamide