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1-(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidine
5-(3-acetylphenoxymethyl)-N-(1,3-dihydroxypropan-2-yl)-1H-pyrazole-3-carboxamide
6-fluoro-N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}-2-oxo-1,2-dihydroquinoline-4-carboxamide
2-(5-methyl-1,3-oxazole-4-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
1-(5-chloropyridin-2-yl)-4-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]piperazine
N-[4-({[2-(2-ethylphenoxy)ethyl](methyl)amino}methyl)phenyl]acetamide
8-(7-chloro-9-oxo-9H-fluorene-1-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
4-{4-[(2-methylphenyl)methyl]piperazin-1-yl}-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
4-[3-(3-methoxy-4-methylphenyl)propanoyl]-1-(4-methoxyphenyl)piperazin-2-one
(3R,5R)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
(2S,4S)-4-amino-N-methyl-1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]pyrrolidine-2-carboxamide
6-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-N2,N2-dimethylpyrimidine-2,4-diamine
(1S,5R)-3-(3-cyclopropyl-1,2-oxazole-5-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-fluoro-2-{[3-(2-methoxyphenoxy)azetidin-1-yl]methyl}-1-methyl-1H-indole
{2-[2-(1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperidin-4-yl)-1H-imidazol-1-yl]ethyl}dimethylamine
1-(thiophen-2-ylmethyl)-5-(2,3,6-trifluorophenyl)-1H,4H-pyrazolo[3,4-d]imidazole
N-(cyclopropylmethyl)-2-[(2S)-2-hydroxypropanoyl]-N-propyl-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
1-[(1S,5R)-6-(9H-fluorene-9-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]acetamide
N-ethyl-3-oxo-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-{1-[1-(1H-indol-3-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-phenylbutanamide
3-[(3R,4S)-1-[(4-methoxy-3-methylphenyl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
2-(2-ethoxypyridin-3-yl)-4-(3,3,3-trifluoropropyl)pyrimidine
6-(propan-2-yl)-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]-1H-indole-2-carboxamide
4-(4-{[(2,3-dimethoxyphenyl)methyl]amino}piperidin-1-yl)-N-(1-phenylethyl)benzamide
1-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
9-[2-(pyridin-2-ylsulfanyl)propanoyl]-1,4,9-triazaspiro[5.5]undecan-5-one
2-(cyclopropylmethyl)-9-(dimethyl-1,3-oxazole-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
4-[3-(pyridin-3-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]-1,2,3,4-tetrahydroquinolin-2-one
(5-{1-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-1H-1,2,3-triazol-4-yl}furan-2-yl)methanol
2-(4-chlorophenyl)-4-[3-(1H-pyrazol-1-ylmethyl)benzoyl]morpholine
3-{1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}pyridine
2-[2-(dimethylamino)ethyl]-8-(4-methyl-1H-imidazole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
5-cyclopropyl-1-{8-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-N-[3-(morpholin-4-yl)propyl]-1H-pyrazole-4-carboxamide
1-[(3-fluorophenyl)methyl]-4-{[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]amino}pyrrolidin-2-one
7-fluoro-N,2-dimethyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}quinoline-4-carboxamide
N-[(5-ethylpyridin-2-yl)methyl]-2-(2-fluorophenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
2-{3-[(2,6-dichlorophenyl)methyl]-5-[2-(1H-1,2,4-triazol-1-yl)ethyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
2-[(5-methylpyrazin-2-yl)methyl]-8-(5-methylthiophene-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
5-[({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}(methyl)amino)methyl]-N-methylpyrimidin-2-amine
2-methoxy-1-{4-[3-(pyridine-2-carbonyl)piperidine-1-carbonyl]piperidin-1-yl}ethan-1-one
ethyl 4-[1-(1,3-thiazol-2-ylmethyl)piperidin-3-yl]piperazine-1-carboxylate
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-4-(piperidin-1-ylmethyl)benzamide
2-(2-{[(4aR,8aR)-7-acetyl-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]methyl}phenoxy)acetic acid
4-[(1-{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methyl]morpholine
3-(4-benzyl-1H-pyrazol-5-yl)piperidine
4-[2-(benzyloxy)acetyl]-1-(4-methoxyphenyl)-5-methylpiperazin-2-one
1-[8-methyl-2-(1H-pyrazol-4-yl)quinoline-4-carbonyl]piperidine-4-carbonitrile
3-({[1-(dimethylcarbamoyl)ethyl](methyl)amino}methyl)-N-(2,6-dimethylphenyl)benzamide
1-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one