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1-(4-fluorophenyl)-4-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}butane-1,4-dione
3-ethyl-2-[2-(propan-2-yl)-2,5-dihydro-1H-pyrrole-1-carbonyl]-1H-indole
2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-5-methoxy-3-methyl-1H-indole
3-(4-methylphenyl)-3-({5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)propan-1-ol
2-methoxy-1-{1'-[(2S)-1-(propan-2-yl)pyrrolidine-2-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
5-[(4-hydroxypiperidin-1-yl)methyl]-N-[(3-methylpyridin-4-yl)methyl]-1,2-oxazole-3-carboxamide
N-(cyclobutylmethyl)-4-(2,4-dioxoimidazolidin-1-yl)-N-(oxolan-2-ylmethyl)benzamide
N-[2-(1-methylpyrrolidin-2-yl)ethyl]-2-(trimethyl-1H-pyrazol-1-yl)acetamide
1-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-3-(2-methyl-1H-imidazol-1-yl)butan-1-one
N-methyl-N-propyl-2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
4-(2,3-dihydro-1H-inden-5-yloxy)-1-(pyridin-4-ylmethyl)piperidine-4-carboxylic acid
N-{2-[1-(furan-2-ylmethyl)piperidin-3-yl]ethyl}cyclopropanesulfonamide
N-(1-benzylpyrrolidin-3-yl)-3-[1-(cyclohex-1-ene-1-carbonyl)piperidin-4-yl]propanamide
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-N-{2-[(1,3-thiazol-2-yl)carbamoyl]ethyl}propanamide
N-[1-(4-methoxyphenyl)-5-oxopyrrolidin-3-yl]-1H-1,3-benzodiazole-2-carboxamide
3-(azepan-1-ylmethyl)-3-hydroxy-1-(2-methoxyethyl)piperidin-2-one
2-(methylamino)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}pyridine-4-carboxamide
2-(dimethylamino)-2-(4-methylphenyl)-N-[(1r,4r)-4-hydroxycyclohexyl]acetamide
N-[(3S,4R)-4-(4-methylphenyl)-1-[2-(1H-1,2,4-triazol-1-yl)acetyl]pyrrolidin-3-yl]cyclopropanecarboxamide
N-ethyl-1-[2-(3-fluorophenyl)ethyl]-6-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]piperidine-3-carboxamide
(1R,2R,6S,7S)-N-[6-(3-methoxyphenoxy)pyridin-3-yl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane-4-carboxamide
5-(7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decane-2-carbonyl)-2,1,3-benzoxadiazol-1-ium-1-olate
1-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}-2-(methylsulfanyl)ethan-1-one
N-ethyl-N-{1-[2-(methylamino)pyridine-4-carbonyl]pyrrolidin-3-yl}acetamide
ethyl 2-[1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)piperidin-2-yl]acetate
[(2Z)-2-chloro-3-phenylprop-2-en-1-yl](methyl)({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine
1-(2-fluorophenyl)-4-[1-(2-methylfuran-3-carbonyl)piperidin-3-yl]piperazine
4-(1H-imidazol-2-yl)-3-(3-methoxyphenyl)-1-phenyl-1H-pyrazole
2-methyl-3-[3-(pyridin-2-yl)azetidine-1-carbonyl]-4,5,6,7-tetrahydro-1H-indol-4-one
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-(furan-2-ylmethyl)piperidine-4-carboxamide
1-methyl-2-oxo-8-(quinolin-2-yl)-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-[(1-butyl-3-ethyl-1H-1,2,4-triazol-5-yl)methyl]-1,2-dihydropyrimidin-2-one
5-[5-(1H-imidazol-1-ylmethyl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
4-[2,2-bis(prop-2-en-1-yl)pyrrolidine-1-carbonyl]-2,6-dimethylpyrimidine
6-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
7-methyl-2-(2-phenoxybenzoyl)-2,7-diazaspiro[4.5]decan-6-one
9-(cyclopropylmethyl)-1-methyl-4-{[3-(methylsulfanyl)phenyl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)-1-(thiophene-2-sulfonyl)piperidine
5-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-N-methyl-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-(4-methyl-1H-pyrazol-1-yl)-1-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
1-{2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}azepan-4-ol
N-[4-(4-cyclopentyl-1,4-diazepane-1-carbonyl)phenyl]ethane-1-sulfonamide
1-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]-4-(1H-imidazol-1-yl)butan-1-one
9-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-1,3-benzodiazole
4-[(2-fluoro-4-methoxyphenyl)methyl]-1-methyl-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
5-methyl-1'-(3-phenyl-1H-pyrazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
[(2S)-1-{5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}pyrrolidin-2-yl]methanol
(3S,5R)-1-benzyl-5-[(4-fluorophenyl)carbamoyl]piperidine-3-carboxylic acid
2-{[2-(1-methylpyrrolidin-2-yl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid