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4-methyl-3-(2-oxoimidazolidin-1-yl)-N-{1-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}benzamide
N-[4-(1,3-thiazol-4-yl)phenyl]-4-(2,2,2-trifluoroethyl)piperazine-1-carboxamide
N,N,1-trimethyl-2-oxo-3-phenyl-1,8-diazaspiro[4.5]decane-8-sulfonamide
1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]ethan-1-one
2-{2-oxo-1'-[(1-propyl-1H-imidazol-2-yl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1-yl}acetamide
3-(4-methylphenyl)-1-{2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}propan-1-one
(1R,3S)-3-(2-aminoethoxy)-7-[1-(2-chlorophenyl)piperidin-4-yl]-7-azaspiro[3.5]nonan-1-ol
4-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-6-(morpholin-4-yl)pyrimidin-2-amine
4,6-dimethyl-2-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidine
2-(5-acetylthiophen-3-yl)-N-[(3-fluoro-4-methylphenyl)methyl]acetamide
1-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}-4-(6-methylpyridin-2-yl)piperazine
N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-5-(1H-indol-1-ylmethyl)-1H-pyrazole-3-carboxamide
5-(2,3-dihydro-1-benzofuran-5-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2-methyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]benzamide
N,N-dimethyl-2-[(1S,5R)-6-[(2-phenyl-1,3-thiazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
N,N-diethyl-1-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
N-{1-[(4-chlorophenyl)methyl]cyclopropyl}-2,6-dimethylpyridine-4-carboxamide
2-[3-(5-chlorothiophen-2-yl)-1H-pyrazol-1-yl]-N-[2-(propan-2-yl)-2H-1,2,3-triazol-4-yl]acetamide
1-[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
N-(2-hydroxyethyl)-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
2-(4-hydroxyphenyl)-4,6-dimethylpyridine-3-carbonitrile
6-[(4aS,8aR)-2-oxo-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-6-yl]pyridine-3-carbonitrile
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-[(1-propyl-1H-imidazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-phenylpiperidine
(2S,4S)-4-amino-N-benzyl-1-methyl-N-(1,3-thiazol-2-ylmethyl)pyrrolidine-2-carboxamide
4'-ethyl-1-(pentan-2-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-(3-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)benzonitrile
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(3-fluoropyridin-2-yl)pyrrolidin-3-yl]methanol
N-[1-(cyclohex-1-en-1-yl)ethyl]-2-(methylamino)pyridine-4-carboxamide
4-{[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1-methyl-1H-pyrazole
3-{[6-hydroxy-4-(1-methyl-1H-pyrazole-5-carbonyl)-1,4-diazepan-1-yl]methyl}benzonitrile
3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)-N-[(4-phenyloxan-4-yl)methyl]propanamide
3-methyl-7-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
3-{[4-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}benzonitrile
methyl[1-(4-methylpyridin-2-yl)propan-2-yl]{[5-(1H-pyrazol-5-yl)thiophen-2-yl]methyl}amine
8-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)-2-(pyrimidin-5-yl)quinoline-4-carboxamide
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine
1-{4-[2-(oxolan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidin-1-yl}-3-phenylpropan-1-one
8-methoxy-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-[2-(5-{6-methylimidazo[2,1-b][1,3]thiazol-5-yl}-4-phenyl-1H-imidazol-1-yl)ethyl]pyridine
4-({3-[1-(oxolan-3-ylmethyl)-1H-imidazol-2-yl]phenyl}methyl)morpholine
1-[3-(1H-imidazol-2-yl)-8-methylimidazo[1,2-a]pyridine-2-carbonyl]piperidine
3-(quinolin-5-yl)-5-(thiomorpholine-4-sulfonyl)benzoic acid
9-(1-benzylpiperidin-4-yl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-cyclopentyl-N3-{imidazo[1,2-a]pyridin-2-ylmethyl}-N5-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
4-{[1-(1,2,4-oxadiazol-3-ylmethyl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
1-{2-amino-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-5-yl}-2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)ethan-1-one
2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-1-[4-(pyridin-3-yloxy)piperidin-1-yl]ethan-1-one
ethyl 1-[3-(1,2-oxazolidin-2-yl)propanoyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
[(1-cyclopentylpiperidin-4-yl)methyl][(6-methylpyridin-2-yl)methyl](oxolan-2-ylmethyl)amine