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(4aS,8aR)-6-(5,6-dimethylpyrimidin-4-yl)-1-[3-(methylsulfanyl)propyl]-decahydro-1,6-naphthyridin-2-one
2-(3-methoxypropyl)-9-[2-(2-methyl-1H-imidazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
3-methoxy-1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
5-methyl-1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-5-phenylpiperidin-2-one
1-{2-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-2-yl]ethyl}pyrrolidin-2-one
1-(cyclopropylmethyl)-2-(propan-2-yl)-4-[3-(pyridin-4-yl)-1H-pyrazole-5-carbonyl]-1,4-diazepane
(1R,3S)-3-(2-aminoethoxy)-7-(5-chlorofuran-2-carbonyl)-7-azaspiro[3.5]nonan-1-ol
methyl 3-(2-chlorobenzenesulfonamido)-5-{[(2-methylphenyl)formamido]methyl}benzoate
N-methyl-N-{2-[2-(prop-2-en-1-yl)phenoxy]ethyl}-1H-1,2,3-benzotriazole-5-carboxamide
{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)[(5-methyl-1H-pyrazol-3-yl)methyl]amine
N-[4-(azepan-1-yl)butyl]-1-cyclopentyl-6-oxopiperidine-3-carboxamide
3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}-3-({[2-(1,3-thiazol-2-yl)ethyl]amino}methyl)piperidin-2-one
4-[(1R,5S)-3,8-diazabicyclo[3.2.1]octane-8-carbonyl]-7-fluoro-2-methylquinoline
3-{1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}-4-methyl-1,2,5-oxadiazole
2-{4-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}-1,3-thiazole-4-carboxamide
4-(2-{[(6-hydroxy-1,4-oxazepan-6-yl)methyl]amino}ethyl)benzene-1-sulfonamide
2-[3-(furan-2-yl)-1-(2-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-methylacetamide
5-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-{[3-(cycloheptyloxy)-4-methoxyphenyl]methyl}-N-cyclopropyl-4-(1H-pyrazol-1-yl)benzamide
ethyl 2-[4-(4-methoxyphenyl)-2-methyl-3-oxopiperazin-1-yl]acetate
4-{5-[3-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyrimidin-2-yl}morpholine
1-{2-[2-(9H-fluoren-2-yl)-1H-imidazol-1-yl]ethyl}imidazolidin-2-one
(2R,3R,6R)-3-(4-fluorophenyl)-5-(quinoxaline-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzoyl)pyrrolidin-3-amine
4-(2-acetyl-3-methoxyphenoxy)thiane-4-carboxylic acid
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1-[3-(2-methylpyrimidin-4-yl)phenyl]piperidin-4-amine
8-(2-chloro-6-fluorobenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-(3-chloro-4-methoxyphenyl)-3-{1-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]piperidin-3-yl}propanamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-4-(4-methylpiperazin-1-yl)benzamide
4-[5-(oxolan-2-yl)thiophene-2-carbonyl]morpholine
(2S,4R)-N-ethyl-4-[2-(3-methyl-1,2-oxazol-5-yl)acetamido]-1-(thiophen-3-ylmethyl)pyrrolidine-2-carboxamide
N-(2,3-dihydro-1H-inden-1-yl)-3-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propanamide
(2S)-2-amino-N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)propanamide
1-({2-[(benzenesulfonyl)methyl]phenyl}methyl)imidazolidin-2-one
6-chloro-N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
ethyl 3-[(3-chlorophenyl)methyl]-1-[2-(2,4-dioxo-1,3-thiazolidin-3-yl)acetyl]piperidine-3-carboxylate
3-[3-({[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl](methyl)carbamoyl}amino)phenyl]-N,N-dimethylpropanamide
methyl 4-[4-(1H-imidazol-2-ylmethyl)piperazin-1-yl]benzoate
N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-5-[3-(trifluoromethyl)phenoxymethyl]-1H-pyrazole-3-carboxamide
4-[(2,4-dimethoxyphenyl)methyl]-3-[2-(1,2-oxazinan-2-yl)-2-oxoethyl]piperazin-2-one
1-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)-3-(hydroxymethyl)piperidin-3-ol
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-6-(piperidine-1-carbonyl)pyrazin-2-amine
(1R,3S)-3-(2-hydroxyethoxy)-7-(1-phenylcyclopentanecarbonyl)-7-azaspiro[3.5]nonan-1-ol
N-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-1-methyl-1H-imidazole-2-carboxamide
1-ethyl-3-{2-oxo-2-[4-(pyridin-3-yloxy)piperidin-1-yl]ethyl}-3-[3-(trifluoromethyl)phenyl]pyrrolidine-2,5-dione
2-ethyl-9-[6-methyl-2-(propan-2-yl)pyrimidin-4-yl]-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(5-methoxy-1H-indol-3-yl)ethyl]-3-(1H-pyrazol-4-yl)benzamide
1-[1-(1,3-thiazole-4-carbonyl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine
1-[(2-fluorophenyl)methoxy]-8-[4-(2-oxopropyl)phenoxy]-1,8-diazaspiro[4.5]decan-2-one
1-{4-[4-(2-hydroxypropan-2-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-2-(2,2,6,6-tetramethylpiperidin-4-yl)ethan-1-one