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5-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-4-propylpyrimidine
3-(2-amino-1,3-thiazol-4-yl)-1-{2-[(4-methoxyphenyl)methyl]morpholin-4-yl}propan-1-one
(4aS,8aR)-6-benzyl-1-(piperidin-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
1-[(3,5-dimethylphenyl)methyl]-4-[2-(propan-2-yloxy)acetyl]piperazin-2-one
N,2-dimethyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]pyrido[2,3-d]pyrimidin-4-amine
3-[1-(furan-3-ylmethyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)propanamide
(2S)-2-hydroxy-N-[2-(2-methylphenyl)-1,3-benzoxazol-6-yl]-2-phenylacetamide
2-{4-[(3-fluorophenyl)methyl]-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-{[4-(4-chloro-2-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyridine
4-({3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}methyl)benzoic acid
N-{1-[1-(1-ethylpiperidin-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
8-(1H-indole-6-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[(3-methoxyphenyl)methyl]-4-(3-phenylbutanoyl)piperazin-2-one
2-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-ol
2-{2-[5-(1-ethyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]propyl}pyrazine
methyl (2S)-2-[1-(5-{[benzyl(methyl)amino]methyl}-1,2-oxazol-3-yl)-N-methylformamido]propanoate
2-[1-benzyl-4-(thiophen-2-ylmethyl)piperazin-2-yl]ethan-1-ol
5-phenyl-3-[4-(pyrazin-2-yl)piperazin-1-yl]-1,2,4-triazine
3-(2-hydroxyethyl)-N-[4-methyl-3-(propan-2-yl)phenyl]-4-(2-methylpropyl)piperazine-1-carboxamide
1-(4-fluorophenyl)-3-{[1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]methyl}urea
(2H-1,3-benzodioxol-4-ylmethyl)(methyl){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
(3S,4R)-1-(ethanesulfonyl)-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
1-[4-(2-phenoxyethyl)piperazin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
N-{3-[2-(2-aminoethyl)phenyl]phenyl}acetamide
(2H-1,3-benzodioxol-5-ylmethyl)[(5-tert-butyl-1H-pyrazol-3-yl)methyl](pyridin-3-ylmethyl)amine
3-cyclopropyl-5-[2-(3-methyl-1,2,4-oxadiazol-5-yl)phenoxymethyl]-1,2,4-oxadiazole
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-(dimethylamino)pyridine-3-carboxamide
(2S)-4-methanesulfonyl-2-[(1-methyl-3-propyl-1H-pyrazol-5-yl)formamido]butanoic acid
3-[(3R,4S)-3-amino-4-cyclopropylpyrrolidine-1-carbonyl]-6-methoxy-1,4-dihydroquinolin-4-one
[(1S,3S,3aS,6aR)-5-ethyl-3-(2-methoxypyridin-3-yl)-1-phenyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
2-chloro-4-[2-(morpholin-4-ylmethyl)phenyl]benzoic acid
3-[3-(5-methylfuran-2-yl)-5-[(propylsulfanyl)methyl]-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
N-methyl-4-(piperazine-1-sulfonyl)-N-(1H-pyrazol-3-ylmethyl)benzamide
(2R)-2-{[5-(2-methoxyphenoxymethyl)-1H-pyrazol-3-yl]formamido}propanamide
[(5-chlorofuran-2-yl)methyl](1,4-dioxan-2-ylmethyl)methylamine
N-(2-hydroxyethyl)-N-methyl-1-[1-(6-methylhept-5-en-2-yl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
6-(cyclopropylmethoxy)-1-[3-(2-oxopyrrolidin-1-yl)propyl]-4-(1H-pyrazol-4-ylmethyl)-1,4-diazepan-2-one
N-(1,1-dioxo-1λ6-thian-4-yl)-6-methoxy-N,3-dimethyl-1-benzofuran-2-carboxamide
2-[5-(1H-imidazole-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-1-methyl-1H-1,3-benzodiazole
(3S)-1-[5-(3-hydroxyazetidine-1-carbonyl)-1-methyl-1H-1,3-benzodiazol-2-yl]pyrrolidin-3-ol
N-[(2S)-1-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-4-methyl-1-oxopentan-2-yl]acetamide
{[2-(butan-2-ylsulfanyl)pyrimidin-5-yl]methyl}(methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
3-[(3S,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(5-chloro-2-methylphenyl)urea
1-methyl-N-[3-(4H-1,2,4-triazol-4-yl)propyl]azepane-2-carboxamide
5-(3-methyl-3-phenylpiperidine-1-carbonyl)pyrazin-2-ol
(furan-2-ylmethyl)[(2E)-2-methylbut-2-en-1-yl][2-(morpholin-4-yl)ethyl]amine
4-(4-methylphenoxy)-1-(1,3-thiazol-2-yl)piperidine-4-carboxylic acid
1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-yl]-4-(4-methoxyphenyl)butane-1,4-dione
3-{3-amino-4,6-dimethyl-1H-pyrazolo[3,4-b]pyridin-5-yl}-N,N-diethylbenzamide
5-[1-(2,1,3-benzothiadiazol-5-ylmethyl)pyrrolidin-2-yl]-N-(2-hydroxyethyl)thiophene-2-carboxamide