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2-(2-phenyl-1H-imidazol-1-yl)-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]acetamide
2-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-{[1-(propan-2-yl)piperidin-3-yl]methyl}acetamide
ethyl 4-[(4-chlorophenyl)methyl]-1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxylate
7-(cyclopropylmethyl)-2-(3-methoxybenzoyl)-2,7-diazaspiro[4.5]decan-6-one
9-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
7-(propan-2-yl)-2-[5-(trifluoromethyl)pyridin-2-yl]-2,7-diazaspiro[4.5]decan-6-one
3-cyclopropanecarbonyl-9-[(3-ethenylphenyl)methyl]-3,9-diazaspiro[5.5]undecane
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1,1-dioxo-1λ6-thiolane-3-carboxamide
2-{4-[3-oxo-3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]piperazin-1-yl}pyridine-3-carbonitrile
2-cyclohexyl-6-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]-1,3-benzoxazole
(2S)-1-[1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carbonyl]pyrrolidine-2-carboxamide
1-[2-(dimethylamino)-2-(3-fluorophenyl)acetamido]cycloheptane-1-carboxamide
2-{9-[(1R,3S)-3-aminocyclohexanecarbonyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
4-{[(2-amino-6-methoxypyrimidin-4-yl)amino]methyl}-1-cyclopropylpyrrolidin-2-one
3-(5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}-1,3,4-oxadiazol-2-yl)pyridine
N-benzyl-N-methyl-3-(1,2,3,6-tetrahydropyridin-1-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
(3S,4S)-1-[(cycloheptylcarbamoyl)methyl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
3-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}-2-methylpyridine
1-[(3-chloropyridin-4-yl)methyl]-4-(pyrrolidine-1-sulfonyl)-1,4-diazepane
[(3R,4R)-4-(piperidin-1-ylmethyl)-1-[4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazolin-2-yl]pyrrolidin-3-yl]methanol
[1-(2,1,3-benzoxadiazol-4-ylmethyl)-4-[(2-chlorophenyl)methyl]piperidin-4-yl]methanol
3-[3-({[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]amino}methyl)-1H-indol-1-yl]propanamide
N-(2-methoxyethyl)-1-(1-{2-[3-(trifluoromethyl)phenyl]acetyl}piperidin-3-yl)-1H-1,2,3-triazole-4-carboxamide
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-1,1-dioxo-1λ6-thiane-4-carboxamide
2-[4-methyl-2-(6-methyl-9H-purin-9-yl)phenoxy]acetamide
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N,6-dimethylpyrazolo[1,5-a]pyrimidine-3-carboxamide
3-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidine-1-carbonyl]-1H-pyrazol-5-amine
3-[(3S,4R)-4-(dimethylamino)-1-(naphthalen-2-ylmethyl)piperidin-3-yl]-N-(4-fluorophenyl)propanamide
2-[2-(4-tert-butylphenoxymethyl)pyrimidin-4-yl]pyridine-4-carboxylic acid
4-{3-[5-(1-ethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]propyl}piperazin-2-one
2-(cyclohex-1-en-1-yl)-1-[7-(1-hydroxy-3-phenylpropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
2-(1,1-dioxo-1λ6-thiomorpholin-4-yl)-2-(4-fluoro-3-methylphenyl)acetic acid
4-hydroxy-2-(3-methylphenyl)-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]pyrimidine-5-carboxamide
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-5-methoxy-4-oxo-1,4-dihydropyridine-2-carboxamide
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(morpholin-4-yl)ethan-1-one
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}[(1-phenyl-1H-pyrazol-4-yl)methyl](pyridin-4-ylmethyl)amine
3-[1-(2-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]-1,5,6-trimethyl-1,2-dihydropyridin-2-one
5-ethyl-2-methyl-4-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
methyl({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)(pyrazin-2-ylmethyl)amine
(2S,4S)-N-ethyl-4-[2-(pyridin-3-yl)acetamido]-1-(1,3-thiazol-2-ylmethyl)pyrrolidine-2-carboxamide
methyl 3-{[(5-propyl-1,2-oxazol-3-yl)formamido]methyl}-5-[3-(trifluoromethyl)benzamido]benzoate
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-methyl-1-[(2E)-3-phenylprop-2-en-1-yl]-3-[3-(piperidine-1-carbonyl)phenyl]urea
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetamide
(3aR,6aR)-2-benzyl-5-cyclopentanecarbonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[2-(3,4-dichlorophenyl)morpholin-4-yl]-2-(pyrrolidin-1-yl)ethan-1-one
2-propyl-N-{1-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1,3-thiazole-4-carboxamide
2,5-dimethyl-N-(1-methylpiperidin-4-yl)-N-(pyridin-3-ylmethyl)-1,3-thiazole-4-carboxamide
(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
2-{1-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]piperidin-2-yl}pyridine