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1-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-(1H-pyrazol-1-yl)propan-1-one
4-(4-methyl-1H-pyrrole-2-carbonyl)piperazine-2-carboxylic acid
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(2-methoxyacetyl)pyrrolidine-3-carboxylic acid
3-(methoxymethyl)-1-{[4-(methylsulfanyl)phenyl]methyl}pyrrolidine
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N,1,4,6-tetramethyl-N-[2-(2-methylpiperidin-1-yl)ethyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
4-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-oxo-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
1-{1-[5-(5-ethylfuran-2-yl)-4-phenyl-1H-imidazol-1-yl]propan-2-yl}-1H-1,2,4-triazole
5-{4-[(2-cyanophenyl)methyl]piperazin-1-yl}-1-ethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-(3,4-difluorophenyl)-1-[4-(propan-2-yl)-1,2,3-thiadiazole-5-carbonyl]piperidin-3-amine
1-(4-methylphenyl)-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclopropane-1-carboxamide
2-({4-phenyl-5-[1-(pyridin-2-yl)-1H-pyrrol-2-yl]-1H-imidazol-1-yl}methyl)morpholine
2-{1,9-dioxaspiro[5.5]undecan-4-yl}-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine
5-(cyclooctylamino)-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-ethyl-N-(2-hydroxyethyl)-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1H-pyrazole-3-carboxamide
3-(2H-1,3-benzodioxol-5-yl)-N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
{4-[3-(2-methylphenyl)benzoyl]morpholin-2-yl}methanamine
2-cyclopropyl-N-[2-(dimethylamino)ethyl]-N-(oxolan-2-ylmethyl)quinoline-4-carboxamide
1-[4-(cyclopropylamino)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-2-(4-methyl-1,4-diazepan-1-yl)ethan-1-one
2-oxo-2-[9-oxo-8-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-2-yl]acetamide
8-methoxy-N-{3-[(5-methylpyridin-2-yl)amino]propyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]-1,2,3-thiadiazole-4-carboxamide
4-(4-chlorophenoxy)-N-[4-(1H-pyrazol-1-yl)butan-2-yl]piperidine-4-carboxamide
N-{[2-(2-methoxyethyl)pyrimidin-5-yl]methyl}-N-methyl-1-(2-phenylethyl)piperidin-3-amine
N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-2-(phenylamino)pyrimidine-5-carboxamide
3-ethyl-1-(1-oxo-1,2-dihydroisoquinoline-4-carbonyl)piperidine-3-carboxylic acid
{3-[1-(3-chlorophenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]propyl}dimethylamine
N-(furan-2-ylmethyl)-4-oxo-N-(prop-2-yn-1-yl)-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
4-(1-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)pyrimidin-2-amine
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperazine
4-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-(1H-imidazol-2-ylmethyl)-N-methylbenzamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
1-benzyl-4-[(3-methylquinoxalin-2-yl)methyl]-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
3-(2-ethyl-1H-imidazol-1-yl)-1-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]amine
1-methyl-5-(4-methyl-3-phenylpiperazine-1-carbonyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-(dimethyl-1H-1,2,4-triazol-3-yl)-1-(1,2,3,4-tetrahydronaphthalen-2-yl)urea
3-[ethyl({[2-(methylsulfanyl)phenyl]methyl})amino]-1λ6-thiolane-1,1-dione
2-(3,4-dichlorophenyl)-4-(3-fluoropyridin-4-yl)morpholine
3-(3-methoxyphenyl)-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]propanamide
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-(quinoxalin-5-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-methyl-1-[3-(2-methylpyrimidin-4-yl)phenyl]-3-[(trimethyl-1H-pyrazol-4-yl)methyl]urea
2-(pyridin-2-yl)-5-[4-(pyridin-4-yl)piperidine-1-carbonyl]pyrimidin-4-ol
ethyl 4-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)piperazine-1-carboxylate
1-[(2S)-2-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]pyrrolidin-1-yl]ethan-1-one
N-[(3S,4R)-1-[2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
6-(1-benzylpiperidin-4-yl)-N-(3,4-difluorophenyl)-6-azaspiro[2.5]octane-1-carboxamide
1-[1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)ethyl]-4-[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1H-1,2,3-triazole
1-methyl-3-[4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]-6-(propan-2-yl)-1,2-dihydropyridin-2-one