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2-(1,4-dioxan-2-ylmethyl)-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
N-[(5-methylpyrazin-2-yl)methyl]-2,3-dihydro-1-benzothiophene-2-carboxamide
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-2,6-dihydroxybenzamide
9-[2-(dimethylamino)acetyl]-2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
(2S,3R)-2-amino-3-hydroxy-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)butanamide
2-[methyl(pyridin-3-ylmethyl)amino]-N-(2-methylpropyl)-N-(thiophen-3-ylmethyl)acetamide
2-ethoxy-5-(4-methyl-1H-pyrazol-1-yl)benzamide
3-(3-hydroxy-1,2-oxazol-5-yl)-N-[1-methyl-4-(propan-2-yloxy)-1H-indazol-3-yl]propanamide
9-[2-(3-oxopiperazin-1-yl)acetyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(2-hydroxyethyl)-2-methyl-N-{[4-(methylsulfanyl)phenyl]methyl}-1-benzofuran-5-carboxamide
5-oxo-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
4-[3-(4-methanesulfonylphenyl)phenyl]-4H-1,2,4-triazole
7-hydroxy-4-(3-hydroxy-6-methylpyridin-2-yl)-6-methoxy-1,2,3,4-tetrahydroquinolin-2-one
5-(naphthalen-1-yl)-3-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}-1,2,4-triazine
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-[(3-methylpyridin-4-yl)methyl]benzamide
3-(2-fluorophenyl)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1H-pyrazole-5-carboxamide
3-(dimethyl-1,2-oxazol-4-yl)-N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]propanamide
N'-(2-methylphenyl)-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)propanediamide
1-(1-methyl-3-phenyl-1H-pyrazol-5-yl)-3-[3-(propan-2-yloxy)propyl]urea
N-(3-methoxyphenyl)-3-[1-(1H-pyrrole-3-carbonyl)piperidin-4-yl]propanamide
dimethyl[1-(3-{1-propyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenyl)ethyl]amine
2-(5-chloro-6-methyl-1-benzofuran-3-yl)-N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]acetamide
N-[2-(dimethylamino)ethyl]-N,2,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
1-[4-(furan-2-ylmethoxy)phenyl]-3-[(1-hydroxycyclohexyl)methyl]urea
1-(furan-2-carbonyl)-4-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,4-diazepane
1-(adamantan-1-yl)-4-(dimethyl-1,3-oxazole-4-carbonyl)piperazine
2-[(4-chlorophenyl)methyl]-8-[(2S)-3-hydroxy-2-methylpropyl]-2,8-diazaspiro[4.5]decan-3-one
(1S,5R)-3-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
14-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[5,8-dimethoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
4-{3-[1-(cyclopropylmethyl)-1H-pyrazol-3-yl]phenyl}-2-methylpyridine
(1R,9aR)-1-{[(2-methylpyridin-3-yl)oxy]methyl}-octahydro-1H-quinolizine
(1R,2S,6R,7S)-4-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-azatricyclo[5.2.2.02,6]undecane
1-{3,9-diazaspiro[5.6]dodecan-9-yl}-5-phenylpentane-1,5-dione
methyl 3-(3-methoxybenzoyl)-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-1-(furan-2-ylmethyl)piperidine-3-carboxamide
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(1H-pyrazol-1-yl)butanamide
3-(hydroxymethyl)-N-{2-[(2-methylprop-2-en-1-yl)oxy]phenyl}morpholine-4-carboxamide
({4-[1-(5-cyclopropyl-3-methyl-1H-pyrazole-4-carbonyl)piperidin-2-yl]phenyl}methyl)dimethylamine
8-fluoro-2-[4-(4-methoxybutyl)piperazine-1-carbonyl]quinoline
3-{2-[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-indole
N'-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)butanediamide
2-({2-[1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
3-{[cyclohexyl(methyl)amino]methyl}-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-2-one
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(3-propyl-1H-pyrazole-4-carbonyl)piperidine
3-({[1-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-4-yl]oxy}methyl)pyridine
1-(1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}azetidin-3-yl)-3,5-dimethyl-1H-pyrazole
1-[4-(3-acetylphenyl)phenyl]-3-[3-(morpholin-4-yl)propyl]urea