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(1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(hydroxymethyl)piperidin-3-yl)methanol
4-{7-methylimidazo[1,2-a]pyridin-2-yl}-N-(pyridin-2-ylmethyl)aniline
3-[2-(3-fluorophenyl)ethyl]-1-(1,3-thiazol-2-yl)piperidine
4-{6-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]pyrimidin-4-yl}morpholine
2-chloro-N-{[1-(5-phenylpentanoyl)piperidin-3-yl]methyl}benzamide
N-[(3S,4R)-4-(propan-2-yl)-1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]pyrrolidin-3-yl]methanesulfonamide
3-[({[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}amino)methyl]piperidin-3-ol
2-{[2-(furan-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}-N-methylethane-1-sulfonamide
N-(2-{7-cyclopentyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)methanesulfonamide
[5-methyl-7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
3-(3-fluorophenyl)-4-(3-methyl-1H-indole-2-carbonyl)piperazin-2-one
N,N-dimethyl-4-({spiro[indene-1,4'-piperidine]-1'-yl}carbonyl)piperidine-1-carboxamide
6-ethyl-N-[(1-methanesulfonylpiperidin-3-yl)methyl]-1,5-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
(2S)-2-amino-3-hydroxy-1-[3-(4-methylphenoxy)azetidin-1-yl]propan-1-one
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N-methylacetamide
3-chloro-N-cyclopentyl-4-({1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}oxy)benzamide
(4aR,8aR)-4-{[2-(difluoromethoxy)phenyl]methyl}-octahydro-2H-1,4-benzoxazine
3-[1-(but-2-ynoyl)piperidin-3-yl]-N-(4-methoxy-2-methylphenyl)propanamide
1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethan-1-amine
2-cyclopropyl-5-[4-(piperidine-1-carbonyl)piperidine-1-carbonyl]pyrimidine
N-(1-benzylpiperidin-4-yl)-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carboxamide
1-{5-[4-(diphenylmethyl)piperazine-1-carbonyl]-1H-pyrazol-3-yl}ethan-1-one
5-{2-[(3-fluorophenyl)methoxy]phenyl}-3-(methoxymethyl)-1H-1,2,4-triazole
2-(6-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]acetamide
6-[4-(4-methylpiperazin-1-yl)benzoyl]-N-[4-(methylsulfanyl)phenyl]-6-azaspiro[2.5]octane-1-carboxamide
1-{2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}-2-(2,2,3,3-tetrafluoropropoxy)ethan-1-one
(4aS,8aR)-1-(2-aminoethyl)-6-{[3-(furan-2-yl)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
2-amino-6-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-4-(4-hydroxyphenyl)pyridine-3-carbonitrile
(1R,3S)-7-(3-hydroxy-4-methylbenzoyl)-7-azaspiro[3.5]nonane-1,3-diol
methyl[1-(1,2-oxazol-3-yl)ethyl]{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}amine
(3R,4S)-4-cyclopropyl-1-(5-fluoro-3-methyl-1H-indole-2-carbonyl)pyrrolidin-3-amine
2-{1-cyclopentyl-4-[(4-fluoro-3-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
ethyl 2-(4-{5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carbonyl}morpholin-3-yl)acetate
1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-phenyl-5-(1-propyl-1H-imidazol-2-yl)-1H-imidazole
1-(3-methoxyphenyl)-6-methyl-4-(5-methyl-1,2-oxazole-3-carbonyl)piperazin-2-one
N-(1-cyclopentyl-1H-pyrazol-5-yl)-4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidine-1-carboxamide
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-{9-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}ethan-1-one
N-[(3S,4S)-4-methoxy-1,1-dioxo-1λ6-thiolan-3-yl]-4-oxo-4-phenylbutanamide
1-{[(2-chloro-4-fluorophenyl)carbamoyl]amino}-N-methylcyclohexane-1-carboxamide
[1-(5-{3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)piperidin-3-yl]methanol
2-[(4aR,7aS)-4-{2-[(2-methoxyethyl)(methyl)amino]acetyl}-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3-(piperidin-4-ylmethyl)benzamide
N-[3-(1H-imidazol-1-yl)propyl]-3-[(3-methylbutyl)amino]-5-(pyrrolidine-1-sulfonyl)benzamide
3-(oxolan-2-ylmethyl)-5-{1-[(2E)-3-phenylprop-2-enoyl]piperidin-4-yl}-5-(pyridin-2-yl)imidazolidine-2,4-dione
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-(1H-pyrazol-1-yl)-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)butanamide
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-6-(morpholin-4-yl)pyridine-3-carboxamide
1-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(thiophen-2-yl)propan-1-one
methyl 2-({[1-(cyclohexylmethyl)-3-hydroxy-2-oxopiperidin-3-yl]methyl}amino)acetate
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-1,4-dithiepan-6-amine