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(2E)-N-[1-(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)-2-phenylethyl]-3-(4-methoxyphenyl)prop-2-enamide
[(1R,3S,3aS,6aR)-3-(4-methoxy-2,5-dimethylphenyl)-5-phenyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
8-[(6-methoxy-2H-chromen-3-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
6-methyl-2-{[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]methyl}pyridin-3-ol
2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N-(3-methoxypropyl)acetamide
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-1-(2-methoxyacetyl)piperidine-3-carboxamide
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2-(1H-pyrazol-1-yl)butanamide
1-{3-[3-(1-ethyl-1H-pyrazol-4-yl)-4H-1,2,4-triazol-4-yl]phenyl}ethan-1-one
1-(3-acetylphenoxy)cyclohexane-1-carboxylic acid
N-cyclopropyl-N-{[2-(2,5-dimethoxyphenyl)-8-methylquinolin-3-yl]methyl}-3-(2-methoxyphenyl)propanamide
4-hydroxy-4-(5-methylpyridin-2-yl)-N-[3-(4H-1,2,4-triazol-4-yl)phenyl]piperidine-1-carboxamide
N-cyclopropyl-4-{[(8-methoxyquinolin-5-yl)methyl](methyl)amino}pyridine-2-carboxamide
1-(2-cyclobutylacetyl)-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
3-(1-methyl-1H-pyrazol-4-yl)-N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}propanamide
4-benzyl-1-methyl-3-[1-(2-methylpentanoyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[2-(4-fluorophenyl)morpholin-4-yl]-6-methylpyrimidin-2-amine
7-[(2,3-dimethoxyphenyl)methyl]-2-(2-methylpropyl)-2,7-diazaspiro[4.5]decane
(2S,4S)-4-acetamido-N-ethyl-1-{[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl}pyrrolidine-2-carboxamide
1-[2-(trifluoromethyl)morpholin-4-yl]-2-(4,6,7-trimethyl-1-benzofuran-3-yl)ethan-1-one
N-[(2-aminopyrimidin-5-yl)methyl]-4-(4-chlorophenyl)-N-methylbutanamide
N-(2-{1-[(2-cyanophenyl)methyl]piperidin-3-yl}ethyl)-2,2-dimethylpropanamide
methyl 3-{6-chloroimidazo[1,2-a]pyridine-2-amido}azepane-1-carboxylate
2-methyl-4-(4-{[methyl(1H-pyrazol-3-ylmethyl)amino]methyl}phenyl)butan-2-ol
(1S,6R)-9-[(6-methyl-4-oxo-4H-chromen-3-yl)methyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
2-(2H-1,2,3-benzotriazol-2-yl)-1-(6-hydroxy-4-methyl-1,4-diazepan-1-yl)ethan-1-one
(3S,4R)-1-(3,5-di-tert-butyl-4-hydroxybenzoyl)-4-methylpiperidine-3,4-diol
N-[(1-{[3-(pyridin-2-ylmethoxy)phenyl]methyl}piperidin-4-yl)methyl]acetamide
{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]methylamine
1-methyl-3-[1-(3-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(2R)-2-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-2-phenylethan-1-ol
(1S,4S)-2-(5-chloro-2-methoxyphenyl)-5-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}-2,5-diazabicyclo[2.2.1]heptan-3-one
2-methyl-5-{[4-(2,3,4-trimethoxyphenyl)-1H-1,2,3-triazol-1-yl]methyl}pyrazine
(3S,4S)-4-(naphthalen-2-yl)-1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-3-ol
N-[3-(dimethylamino)propyl]-5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-amine
3-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-3-yl]-N-(4-fluoro-2-methylphenyl)propanamide
1-{1-[5-(4-methoxyphenyl)furan-2-carbonyl]piperidin-4-yl}-2-(oxolan-2-yl)-5-(trifluoromethyl)-1H-1,3-benzodiazole
4-(5-methyl-2-oxo-4-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperazin-1-yl)benzonitrile
3-(1-methyl-1H-pyrrol-2-yl)-N-[1-(pyrimidin-2-yl)piperidin-3-yl]-1H-pyrazole-5-carboxamide
N-cyclopropyl-N-[(2-methoxyphenyl)methyl]-2-(pyridin-2-ylsulfanyl)propanamide
4-{1-ethyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-5-methyl-1-phenyl-1H-pyrazole
N-{[7-(5-chloro-3-methyl-1H-indole-2-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}thiophene-3-carboxamide
8-fluoro-2-{1-[1-(1H-pyrazol-1-yl)propan-2-yl]-1H-imidazol-2-yl}quinoline
1-{2,7-dimethylimidazo[1,2-a]pyridine-3-carbonyl}-4-(2-methanesulfonylethyl)piperazine
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-ethyl-1-(propan-2-yl)-4-[6-(pyrrolidin-1-yl)pyridine-3-carbonyl]piperazine
4-[1-(1-{[4-(trifluoromethyl)phenyl]methyl}piperidin-3-yl)-1H-1,2,3-triazole-4-carbonyl]morpholine
1-{[(3R,4R)-4-(hydroxymethyl)-1-{6-methylthieno[2,3-d]pyrimidin-4-yl}pyrrolidin-3-yl]methyl}piperidin-4-ol
1-[1-(6-{[(1-ethylcyclopropyl)methyl]amino}pyridine-3-carbonyl)piperidin-3-yl]-3-methylbutan-1-one
N-methyl-2-[methyl(pyridin-3-ylmethyl)amino]-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]acetamide
5-ethyl-2,3-dimethyl-N-(1,2-oxazol-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine