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1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-(4-fluorophenoxy)ethan-1-one
N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
2-(4-{[2-methanesulfonyl-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}piperazin-1-yl)pyrazine
5-fluoro-2-{1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
4-[5-(pyridin-3-ylmethyl)-1,2,4-oxadiazol-3-yl]-1H-indole
5-fluoro-4-(3-phenylpiperazin-1-yl)quinazoline
5-methyl-1'-(5-phenyl-1,3,4-thiadiazol-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-{1-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-6-azaspiro[2.5]octane-6-carbonyl}-5-fluoro-1H-indole
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}acetamide
2-{4-[3-(1H-pyrazol-5-yl)phenyl]-1H-pyrazol-1-yl}acetamide
2-(methoxymethyl)-5-{[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}pyrimidine
8-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
2-cyclopropyl-N-[1-(3-methylphenyl)-5-oxopyrrolidin-3-yl]-6-oxo-1,6-dihydropyrimidine-5-carboxamide
3-[1-(2,3-dihydro-1-benzofuran-7-carbonyl)piperidin-4-yl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N3-cyclohexyl-1-cyclopropyl-N5-[(3,4-dimethoxyphenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
5-cyclohexaneamido-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1-(2-methoxyethyl)-1H-1,3-benzodiazole-7-carboxamide
3-butyl-1-methyl-4-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]piperazin-2-one
N-methyl-3-{N-methyl-1-[1-methyl-3-(2-methylpropyl)-1H-pyrazol-5-yl]formamido}butanamide
3-{2-[cyclohexyl(methyl)amino]ethyl}-8-(1H-imidazol-2-ylmethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
5-(1,2,3,4-tetrahydroisoquinolin-5-yl)thiophene-2-carboxamide
(2S)-4-methyl-1-[2-(phenoxymethyl)-1,3-oxazole-4-carbonyl]-2-phenylpiperazine
ethyl 3-benzyl-1-[(3,4-dimethoxyphenyl)carbamoyl]piperidine-3-carboxylate
N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
1-benzyl-5-[(1-benzylpiperidin-4-yl)amino]-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-2-(1-methyl-1H-pyrrol-3-yl)acetamide
2-{imidazo[1,2-a]pyridin-3-yl}-1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
4-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}-N,N-dimethyl-4-oxobutanamide
4-(4-chlorophenyl)-N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]butanamide
6,7-dimethoxy-3-[(3-methoxyphenyl)methyl]-3,4-dihydroquinazolin-4-one
N'-cyclooctyl-N-ethyl-N-(oxan-4-yl)butanediamide
N,1,3-trimethyl-2,6-dioxo-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,2,3,6-tetrahydropyrimidine-4-carboxamide
1-(furan-2-ylmethyl)-4-(oxolane-3-carbonyl)piperazine
7-methyl-12-oxo-N-propyl-3,7,11-triazaspiro[5.6]dodecane-3-carboxamide
N-[(3R,4S)-1-(2-methanesulfonylethyl)-4-(propan-2-yl)pyrrolidin-3-yl]-6-oxo-1,6-dihydropyridine-3-carboxamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]acetamide
(3aS,6aS)-2-[3-(2-methyl-1H-imidazol-1-yl)propyl]-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[4-(3-chlorophenyl)phenyl]-4-hydroxy-4-(hydroxymethyl)piperidine-1-carboxamide
N-(3-fluorophenyl)-4-[4-(1-hydroxypropyl)piperidin-1-yl]-4-oxobutanamide
2-(dimethylamino)-2-(2-fluorophenyl)-1-[3-(morpholin-4-yl)azetidin-1-yl]ethan-1-one
N-[(7-{2-methylthieno[2,3-d]pyrimidin-4-yl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]acetamide
4-methyl-7-({methyl[2-(morpholin-4-yl)propyl]amino}methyl)-2H-chromen-2-one
2-(ethylamino)-N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]pyrimidine-5-carboxamide
2,7,8-trimethyl-N-[2-(1H-pyrrol-1-yl)ethyl]quinoline-4-carboxamide
1-{1-methyl-2-oxo-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}propane-1,2-dione
2-{1'-[(2-methoxyphenyl)methyl]-2-oxo-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1-yl}acetamide
N-[2-(pyrrolidine-1-sulfonyl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
6-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
1-(furan-2-ylmethyl)-N-methyl-N-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)piperidine-3-carboxamide
5,5-dimethyl-1-(2-{7-methyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)imidazolidine-2,4-dione