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(2S,3S)-2-amino-1-{4-[(4-tert-butyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}-3-methylpentan-1-one
N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)-2-(1H-1,2,3,4-tetrazol-1-yl)pyridine-4-carboxamide
4-[2-(benzenesulfonyl)ethyl]-1-{[3-(2-methylphenyl)phenyl]methyl}-1,4-diazepan-5-one
5-(4-{[4-(morpholin-4-yl)piperidin-1-yl]methyl}phenoxy)-1-azabicyclo[3.2.1]octane
4-methoxy-N-({1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-3-yl}methyl)benzene-1-sulfonamide
6-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-methoxy-6-(propan-2-yl)-3-{[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
1-[3-(4-methylpiperazin-1-yl)propyl]-3-[1-phenyl-3-(propan-2-yl)-1H-pyrazol-5-yl]urea
2-(2-acetyl-4,5-dimethoxyphenyl)-1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]ethan-1-one
4-(4-methylphenyl)-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-5-(pyrimidin-5-yl)pyrimidin-2-amine
3-(2H-1,3-benzodioxol-5-yl)-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-3-phenylpropanamide
4-{1-butyl-5-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-3-yl}pyridine
1-(3-chlorophenyl)-4-[(3-{2-[1-(pyridine-4-carbonyl)piperidin-2-yl]ethoxy}phenyl)methyl]piperazine
3-{1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
(4aS,8aS)-2-{2-[(2-methoxyethyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-decahydroisoquinolin-4a-ol
2,3-dimethyl-6-(thiomorpholine-4-carbonyl)quinoxaline
1-(azepan-1-yl)-3-[3-({[(5-fluoro-1H-indol-2-yl)methyl](methyl)amino}methyl)phenoxy]propan-2-ol
2-(2-fluoro-5-methoxyphenyl)-1,3-thiazole
3-methyl-3-[(4-methyl-1,3-thiazol-2-yl)methyl]-1-[2-(piperidin-1-ylmethyl)phenyl]urea
4-[(E)-2-(4-hydroxy-3-methoxyphenyl)ethenyl]-3-(propan-2-yl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-methyl-6-[2-(morpholin-4-ylmethyl)phenyl]-2,3-dihydropyridazin-3-one
(4aR,7aS)-1-(2-methoxyacetyl)-4-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{[3-(2-hydroxyethyl)-4-(3-phenylpropyl)piperazin-1-yl]methyl}-4-methoxyphenol
1-(4-cyano-2-ethylphenyl)-3-[2-(ethylsulfanyl)ethyl]urea
6-[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
7-methyl-3-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}-3,7,11-triazaspiro[5.6]dodecan-12-one
(8aS)-2-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
1-ethyl-5-{[(4-fluorophenyl)methyl]amino}-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-[1-(3-methyl-1-benzothiophene-2-carbonyl)azetidin-3-yl]pyridine
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)propanamide
2-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-6-fluoro-4-methylquinoline
6-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
5-(cyclohex-3-en-1-yl)-1-methyl-3-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
5-methyl-1-[(5-methyl-1,2-oxazol-3-yl)methyl]-5-(4-methylpent-3-en-1-yl)piperidin-2-one
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-3,6-dimethyl-1-benzofuran-2-carboxamide
N-(2,5-difluorophenyl)-3-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carboxamide
3-{[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]methyl}benzonitrile
1-[3-(methylsulfanyl)butyl]-4-(pyridin-2-ylmethyl)-1,4-diazepane
2-(2-{[3-(2-fluorophenyl)pyrrolidin-1-yl]methyl}phenoxy)acetic acid
2-(3-fluorophenyl)-1-(5-phenyl-1,2-oxazole-3-carbonyl)azepane
(3aS,6aS)-2-cyclopentyl-5-{2-[4-(dimethylamino)phenyl]acetyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N3-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}-1-[(5-methylfuran-2-yl)methyl]-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
7-[1-ethyl-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-5-yl]-3-methyl-3,4-dihydroquinazolin-4-one
(4aR,7aS)-1-acetyl-4-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-cyclopentyl-N-[3-(4-{[(5-phenyl-1,2-oxazol-3-yl)methyl]amino}piperidin-1-yl)phenyl]acetamide
5-[3-(3-ethylphenoxy)azetidine-1-carbonyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole
(3R,4R)-1-[(5-ethylfuran-2-yl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-ol
N-{1-[(2-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-3-hydroxypyridine-2-carboxamide
6-chloro-2-{2-[4-(1-methyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]ethyl}-1H-1,3-benzodiazole
6-[2-(aminomethyl)-5-fluoro-2,3-dihydro-1-benzofuran-7-yl]-N,N-dimethylpyrazine-2-carboxamide