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(3R,4S)-4-cyclopropyl-1-[4-(4-methylphenoxymethyl)benzoyl]pyrrolidin-3-amine
3-{[4-(3-hydroxypropyl)piperazin-1-yl]methyl}-7-methoxy-1,2-dihydroquinolin-2-one
N-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-methyloxan-4-amine
2-{[(3aS,6aR)-3-[3-(morpholin-4-yl)propyl]-2-oxo-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-5-yl]methyl}benzonitrile
4-(4-methyl-1H-pyrazol-1-yl)-1-[2-(pyridin-3-yloxy)acetyl]piperidine-4-carboxylic acid
1-methyl-N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
2-({[(3R,4R)-1-(4-aminopyrimidin-2-yl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(ethyl)amino)ethan-1-ol
1-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]ethan-1-one
7-methyl-3-[4-(trifluoromethyl)benzoyl]-3,7,11-triazaspiro[5.6]dodecan-12-one
4-methoxy-3,5-dimethyl-2-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}pyridine
3-(1H-indol-6-yl)-5-(thiomorpholine-4-sulfonyl)benzoic acid
7-(7-chloroquinolin-4-yl)-2,7-diazaspiro[4.5]decane
N-ethyl-2-(4-ethylpiperazin-1-yl)-N-(2-methylprop-2-en-1-yl)-2,3-dihydro-1H-indene-2-carboxamide
N-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-propyl-1,3-thiazole-4-carboxamide
1-benzyl-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
2-{[4-(2-phenylpropyl)-1H-1,2,3-triazol-1-yl]methyl}-3,4-dihydroquinazolin-4-one
(2R)-N-[(1-benzylpiperidin-4-yl)methyl]-2-cyclohexyl-2-hydroxy-N-methylacetamide
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}propanamide
1-[3-(hydroxymethyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one
(1R,7S)-3-(2-methoxyethyl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
5-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-4-propylpyrimidine
5-chloro-3-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]pyridin-2-ol
N-cyclopentyl-N'-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]butanediamide
(4-{pyrazolo[1,5-a]pyridine-3-carbonyl}-1,4-oxazepan-6-yl)methanol
1-(2-methoxyphenyl)-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-1H-pyrazole-4-carboxamide
N-methyl-N-[2-(morpholin-4-yl)propyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
4-[7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]oxane-4-carbonitrile
4-hydroxy-1-[(4-methoxy-3-methylphenyl)methyl]piperidine-4-carboxylic acid
N-methyl-N-{[5-oxo-4-(thiophen-2-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-3-yl]methyl}methanesulfonamide
(4aS,7aR)-1-[1-(methoxymethyl)cyclobutanecarbonyl]-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-({2-[1-(3-ethyl-1,2-oxazole-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
4-(cyclopropylmethyl)-1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-3-(propan-2-yl)-1,4-diazepan-5-one
N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-2-(1H-pyrazol-1-yl)acetamide
N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
3-{[(3,4-dichlorophenyl)methyl]amino}-N-(pyridin-3-yl)propanamide
2-(4-chloro-3-methyl-1H-pyrazol-1-yl)-N-{[1-(furan-2-ylmethyl)pyrrolidin-3-yl]methyl}acetamide
N-[(4-acetamidophenyl)methyl]-2-[(2-phenylethyl)amino]acetamide
3-[(dimethylamino)methyl]-1-(1H-indol-5-ylmethyl)piperidin-3-ol
4-[2-(2-chlorophenyl)-2-hydroxyacetyl]-1-(2-methoxyphenyl)piperazin-2-one
2-amino-4-(2-methyl-1H-imidazol-4-yl)-6-(thiophen-3-yl)pyridine-3-carbonitrile
[(1-ethyl-1H-imidazol-2-yl)methyl]({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})amine
N-cyclopentyl-2-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)furan-3-carboxamide
4,6-dimethyl-1-(2-{[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}ethyl)-1,2-dihydropyrimidin-2-one
5-ethyl-5-{1-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperidin-4-yl}imidazolidine-2,4-dione
(2R)-N1-(1-tert-butyl-4-phenyl-1H-pyrazol-5-yl)pyrrolidine-1,2-dicarboxamide
N-[2-methoxy-2-(thiophen-2-yl)ethyl]-6-(morpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
N-[2-(3,4-dimethylphenoxy)ethyl]-3-[4-(3-methylphenyl)piperazin-1-yl]propanamide
4-methyl-2-phenyl-5-(3-phenylpiperazine-1-carbonyl)pyrimidine
5-[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1,2-dihydropyridin-2-one
N-[(3S)-1-[5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]pyrrolidin-3-yl]acetamide