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8-methyl-N-[1-(6-methylpyridin-3-yl)ethyl]-2-(pyrimidin-5-yl)quinoline-4-carboxamide
2-[1-methyl-4-({4-[methyl(phenyl)amino]phenyl}methyl)piperazin-2-yl]ethan-1-ol
(1R,2S,9R)-11-{pyrazolo[1,5-a]pyridine-3-carbonyl}-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
5-[({1-[2-(dimethylamino)-6-methylpyrimidin-4-yl]piperidin-4-yl}amino)methyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
7-(propan-2-yl)-2-(1,3,4-thiadiazol-2-yl)-2,7-diazaspiro[4.5]decan-6-one
1-(4-hydroxy-1,2-oxazolidin-2-yl)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one
{[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}[1-(1H-pyrazol-1-yl)propan-2-yl]amine
1-(2-methyl-7-{4H-thieno[3,2-b]pyrrole-5-carbonyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl)pyrrolidine
4-[(4S)-4-hydroxy-3,3,4-trimethylpiperidine-1-carbonyl]-1,2-dihydroquinazolin-2-one
2-[(5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-yl)amino]acetamide
3-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methoxy}pyridine-2-carbonitrile
1-[(2,6-difluorophenyl)methyl]-N-[3-(methylsulfanyl)propyl]-1H-1,2,3-triazole-4-carboxamide
(3S,4R)-1-(3-methoxybenzoyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
1-ethyl-4,6-dimethyl-N-[2-(2-methylpropanesulfonyl)ethyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
1-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
N-[(3S,7S,8aS)-1,4-dioxo-3-propyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-methoxybenzamide
3-cyclopropaneamido-N-[(6-hydroxypyrimidin-4-yl)methyl]-4-methylbenzamide
N-(1-carbamoylcyclopentyl)-4-(pyrrolidin-1-ylmethyl)benzamide
2-{4-[(3-ethoxyphenyl)methyl]-1-[(4-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
8-[2-(4-chloro-3-methyl-1H-pyrazol-1-yl)acetyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
3-{2-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]-2-oxoethyl}-1,3-diazinane-2,4-dione
N-(2-methylpropyl)-3-oxo-N-(3-phenylprop-2-yn-1-yl)-3,4-dihydro-2H-1,4-benzoxazine-7-carboxamide
N-methyl-5-(morpholin-4-ylmethyl)-N-[2-(piperidin-1-yl)ethyl]-1,2-oxazole-3-carboxamide
N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-methylfuran-3-carboxamide
2-[2-(1-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethyl]pyridine
N-(3-{[(2H-1,3-benzodioxol-5-ylmethyl)(cyclopropyl)carbamoyl]methoxy}phenyl)propanamide
N-methyl-3-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}propanamide
5-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-3,4-dihydropyrimidin-4-one
3-({[(3-methoxyphenyl)methyl](prop-2-en-1-yl)amino}methyl)benzonitrile
1-[benzyl(methyl)amino]-3-{4-[(benzylamino)methyl]phenoxy}propan-2-ol
(2S)-N-(6-cyanopyridin-3-yl)-2-(methoxymethyl)pyrrolidine-1-carboxamide
4-({2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)benzonitrile
2-cyclopentyl-9-[(4-methyl-1H-imidazol-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(4-butylpiperazin-1-yl)-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
9-(cyclopropylmethyl)-4-(3,6-dimethylpyrazin-2-yl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-[4-(5-fluoropyridin-2-yl)-1H-pyrazol-1-yl]-N-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[(5-methylpyrazin-2-yl)methyl]-1H-pyrazole-3-carboxamide
2-(dimethylamino)-2-(3-methylphenyl)-1-{4-[2-(pyrrolidin-1-yl)ethyl]piperazin-1-yl}ethan-1-one
1-[(2-chlorophenyl)methyl]-N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-1H-1,2,3-triazole-4-carboxamide
4-({methyl[1-(pyridin-2-yl)ethyl]amino}methyl)-1H-pyrazole-3-carboxylic acid
(3aS,6aS)-2-cyclobutanecarbonyl-5-{[3-(methylsulfanyl)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(4-chloro-3-methyl-1H-pyrazol-1-yl)-1-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]ethan-1-one
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-1H-pyrrole-3-carboxamide
(1S,6R)-3-[(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)sulfonyl]-3,9-diazabicyclo[4.2.1]nonane
3-(2H-1,3-benzodioxol-5-ylmethyl)-N-[(5-phenyl-1H-pyrazol-3-yl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
[(3R,4R)-4-[(dimethylamino)methyl]-1-({2-[(2-methylphenyl)methoxy]phenyl}methyl)pyrrolidin-3-yl]methanol
(3S,7S,8aS)-3-[(benzyloxy)methyl]-7-[({3-[(diethylamino)methyl]-4-methoxyphenyl}methyl)amino]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
1-[1-(2,5-difluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-methoxypropan-1-one
4-(4-ethyl-6-{4-[1-(morpholin-4-yl)ethyl]phenyl}pyrimidin-2-yl)morpholine