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N-(adamantan-2-ylmethyl)-2-oxo-6-({1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl}methyl)-1,2-dihydropyridine-3-carboxamide
9-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-(2-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-2-fluoro-5-sulfamoylbenzamide
2-{1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]pyrrolidin-2-yl}pyridine
1-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-2-methyl-1,4-diazepan-5-one
8-[(5-ethylfuran-2-yl)methyl]-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S,4R)-3-(dimethylamino)-N-[(3-fluorophenyl)methyl]-4-(propan-2-yl)pyrrolidine-1-carboxamide
2-amino-4-[4-(3-hydroxyprop-1-yn-1-yl)phenyl]-6-(propan-2-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-[(2S)-oxolan-2-ylmethyl]pyrimidine-5-carboxamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-5-[3-(trifluoromethyl)phenyl]-1,2,4-triazin-3-amine
9-(5-ethyl-2-methylpyrimidin-4-yl)-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
5-{2-[(cyclopropylmethyl)amino]pyrimidin-4-yl}-2-ethoxybenzoic acid
4-{[1-(3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1,5-dimethyl-1H-pyrazole
methyl 2-[3-(2-methoxybenzoyl)piperidin-1-yl]pyridine-4-carboxylate
8-[5-(2-chlorophenyl)furan-2-carbonyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3S,4R)-1-(1-acetylpiperidin-4-yl)-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
N-cyclohexyl-N-[2-(ethylsulfanyl)ethyl]-2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
N-[(5-methylpyrazin-2-yl)methyl]-1-[2-(methylsulfanyl)pyrimidin-4-yl]piperidin-4-amine
(1R,5R)-6-benzyl-N-methyl-N-phenyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-1-ethyl-3-methyl-1H-pyrazole-5-carboxamide
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-[2-(3-methoxyphenyl)phenyl]-1-(3-methylbut-2-en-1-yl)piperidine-4-carboxamide
3-{4-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}phenol
[1-(5-{[(2-propylpyrimidin-5-yl)methyl]amino}-5,6,7,8-tetrahydroquinazolin-2-yl)piperidin-4-yl]methanol
(butan-2-yl)({[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl})(thiophen-3-ylmethyl)amine
N-[2-(4-fluorophenyl)ethyl]-1-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(2R,6R)-4-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-triene-6-carboxylic acid
1-{1-[(2,3-dichloro-4-methylphenyl)methyl]piperidin-3-yl}pyrrolidin-2-one
2-{2-[2-(1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-4,5,6,7-tetrahydro-1,3-benzothiazole
2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-(1H-indol-6-ylmethyl)acetamide
2-[4-(2-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]-1,4-dihydroquinolin-4-one
3-phenyl-8-[(2E)-3-phenylprop-2-en-1-yl]-1,8-diazaspiro[4.5]decan-2-one
N-(1,3-dimethyl-1H-pyrazol-4-yl)-2-[4-(1-methyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]acetamide
4-[2-(aminomethyl)-5-fluoro-2,3-dihydro-1-benzofuran-7-yl]-6-methoxypyrimidin-2-amine
4-(2-methoxy-5-methylbenzoyl)-1-(4-methylphenyl)piperazin-2-one
1-[(4-ethylphenyl)methyl]-3-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
N-{2-[(4-chlorophenyl)methoxy]ethyl}-3-ethyl-4-methyl-1H-pyrazole-5-carboxamide
N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-1,9-dioxaspiro[5.5]undecan-4-amine
2-(1H-1,3-benzodiazol-1-yl)-N-(1-ethyl-1H-indazol-3-yl)acetamide
4-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-fluoropyridine
N-[2-(dimethylamino)ethyl]-3-{1-[(2-hydroxynaphthalen-1-yl)methyl]piperidin-4-yl}propanamide
2-[(4aR,7aS)-6,6-dioxo-4-(quinolin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
4-chloro-2-methoxy-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]benzamide
3-[1-(3-chloropyridin-2-yl)piperidin-3-yl]-N-(4-methoxy-2-methylphenyl)propanamide
2-methyl-9-(5-methyl-2-phenylfuran-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
3-{[2-(furan-2-yl)ethyl]sulfamoyl}-N-(pyridin-3-ylmethyl)benzamide
2-[4-(1-tert-butyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]-1-[(2R,6S)-2,6-dimethylmorpholin-4-yl]ethan-1-one
2-methoxy-5-{[4-(propan-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}phenol
2-[3-(3-methoxyphenoxymethyl)piperidine-1-carbonyl]-N,N-dimethylaniline
1-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one