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methyl({[5-(oxan-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl})[2-(pyridin-2-yl)ethyl]amine
1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]ethan-1-one
1-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(2-methoxyphenoxy)ethan-1-one
1-[4-(benzyloxy)butanoyl]-N-cyclopropylpiperazine-2-carboxamide
8-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-6,6-dimethyl-5-oxothiomorpholine-3-carboxamide
4-{5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-1,4-oxazepane
(2S,4R)-1-[(2-chlorophenyl)methyl]-N-(propan-2-yl)-4-[(1-propylpiperidin-4-yl)amino]pyrrolidine-2-carboxamide
N-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)-5-methyl-1,3,4-oxadiazole-2-carboxamide
N-({1-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]pyrrolidin-3-yl}methyl)acetamide
(1S,5R)-6-(2-methoxyethyl)-3-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-3,6-diazabicyclo[3.2.2]nonane
N-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(1H-imidazol-2-yl)benzamide
3-(1H-1,3-benzodiazol-2-yl)-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)propanamide
5-(azepane-1-carbonyl)-1-(butan-2-yl)-4-oxo-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-1,4-dihydropyridine-3-carboxamide
1-{5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}azepane
N-[(3R,4S)-4-cyclopropyl-1-(4-methoxy-3-methylbenzenesulfonyl)pyrrolidin-3-yl]acetamide
(3R,4R)-4-(azepan-1-yl)-1-[(6-ethoxyquinolin-2-yl)methyl]piperidin-3-ol
3-({4-[3-(2-chlorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)pyridin-2-amine
3-[2-(benzyloxy)phenyl]-1-[(3R)-piperidin-3-yl]urea
2-[(8-methoxyquinolin-2-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[(3R,5S)-1-cyclopentyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]-1-ethyl-1H-pyrazole-5-carboxamide
1-{4-[1-(4-methylphenyl)-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]piperidin-1-yl}ethan-1-one
N-[(1R,3R)-3-aminocyclopentyl]-4-[(diethylamino)methyl]-5-ethylfuran-2-carboxamide
1-(4-cyclopentylpyrimidin-2-yl)-4-(pyridin-4-ylmethyl)-1,4-diazepane
3-[5-(2-cyclohexylethyl)-1,3,4-oxadiazol-2-yl]-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}propanamide
[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]({[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
7-(2-methoxyacetamido)-N-[(5-methylpyrazin-2-yl)methyl]-1-(2-phenylethyl)-1H-1,3-benzodiazole-5-carboxamide
N-(oxan-4-yl)-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
4-[4-(piperidine-1-carbonyl)phenoxy]-1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidine
(3S,4R)-4-methyl-1-{4-[(pyridin-2-ylsulfanyl)methyl]benzoyl}piperidine-3,4-diol
2-[3-cyclopropyl-1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]-3-fluoropyridine
2-(7-fluoro-2-methyl-1H-indol-3-yl)-1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
2-ethyl-N-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}pyrimidine-5-carboxamide
7-[(3,4-difluorophenyl)methyl]-2-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
5-(4-fluoropiperidine-1-carbonyl)-2-(pyridin-4-yl)pyrimidine
2-amino-1-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}ethan-1-one
(3R,4R)-1-{[3-(methylsulfanyl)phenyl]methyl}-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
3-[2-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)ethyl]-2,3-dihydro-1,3-benzoxazol-2-one
3-hydroxy-3-[({imidazo[1,2-a]pyridin-2-ylmethyl}amino)methyl]-1-[(3-methoxyphenyl)methyl]piperidin-2-one
5-(4-carbamoylpiperidin-1-yl)-N-methyl-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-(dimethyl-1,2-oxazol-4-yl)-3-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyloxolane-3-carboxamide
N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)furan-2-carboxamide
N-{2-[(dimethylcarbamoyl)methyl]phenyl}-2-(3-methoxyphenyl)pyrrolidine-1-carboxamide
4-(furan-2-ylmethyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(1-ethyl-5-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-(4-methyl-1H-imidazole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-[(2-chlorophenyl)methyl]-4-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]morpholine
N-[2-(2-chloro-6-methylphenoxy)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
1-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(1H-pyrazol-1-yl)propan-1-one