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5-(dimethylamino)-2-({9-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-2,3-dihydropyridazin-3-one
5-[(2-methoxyphenyl)methyl]-3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
ethyl 4-(3-{[(1-methoxypropan-2-yl)amino]methyl}-6-methylquinolin-2-yl)piperazine-1-carboxylate
N-[(1-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methyl]acetamide
4-[(4-fluorophenyl)methyl]-N-(furan-2-ylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carboxamide
N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
2-cyclobutanecarbonyl-N-(1-phenylethyl)-1,2,3,4-tetrahydroisoquinoline-8-sulfonamide
1-{1-[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]ethyl}-3-(1H-1,2,3,4-tetrazol-5-yl)urea
2-methyl-3-[4-(2-phenoxyethyl)piperazine-1-carbonyl]-1,2,3,4-tetrahydroisoquinoline
(1-{2-[5-(5-ethylpyridin-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}piperidin-3-yl)methanol
(3R,5S)-1-[(4-hydroxyphenyl)methyl]-5-[(4-methylpiperazin-1-yl)methyl]-N-(oxolan-2-ylmethyl)piperidine-3-carboxamide
1-(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(pyrimidin-2-yl)-1,4-diazepane
N-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
N-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-N-[(1-methyl-1H-imidazol-2-yl)methyl]cyclopropanamine
(1R,3S)-7-[4-(pyrrolidin-1-ylmethyl)benzoyl]-7-azaspiro[3.5]nonane-1,3-diol
(3S,9aR)-3-(2-methylpropyl)-8-(naphthalene-2-sulfonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
{[2-(2,2-dimethylpropanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}[2-(1H-indol-1-yl)ethyl]methylamine
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
N-[2-(2-fluorophenyl)ethyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
2-({[(3R,4R)-4-(hydroxymethyl)-1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-N-[(5-methyl-1H-imidazol-4-yl)methyl]piperidin-4-amine
4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-[(3-fluorophenyl)methyl]piperidine
5-chloro-3-[4-(3,6-dimethylpyrazin-2-yl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
(1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)methanol
6-fluoro-2-oxo-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-[4-(1H-imidazol-1-yl)benzoyl]-4-(2-methanesulfonylethyl)piperazine
(3R,5S)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
1-[(3S,5S)-5-[1-(2,3-dihydro-1H-inden-2-yl)-1H-1,2,4-triazol-5-yl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylic acid
3-{3-[3-(piperidine-1-carbonyl)-5-(1,3-thiazole-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-1-yl]propyl}pyridine
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)butanamide
N-methyl-N-[1-methyl-1-(methylcarbamoyl)ethyl]-2-[(4-methylphenyl)sulfanyl]propanamide
1-cyclopentanecarbonyl-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
2-benzyl-8-[(2R,4S)-4-hydroxypyrrolidine-2-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]acetamide
1-(5-{3-[2-(4-methoxyphenyl)ethyl]piperidine-1-carbonyl}thiophen-2-yl)ethan-1-one
3-{5-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1,3,4-thiadiazol-2-yl}-1-[(5-methylfuran-2-yl)methyl]urea
1-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-3-(hydroxymethyl)pyrrolidin-3-ol
1-(1H-indazol-5-yl)-4-[2-(methylsulfanyl)benzoyl]piperazin-2-one
6-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridine-1-carbonyl]piperazin-2-one
5-propyl-4-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
(4S)-4-(methoxymethyl)-3,3-dimethyl-1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidin-4-ol
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1-phenyl-1H-1,2,3-triazole-4-carboxamide
N4-ethyl-N2-methyl-N2-[2-(pyridin-2-yl)ethyl]pyrimidine-2,4-diamine
3-(3-fluorophenyl)-N-[2-(2-methoxyphenyl)ethyl]-1H-pyrazole-4-carboxamide
(4aR,8aR)-2-cyclopentanecarbonyl-7-[(6-methyl-1H-1,3-benzodiazol-2-yl)methyl]-decahydro-2,7-naphthyridin-4a-ol
1-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-3-(1H-imidazol-1-yl)propan-1-one
3-[(3R,4S)-4-(dimethylamino)-1-(pyridin-4-ylmethyl)piperidin-3-yl]propan-1-ol
N-[1-(1-cyclopentanecarbonylpiperidin-4-yl)-1H-pyrazol-5-yl]-3-methylbutanamide
1-[(1R,5R)-6-{[4-(trifluoromethyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
(2S,4S)-N-ethyl-1-(1,3-thiazol-2-ylmethyl)-4-[2-(thiophen-2-yl)acetamido]pyrrolidine-2-carboxamide